JP2024542248A5 - - Google Patents

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Publication number
JP2024542248A5
JP2024542248A5 JP2024530029A JP2024530029A JP2024542248A5 JP 2024542248 A5 JP2024542248 A5 JP 2024542248A5 JP 2024530029 A JP2024530029 A JP 2024530029A JP 2024530029 A JP2024530029 A JP 2024530029A JP 2024542248 A5 JP2024542248 A5 JP 2024542248A5
Authority
JP
Japan
Prior art keywords
fluoro
quinoline
methyl
azabicyclo
hexane
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2024530029A
Other languages
English (en)
Japanese (ja)
Other versions
JP2024542248A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2022/050558 external-priority patent/WO2023091746A1/en
Publication of JP2024542248A publication Critical patent/JP2024542248A/ja
Publication of JP2024542248A5 publication Critical patent/JP2024542248A5/ja
Pending legal-status Critical Current

Links

JP2024530029A 2021-11-22 2022-11-21 Fgfr阻害剤とkras阻害剤を含む併用療法 Pending JP2024542248A (ja)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US202163282017P 2021-11-22 2021-11-22
US63/282,017 2021-11-22
US202263317654P 2022-03-08 2022-03-08
US63/317,654 2022-03-08
US202263352491P 2022-06-15 2022-06-15
US63/352,491 2022-06-15
PCT/US2022/050558 WO2023091746A1 (en) 2021-11-22 2022-11-21 Combination therapy comprising an fgfr inhibitor and a kras inhibitor

Publications (2)

Publication Number Publication Date
JP2024542248A JP2024542248A (ja) 2024-11-13
JP2024542248A5 true JP2024542248A5 (https=) 2025-12-03

Family

ID=84901810

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2024530029A Pending JP2024542248A (ja) 2021-11-22 2022-11-21 Fgfr阻害剤とkras阻害剤を含む併用療法

Country Status (11)

Country Link
US (1) US20230226040A1 (https=)
EP (1) EP4436578A1 (https=)
JP (1) JP2024542248A (https=)
KR (1) KR20240122783A (https=)
AU (1) AU2022389961A1 (https=)
CA (1) CA3239205A1 (https=)
CL (1) CL2024001523A1 (https=)
IL (1) IL312886A (https=)
MX (1) MX2024006113A (https=)
TW (1) TW202320792A (https=)
WO (1) WO2023091746A1 (https=)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MX2024000357A (es) * 2021-07-07 2024-02-12 Incyte Corp Compuestos triciclicos como inhibidores de homologo de oncogen viral de sarcoma de rata kirsten (kras).
US20240101557A1 (en) * 2022-07-11 2024-03-28 Incyte Corporation Fused tricyclic compounds as inhibitors of kras g12v mutants
US20250114346A1 (en) * 2023-10-09 2025-04-10 Incyte Corporation Combination therapy using a kras g12d inhibitor and pd-1 inhibitor or pd-l1 inhibitor

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