JP2024534840A5 - - Google Patents

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Publication number
JP2024534840A5
JP2024534840A5 JP2024513015A JP2024513015A JP2024534840A5 JP 2024534840 A5 JP2024534840 A5 JP 2024534840A5 JP 2024513015 A JP2024513015 A JP 2024513015A JP 2024513015 A JP2024513015 A JP 2024513015A JP 2024534840 A5 JP2024534840 A5 JP 2024534840A5
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JP
Japan
Prior art keywords
alkyl
group
cycloalkyl
ring
pharmaceutically acceptable
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Pending
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JP2024513015A
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English (en)
Japanese (ja)
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JP2024534840A (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/US2022/075472 external-priority patent/WO2023028564A1/en
Publication of JP2024534840A publication Critical patent/JP2024534840A/ja
Publication of JP2024534840A5 publication Critical patent/JP2024534840A5/ja
Pending legal-status Critical Current

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JP2024513015A 2021-08-26 2022-08-25 Kif18aのスピロインドリン阻害剤 Pending JP2024534840A (ja)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US202163237275P 2021-08-26 2021-08-26
US63/237,275 2021-08-26
US202263306452P 2022-02-03 2022-02-03
US63/306,452 2022-02-03
US202263344435P 2022-05-20 2022-05-20
US63/344,435 2022-05-20
PCT/US2022/075472 WO2023028564A1 (en) 2021-08-26 2022-08-25 Spiro indoline inhibitors of kif18a

Publications (2)

Publication Number Publication Date
JP2024534840A JP2024534840A (ja) 2024-09-26
JP2024534840A5 true JP2024534840A5 (enExample) 2025-08-26

Family

ID=83457176

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2024513015A Pending JP2024534840A (ja) 2021-08-26 2022-08-25 Kif18aのスピロインドリン阻害剤

Country Status (12)

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US (2) US12084420B2 (enExample)
EP (1) EP4392407A1 (enExample)
JP (1) JP2024534840A (enExample)
KR (1) KR20240109977A (enExample)
CN (1) CN119241504A (enExample)
AU (1) AU2022334480A1 (enExample)
CA (1) CA3230123A1 (enExample)
CL (1) CL2024000560A1 (enExample)
IL (1) IL310863A (enExample)
MX (1) MX2024002391A (enExample)
TW (1) TW202317092A (enExample)
WO (1) WO2023028564A1 (enExample)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MA54543A (fr) 2018-12-20 2022-03-30 Amgen Inc Inhibiteurs de kif18a
TW202416973A (zh) 2022-08-18 2024-05-01 美商雅客森醫療公司 Kif18a抑制劑及其用途
CN119790049A (zh) * 2022-09-30 2025-04-08 楚浦创制(武汉)医药科技有限公司 2-氨基嘧啶类化合物及其应用、药用组合物
WO2024114730A1 (zh) * 2022-11-30 2024-06-06 微境生物医药科技(上海)有限公司 一种用于癌症治疗的药物组合物
TW202438053A (zh) * 2023-02-23 2024-10-01 美商佛拉斯托醫療公司 Kif18a吲哚啉抑制劑之固體調配物及多晶形式
WO2024188338A1 (zh) * 2023-03-16 2024-09-19 微境生物医药科技(上海)有限公司 Kif18a抑制剂
CN121909029A (zh) 2023-06-14 2026-04-21 沃拉斯查疗法公司 用kif18a的吲哚啉抑制剂治疗癌症的方法
WO2025190325A1 (zh) * 2024-03-13 2025-09-18 海南先声再明医药股份有限公司 Kif18a抑制剂和微管蛋白抑制剂的药物组合及用途

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