JP2024535343A5 - - Google Patents
Info
- Publication number
- JP2024535343A5 JP2024535343A5 JP2024518302A JP2024518302A JP2024535343A5 JP 2024535343 A5 JP2024535343 A5 JP 2024535343A5 JP 2024518302 A JP2024518302 A JP 2024518302A JP 2024518302 A JP2024518302 A JP 2024518302A JP 2024535343 A5 JP2024535343 A5 JP 2024535343A5
- Authority
- JP
- Japan
- Prior art keywords
- chloro
- methyl
- tetradeca
- difluorophenyl
- trifluoromethyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP21198735 | 2021-09-24 | ||
| EP21198735.9 | 2021-09-24 | ||
| PCT/EP2022/076467 WO2023046877A1 (en) | 2021-09-24 | 2022-09-23 | Pyrido diazepine derivatives as gaba a gamma1 pam |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2024535343A JP2024535343A (ja) | 2024-09-30 |
| JP2024535343A5 true JP2024535343A5 (enExample) | 2025-10-01 |
| JP7899312B2 JP7899312B2 (ja) | 2026-08-03 |
Family
ID=77924305
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2024518302A Active JP7899312B2 (ja) | 2021-09-24 | 2022-09-23 | GABAAγ1 PAMとしてのピリドジアゼピン誘導体 |
Country Status (11)
| Country | Link |
|---|---|
| US (2) | US20230109111A1 (enExample) |
| EP (1) | EP4405356A1 (enExample) |
| JP (1) | JP7899312B2 (enExample) |
| KR (1) | KR20240065086A (enExample) |
| CN (1) | CN117957227A (enExample) |
| AR (1) | AR127127A1 (enExample) |
| AU (1) | AU2022351080A1 (enExample) |
| CA (1) | CA3229125A1 (enExample) |
| IL (1) | IL310444A (enExample) |
| TW (1) | TW202322804A (enExample) |
| WO (1) | WO2023046877A1 (enExample) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TWI878507B (zh) | 2020-03-31 | 2025-04-01 | 瑞士商赫孚孟拉羅股份公司 | 作為 GABA A γ1 PAM 的新穎苯并二氮呯衍生物 |
| JP2024537773A (ja) | 2021-09-29 | 2024-10-16 | エフ. ホフマン-ラ ロシュ アーゲー | GABA Aγ1 PAMとしての新規ベンゾジアゼピン誘導体 |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA1185601A (en) * | 1981-02-27 | 1985-04-16 | Walter Hunkeler | Imidazodiazepines |
| WO2003082832A2 (en) * | 2002-03-28 | 2003-10-09 | Wisys Technology Foundation, Inc. | Anxiolytic agents with reduced sedative and ataxic effects |
| JP2012087069A (ja) * | 2010-10-15 | 2012-05-10 | Osaka Prefecture Univ | 1,4−ベンゾジアゼピン誘導体の製造方法および該誘導体 |
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2022
- 2022-09-22 AR ARP220102559A patent/AR127127A1/es not_active Application Discontinuation
- 2022-09-23 IL IL310444A patent/IL310444A/en unknown
- 2022-09-23 AU AU2022351080A patent/AU2022351080A1/en active Pending
- 2022-09-23 WO PCT/EP2022/076467 patent/WO2023046877A1/en not_active Ceased
- 2022-09-23 EP EP22793720.8A patent/EP4405356A1/en active Pending
- 2022-09-23 KR KR1020247008988A patent/KR20240065086A/ko active Pending
- 2022-09-23 CA CA3229125A patent/CA3229125A1/en active Pending
- 2022-09-23 US US17/934,769 patent/US20230109111A1/en not_active Abandoned
- 2022-09-23 CN CN202280062998.0A patent/CN117957227A/zh active Pending
- 2022-09-23 JP JP2024518302A patent/JP7899312B2/ja active Active
- 2022-09-23 TW TW111136044A patent/TW202322804A/zh unknown
-
2024
- 2024-02-14 US US18/441,558 patent/US20240270744A1/en active Pending