JP2528883B2 - ミルベマイシン誘導体、その製法、および有害生物防除剤 - Google Patents

ミルベマイシン誘導体、その製法、および有害生物防除剤

Info

Publication number
JP2528883B2
JP2528883B2 JP62164112A JP16411287A JP2528883B2 JP 2528883 B2 JP2528883 B2 JP 2528883B2 JP 62164112 A JP62164112 A JP 62164112A JP 16411287 A JP16411287 A JP 16411287A JP 2528883 B2 JP2528883 B2 JP 2528883B2
Authority
JP
Japan
Prior art keywords
milbemycin
formula
substituted
tert
unsubstituted
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
JP62164112A
Other languages
English (en)
Japanese (ja)
Other versions
JPS6333381A (ja
Inventor
コーネリアス オサリバン アンソニー
フライ ブルノ
Original Assignee
チバ−ガイギ− アクチエンゲゼルシヤフト
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by チバ−ガイギ− アクチエンゲゼルシヤフト filed Critical チバ−ガイギ− アクチエンゲゼルシヤフト
Publication of JPS6333381A publication Critical patent/JPS6333381A/ja
Application granted granted Critical
Publication of JP2528883B2 publication Critical patent/JP2528883B2/ja
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D493/00Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
    • C07D493/22Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains four or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/01Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing oxygen
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N53/00Biocides, pest repellants or attractants, or plant growth regulators containing cyclopropane carboxylic acids or derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/10Anthelmintics

Landscapes

  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Plant Pathology (AREA)
  • Veterinary Medicine (AREA)
  • Environmental Sciences (AREA)
  • Zoology (AREA)
  • Wood Science & Technology (AREA)
  • Dentistry (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Public Health (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biochemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
JP62164112A 1986-07-02 1987-07-02 ミルベマイシン誘導体、その製法、および有害生物防除剤 Expired - Lifetime JP2528883B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
CH02668/86-5 1986-07-02
CH2668/86-5 1986-07-02
CH266886 1986-07-02

Publications (2)

Publication Number Publication Date
JPS6333381A JPS6333381A (ja) 1988-02-13
JP2528883B2 true JP2528883B2 (ja) 1996-08-28

Family

ID=4238883

Family Applications (1)

Application Number Title Priority Date Filing Date
JP62164112A Expired - Lifetime JP2528883B2 (ja) 1986-07-02 1987-07-02 ミルベマイシン誘導体、その製法、および有害生物防除剤

Country Status (11)

Country Link
US (1) US4859657A (2)
EP (1) EP0252879B1 (2)
JP (1) JP2528883B2 (2)
KR (1) KR960001480B1 (2)
AT (1) ATE75745T1 (2)
DE (1) DE3778768D1 (2)
DK (1) DK338187A (2)
ES (1) ES2039258T3 (2)
GR (1) GR3004535T3 (2)
IL (1) IL83031A0 (2)
ZA (1) ZA874752B (2)

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WO2000059298A1 (en) * 1999-04-02 2000-10-12 Chung Kwang Suk Multi purpose fish-hook case including fishline binding device
US6787342B2 (en) 2000-02-16 2004-09-07 Merial Limited Paste formulations
US20060205681A1 (en) * 2002-06-21 2006-09-14 Maryam Moaddeb Homogenous paste formulations
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US20080027011A1 (en) * 2005-12-20 2008-01-31 Hassan Nached Homogeneous paste and gel formulations
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RS54772B1 (sr) 2009-12-17 2016-10-31 Merial Sas Antiparazitska jedinjenja dihidroazola i kompozicije koje ih sadrže
BR112012014933B1 (pt) 2009-12-17 2020-10-27 Merial, Inc. composições que compreendem compostos lactonas macrocíclicas e spirodioxepinoindóis
UA108641C2 (uk) 2010-04-02 2015-05-25 Паразитицидна композиція, яка містить чотири активних агенти, та спосіб її застосування
EP2568980B1 (en) 2010-05-12 2015-11-11 Merial, Inc. Injectable parasiticidal formulations of levamisole and macrocyclic lactones
US8822528B2 (en) 2010-11-16 2014-09-02 Merial Limited Monensin derivatives for the treatment and prevention of protozoal infections
WO2012078605A1 (en) 2010-12-07 2012-06-14 Merial Limited Topical combination formulations of macrocyclic lactones with synthetic pyrethroids
US20120329832A1 (en) 2011-06-27 2012-12-27 Jean Delaveau Novel Insect-Repellent Coumarin Derivatives, Syntheses, and Methods of Use
ES2618813T3 (es) 2011-06-27 2017-06-22 Merial, Inc. Compuestos y composiciones de éter amido-piridílico y uso contra los parásitos
RS58417B1 (sr) 2011-09-12 2019-04-30 Merial Inc Paraziticidne kompozicije koje sadrže izoksazolinsko aktivno sredstvo, postupci i upotrebe povezane sa njima
WO2013044118A2 (en) 2011-09-23 2013-03-28 Merial Limited Indirect modeling of new repellent molecules active against insects, acarids, and other arthropods
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US10864193B2 (en) 2014-10-31 2020-12-15 Boehringer Ingelheim Animal Health USA Inc. Parasiticidal compositions comprising fipronil at high concentrations
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Also Published As

Publication number Publication date
DK338187A (da) 1988-01-03
EP0252879B1 (de) 1992-05-06
US4859657A (en) 1989-08-22
JPS6333381A (ja) 1988-02-13
KR880001661A (ko) 1988-04-26
GR3004535T3 (2) 1993-04-28
EP0252879A1 (de) 1988-01-13
ZA874752B (en) 1988-01-04
ATE75745T1 (de) 1992-05-15
DE3778768D1 (de) 1992-06-11
KR960001480B1 (ko) 1996-01-31
DK338187D0 (da) 1987-07-01
IL83031A0 (en) 1987-12-20
ES2039258T3 (es) 1993-09-16

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