JP2025507543A5 - - Google Patents

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Publication number
JP2025507543A5
JP2025507543A5 JP2024547297A JP2024547297A JP2025507543A5 JP 2025507543 A5 JP2025507543 A5 JP 2025507543A5 JP 2024547297 A JP2024547297 A JP 2024547297A JP 2024547297 A JP2024547297 A JP 2024547297A JP 2025507543 A5 JP2025507543 A5 JP 2025507543A5
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JP
Japan
Prior art keywords
optionally substituted
alkyl
disorder
cycloalkyl
pharmaceutically acceptable
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2024547297A
Other languages
English (en)
Japanese (ja)
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JP2025507543A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2023/063113 external-priority patent/WO2023164537A1/en
Publication of JP2025507543A publication Critical patent/JP2025507543A/ja
Publication of JP2025507543A5 publication Critical patent/JP2025507543A5/ja
Pending legal-status Critical Current

Links

JP2024547297A 2022-02-23 2023-02-23 Kv7チャネル活性化剤としてのピラゾリル化合物 Pending JP2025507543A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202263313212P 2022-02-23 2022-02-23
US63/313,212 2022-02-23
PCT/US2023/063113 WO2023164537A1 (en) 2022-02-23 2023-02-23 Pyrazolyl compounds as kv7 channel activators

Publications (2)

Publication Number Publication Date
JP2025507543A JP2025507543A (ja) 2025-03-21
JP2025507543A5 true JP2025507543A5 (enExample) 2025-11-19

Family

ID=87766732

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2024547297A Pending JP2025507543A (ja) 2022-02-23 2023-02-23 Kv7チャネル活性化剤としてのピラゾリル化合物

Country Status (10)

Country Link
US (1) US20250171430A1 (enExample)
EP (1) EP4482486A4 (enExample)
JP (1) JP2025507543A (enExample)
KR (1) KR20240150500A (enExample)
CN (1) CN118678954A (enExample)
AU (1) AU2023225967A1 (enExample)
CA (1) CA3244850A1 (enExample)
IL (1) IL314555A (enExample)
MX (1) MX2024010081A (enExample)
WO (1) WO2023164537A1 (enExample)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW202528310A (zh) * 2023-09-20 2025-07-16 美商深蘋果治療股份有限公司 經取代胺化合物,組合物及使用方法

Family Cites Families (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3098075A (en) * 1956-02-10 1963-07-16 Ciba Geigy Corp New pyrazolo-pyrimidines
ATE410161T1 (de) * 2003-05-02 2008-10-15 Elan Pharm Inc 4-bromo-5-(2-chloro-benzoylamino)-1h-pyrazol-3- carbonsäureamid-derivate und verwandte verbindungen als bradykinin b1 rezeptor antagonisten zur behandlung von entzündlichen erkrankungen
ES2351274T3 (es) * 2007-06-06 2011-02-02 Torrent Pharmaceuticals Ltd Nuevos compuestos.
UA110324C2 (en) * 2009-07-02 2015-12-25 Genentech Inc Jak inhibitory compounds based on pyrazolo pyrimidine
CN103619171B (zh) * 2010-11-03 2015-11-25 陶氏益农公司 杀虫组合物和与其相关的方法
US9067894B1 (en) * 2013-03-07 2015-06-30 Vanderbilt University Compound, composition, and method of activating GIRK potassium channel and use of same for treating conditions of interest
CN107406380B (zh) * 2015-02-04 2020-04-28 上海海雁医药科技有限公司 杂环取代的n-磺酰基苯甲酰胺衍生物、其制法与医药上的用途
WO2016164703A1 (en) * 2015-04-09 2016-10-13 Eisai R & D Management Co., Ltd. Fgfr4 inhibitors
EP3558992A4 (en) * 2016-12-15 2020-12-02 ONO Pharmaceutical Co., Ltd. TREK CHANNEL ACTIVATOR (K + CHANNELS ASSOCIATED WITH TWIK)
CN114127058B (zh) * 2019-07-04 2024-06-25 深圳国顺康医药科技有限公司 一种杂环化合物、其药物组合物及用途
CN110627725B (zh) * 2019-10-14 2022-10-18 遵义医科大学 一种4-取代5-二氟甲基-3-硝基-1h-吡唑类化合物及其制备方法与应用
JP2021121582A (ja) * 2020-01-31 2021-08-26 クミアイ化学工業株式会社 5−(ピラゾール−5−イル)安息香酸アミド誘導体及び有害生物防除剤
EP4482487A4 (en) * 2022-02-23 2026-04-15 Biohaven Therapeutics Ltd PYRAZOLYL COMPOUNDS USED AS KV7 CHANNEL ACTIVATORS
CN118695860A (zh) * 2022-02-23 2024-09-24 拜奥海芬治疗学有限公司 作为kv7通道激活剂的吡唑基化合物

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