JP2025505994A5 - - Google Patents

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Publication number
JP2025505994A5
JP2025505994A5 JP2024546072A JP2024546072A JP2025505994A5 JP 2025505994 A5 JP2025505994 A5 JP 2025505994A5 JP 2024546072 A JP2024546072 A JP 2024546072A JP 2024546072 A JP2024546072 A JP 2024546072A JP 2025505994 A5 JP2025505994 A5 JP 2025505994A5
Authority
JP
Japan
Prior art keywords
alkyl
cycloalkyl
heterocycloalkyl
heteroaryl
aryl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2024546072A
Other languages
English (en)
Japanese (ja)
Other versions
JP2025505994A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2023/012092 external-priority patent/WO2023150150A1/en
Publication of JP2025505994A publication Critical patent/JP2025505994A/ja
Publication of JP2025505994A5 publication Critical patent/JP2025505994A5/ja
Pending legal-status Critical Current

Links

JP2024546072A 2022-02-02 2023-02-01 プロテインチロシンホスファターゼ阻害剤およびその使用 Pending JP2025505994A (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US202263305788P 2022-02-02 2022-02-02
US202263305783P 2022-02-02 2022-02-02
US63/305,788 2022-02-02
US63/305,783 2022-02-02
PCT/US2023/012092 WO2023150150A1 (en) 2022-02-02 2023-02-01 Protein tyrosine phosphatase inhibitors and uses thereof

Publications (2)

Publication Number Publication Date
JP2025505994A JP2025505994A (ja) 2025-03-05
JP2025505994A5 true JP2025505994A5 (https=) 2026-02-09

Family

ID=87552845

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2024546072A Pending JP2025505994A (ja) 2022-02-02 2023-02-01 プロテインチロシンホスファターゼ阻害剤およびその使用

Country Status (4)

Country Link
US (1) US20250134882A1 (https=)
EP (1) EP4472957A4 (https=)
JP (1) JP2025505994A (https=)
WO (1) WO2023150150A1 (https=)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PE20250780A1 (es) * 2022-02-02 2025-03-14 Nerio Therapeutics Inc Inhibidores de proteina tirosina fosfatasa y usos de estos
KR20250090365A (ko) * 2022-11-09 2025-06-19 브리스톨-마이어스 스큅 컴퍼니 암 질환의 치료를 위한 단백질 티로신 포스파타제 (ptpn2)의 억제제로서의 인다졸 치환된 1,2,5-티아디아졸리딘 유도체
WO2024141015A1 (en) * 2022-12-30 2024-07-04 Insilico Medicine Ip Limited Protein tyrosine phosphatase inhibitors and uses thereof
PE20252789A1 (es) 2023-05-24 2025-12-22 Kumquat Biosciences Inc Compuestos heterociclicos y usos de estos
AU2024288616A1 (en) * 2023-07-11 2026-02-12 Shenzhen Zhongge Biological Technology Co., Ltd. Protein tyrosine phosphatase inhibitor, composition comprising same, and medical use thereof
CN121889379A (zh) * 2023-09-15 2026-04-17 深圳众格生物科技有限公司 蛋白酪氨酸磷酸酶抑制剂及其组合物、医药用途
CN120004876B (zh) * 2023-11-16 2026-02-06 英矽智能科技(上海)有限公司 蛋白酪氨酸磷酸酶抑制剂及其应用
CN117343052B (zh) * 2023-12-04 2024-02-06 英矽智能科技(上海)有限公司 蛋白酪氨酸磷酸酶抑制剂及其应用
WO2025242216A1 (zh) * 2024-05-24 2025-11-27 杭州百新生物医药科技有限公司 吲哚啉类化合物及其用途

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
UA94921C2 (en) * 2005-12-08 2011-06-25 Новартис Аг 1-orthofluorophenyl substituted 1, 2, 5-thiazolidinedione derivatives as ptp-as inhibitors
UA94724C2 (en) * 2005-12-08 2011-06-10 Новартис Аг Thiadiazolidinone derivatives as antidiabetic agents
KR20150118158A (ko) * 2013-02-22 2015-10-21 머크 샤프 앤드 돔 코포레이션 항당뇨병 비시클릭 화합물
IL286373B2 (en) * 2019-03-14 2026-03-01 Calico Life Sciences Llc Protein tyrosine phosphate inhibitor compounds and uses thereof
MX2023002953A (es) * 2020-09-11 2023-06-01 Calico Life Sciences Llc Inhibidores de proteína tirosina fosfatasa y métodos para su uso.
WO2022192598A1 (en) * 2021-03-11 2022-09-15 Kumquat Biosciences Inc. Heterocycles and uses thereof

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