JP2025511255A5 - - Google Patents

Info

Publication number
JP2025511255A5
JP2025511255A5 JP2024558178A JP2024558178A JP2025511255A5 JP 2025511255 A5 JP2025511255 A5 JP 2025511255A5 JP 2024558178 A JP2024558178 A JP 2024558178A JP 2024558178 A JP2024558178 A JP 2024558178A JP 2025511255 A5 JP2025511255 A5 JP 2025511255A5
Authority
JP
Japan
Prior art keywords
hydrogen
cyclopropane
carboxamide
halo
difluoro
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2024558178A
Other languages
English (en)
Japanese (ja)
Other versions
JP2025511255A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/IB2023/053132 external-priority patent/WO2023187677A1/en
Publication of JP2025511255A publication Critical patent/JP2025511255A/ja
Publication of JP2025511255A5 publication Critical patent/JP2025511255A5/ja
Pending legal-status Critical Current

Links

JP2024558178A 2022-03-30 2023-03-29 N-(ピロリジン-3-イルまたはピペリジン-4-イル)アセトアミド誘導体 Pending JP2025511255A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202263325452P 2022-03-30 2022-03-30
US63/325,452 2022-03-30
PCT/IB2023/053132 WO2023187677A1 (en) 2022-03-30 2023-03-29 N-(pyrrolidin-3-yl or piperidin-4-yl)acetamide derivatives

Publications (2)

Publication Number Publication Date
JP2025511255A JP2025511255A (ja) 2025-04-15
JP2025511255A5 true JP2025511255A5 (https=) 2026-04-06

Family

ID=86054310

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2024558178A Pending JP2025511255A (ja) 2022-03-30 2023-03-29 N-(ピロリジン-3-イルまたはピペリジン-4-イル)アセトアミド誘導体

Country Status (15)

Country Link
US (1) US20250188037A1 (https=)
EP (1) EP4499224A1 (https=)
JP (1) JP2025511255A (https=)
KR (1) KR20240169050A (https=)
CN (1) CN119585238A (https=)
AR (1) AR128930A1 (https=)
AU (1) AU2023247317A1 (https=)
CA (1) CA3255222A1 (https=)
CL (1) CL2024002937A1 (https=)
CO (1) CO2024014680A2 (https=)
IL (1) IL315998A (https=)
MX (1) MX2024011914A (https=)
PE (1) PE20250749A1 (https=)
TW (1) TW202402735A (https=)
WO (1) WO2023187677A1 (https=)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR121683A1 (es) * 2020-03-31 2022-06-29 Takeda Pharmaceuticals Co Derivados de n-heteroarilalquil-2-(heterociclil y heterociclilmetil)acetamida como agonistas de sstr4
WO2025074305A1 (en) * 2023-10-04 2025-04-10 Takeda Pharmaceutical Company Limited N-(1-(aminomethyl)cyclopropyl)(aryl or heteroaryl) carboxamide derivatives
WO2025247982A1 (en) 2024-05-29 2025-12-04 Grünenthal GmbH Piperazines which act as sstr4 modulators

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR0166088B1 (ko) 1990-01-23 1999-01-15 . 수용해도가 증가된 시클로덱스트린 유도체 및 이의 용도
US5376645A (en) 1990-01-23 1994-12-27 University Of Kansas Derivatives of cyclodextrins exhibiting enhanced aqueous solubility and the use thereof
GB9518953D0 (en) 1995-09-15 1995-11-15 Pfizer Ltd Pharmaceutical formulations
GB9711643D0 (en) 1997-06-05 1997-07-30 Janssen Pharmaceutica Nv Glass thermoplastic systems
TWI834637B (zh) * 2018-03-01 2024-03-11 日商武田藥品工業有限公司 六氫吡啶基-3-(芳氧基)丙醯胺及丙酸酯

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