JP2024542212A5 - - Google Patents

Info

Publication number
JP2024542212A5
JP2024542212A5 JP2024529599A JP2024529599A JP2024542212A5 JP 2024542212 A5 JP2024542212 A5 JP 2024542212A5 JP 2024529599 A JP2024529599 A JP 2024529599A JP 2024529599 A JP2024529599 A JP 2024529599A JP 2024542212 A5 JP2024542212 A5 JP 2024542212A5
Authority
JP
Japan
Prior art keywords
pharmaceutically acceptable
acceptable salt
compound according
cancer
alkyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2024529599A
Other languages
English (en)
Japanese (ja)
Other versions
JP2024542212A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2022/079973 external-priority patent/WO2023091957A1/en
Publication of JP2024542212A publication Critical patent/JP2024542212A/ja
Publication of JP2024542212A5 publication Critical patent/JP2024542212A5/ja
Pending legal-status Critical Current

Links

JP2024529599A 2021-11-17 2022-11-16 治療薬としてのペプチドチューブリン阻害剤のペプチドコンジュゲート Pending JP2024542212A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202163280409P 2021-11-17 2021-11-17
US63/280,409 2021-11-17
PCT/US2022/079973 WO2023091957A1 (en) 2021-11-17 2022-11-16 Peptide conjugates of peptidic tubulin inhibitors as therapeutics

Publications (2)

Publication Number Publication Date
JP2024542212A JP2024542212A (ja) 2024-11-13
JP2024542212A5 true JP2024542212A5 (enExample) 2025-11-25

Family

ID=84799580

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2024529599A Pending JP2024542212A (ja) 2021-11-17 2022-11-16 治療薬としてのペプチドチューブリン阻害剤のペプチドコンジュゲート

Country Status (14)

Country Link
US (1) US20230416331A1 (enExample)
EP (1) EP4433095A1 (enExample)
JP (1) JP2024542212A (enExample)
KR (1) KR20240130157A (enExample)
CN (1) CN118574642A (enExample)
AU (1) AU2022390891A1 (enExample)
CA (1) CA3243300A1 (enExample)
CL (1) CL2024001486A1 (enExample)
CO (1) CO2024007413A2 (enExample)
IL (1) IL312884A (enExample)
MX (1) MX2024005938A (enExample)
PE (1) PE20242180A1 (enExample)
TW (1) TW202330015A (enExample)
WO (1) WO2023091957A1 (enExample)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR20220052918A (ko) 2019-07-10 2022-04-28 싸이브렉사 2, 인크. 치료제로서의 사이토톡신의 펩티드 접합체
PH12022550037A1 (en) 2019-07-10 2023-04-12 Cybrexa 3 Inc Peptide conjugates of microtubule-targeting agents as therapeutics

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2399267T3 (es) * 2005-01-18 2013-03-27 The Board Of Governors For Higher Education State Of Rhode Island And Providence Plantations Suministro selectivo de moléculas al interior de las células o marcación de células en zonas enfermas de tejidos usando un péptido transmembrana sensible a su entorno
JP6262768B2 (ja) * 2013-01-03 2018-01-17 セルトリオン, インク. 抗体−リンカー−薬物結合体、その製造方法およびそれを含む抗癌剤組成物
WO2018023098A1 (en) * 2016-07-29 2018-02-01 Memorial Sloan Kettering Cancer Center Radiolabeled ligands for targeted pet/spect imaging and methods of their use
KR20220052918A (ko) * 2019-07-10 2022-04-28 싸이브렉사 2, 인크. 치료제로서의 사이토톡신의 펩티드 접합체
PH12022550037A1 (en) * 2019-07-10 2023-04-12 Cybrexa 3 Inc Peptide conjugates of microtubule-targeting agents as therapeutics

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