JP2024531064A - ジアリールイソオキサゾリン誘導体を作製するための方法 - Google Patents

ジアリールイソオキサゾリン誘導体を作製するための方法 Download PDF

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Publication number
JP2024531064A
JP2024531064A JP2024503432A JP2024503432A JP2024531064A JP 2024531064 A JP2024531064 A JP 2024531064A JP 2024503432 A JP2024503432 A JP 2024503432A JP 2024503432 A JP2024503432 A JP 2024503432A JP 2024531064 A JP2024531064 A JP 2024531064A
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Japan
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formula
compound
methyl
alkyl
clause
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Pending
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JP2024503432A
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Japanese (ja)
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JP2024531064A5 (https=
Inventor
フ，ジンダン
ウ，グアンミン
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Elanco US Inc
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Elanco US Inc
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Publication of JP2024531064A publication Critical patent/JP2024531064A/ja
Publication of JP2024531064A5 publication Critical patent/JP2024531064A5/ja
Pending legal-status Critical Current

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
JP2024503432A 2021-08-11 2022-08-10 ジアリールイソオキサゾリン誘導体を作製するための方法 Pending JP2024531064A (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US202163231858P 2021-08-11 2021-08-11
US63/231,858 2021-08-11
US202263306240P 2022-02-03 2022-02-03
US63/306,240 2022-02-03
PCT/US2022/039965 WO2023018806A1 (en) 2021-08-11 2022-08-10 Process for making diaryl isoxazoline derivative

Publications (2)

Publication Number Publication Date
JP2024531064A true JP2024531064A (ja) 2024-08-29
JP2024531064A5 JP2024531064A5 (https=) 2025-08-18

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ID=83191860

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JP2024503432A Pending JP2024531064A (ja) 2021-08-11 2022-08-10 ジアリールイソオキサゾリン誘導体を作製するための方法

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Country Link
US (1) US20240308993A1 (https=)
EP (1) EP4384514A1 (https=)
JP (1) JP2024531064A (https=)
KR (1) KR20240046112A (https=)
AU (1) AU2022326468A1 (https=)
BR (1) BR112023026362A2 (https=)
CA (1) CA3224701A1 (https=)
MX (1) MX2023014962A (https=)
TW (1) TW202312880A (https=)
WO (1) WO2023018806A1 (https=)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2021311722A1 (en) 2020-07-24 2023-02-02 Elanco Us Inc. Process for making an isoxazoline compound and intermediate thereof
NO20240925A1 (en) * 2023-09-15 2025-03-17 Evah Atlantic Inc Dihydroisoxazole compound for use in reducing ectoparasite infestations on fish
CN117486869A (zh) * 2023-11-06 2024-02-02 北京康立生医药技术开发有限公司 一种眼科治疗药物新的制备方法

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2747354C (en) 2008-12-19 2016-12-06 Novartis Ag Isoxazoline derivatives and their use as pesticide
AU2011220041A1 (en) 2010-02-25 2012-08-23 Syngenta Limited Process for the preparation of isoxazoline derivatives
JP6075563B2 (ja) 2011-11-08 2017-02-08 日産化学工業株式会社 光学活性イソキサゾリン化合物の触媒的不斉合成方法及び光学活性イソキサゾリン化合物
WO2013079407A1 (en) 2011-11-29 2013-06-06 Novartis Ag Aryl derivatives for controlling ectoparasites
JP2015505560A (ja) 2012-02-03 2015-02-23 ゾエティス・エルエルシー 抗寄生虫薬としてのキラルイソオキサゾリンアゼチジン誘導体の製造法
MX368078B (es) 2012-11-21 2019-09-17 Zoetis Llc Sintesis de derivados de isoxazolina espirociclicos.
WO2014090918A1 (en) * 2012-12-13 2014-06-19 Novartis Ag Process for the enantiomeric enrichment of diaryloxazoline derivatives
EP3018129A1 (en) 2014-11-10 2016-05-11 Novartis Tiergesundheit AG Diaryl isoxazoline compound
DK3440062T3 (da) 2016-04-06 2022-01-03 Boehringer Ingelheim Animal Health Usa Inc Fremgangsmåde til fremstillingen af enantiomerisk berigede isoxazolinforbindelser - krystallinsk toluensolvat af (s)-afoxolaner

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Publication number Publication date
US20240308993A1 (en) 2024-09-19
WO2023018806A1 (en) 2023-02-16
EP4384514A1 (en) 2024-06-19
BR112023026362A2 (pt) 2024-03-05
KR20240046112A (ko) 2024-04-08
AU2022326468A1 (en) 2023-11-30
MX2023014962A (es) 2024-02-13
CA3224701A1 (en) 2023-02-16
TW202312880A (zh) 2023-04-01

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