CA3224701A1 - Process for making diaryl isoxazoline derivative - Google Patents
Process for making diaryl isoxazoline derivative Download PDFInfo
- Publication number
- CA3224701A1 CA3224701A1 CA3224701A CA3224701A CA3224701A1 CA 3224701 A1 CA3224701 A1 CA 3224701A1 CA 3224701 A CA3224701 A CA 3224701A CA 3224701 A CA3224701 A CA 3224701A CA 3224701 A1 CA3224701 A1 CA 3224701A1
- Authority
- CA
- Canada
- Prior art keywords
- formula
- compound
- alkyl
- clause
- methyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US202163231858P | 2021-08-11 | 2021-08-11 | |
| US63/231,858 | 2021-08-11 | ||
| US202263306240P | 2022-02-03 | 2022-02-03 | |
| US63/306,240 | 2022-02-03 | ||
| PCT/US2022/039965 WO2023018806A1 (en) | 2021-08-11 | 2022-08-10 | Process for making diaryl isoxazoline derivative |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CA3224701A1 true CA3224701A1 (en) | 2023-02-16 |
Family
ID=83191860
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA3224701A Pending CA3224701A1 (en) | 2021-08-11 | 2022-08-10 | Process for making diaryl isoxazoline derivative |
Country Status (10)
| Country | Link |
|---|---|
| US (1) | US20240308993A1 (https=) |
| EP (1) | EP4384514A1 (https=) |
| JP (1) | JP2024531064A (https=) |
| KR (1) | KR20240046112A (https=) |
| AU (1) | AU2022326468A1 (https=) |
| BR (1) | BR112023026362A2 (https=) |
| CA (1) | CA3224701A1 (https=) |
| MX (1) | MX2023014962A (https=) |
| TW (1) | TW202312880A (https=) |
| WO (1) | WO2023018806A1 (https=) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU2021311722A1 (en) | 2020-07-24 | 2023-02-02 | Elanco Us Inc. | Process for making an isoxazoline compound and intermediate thereof |
| NO20240925A1 (en) * | 2023-09-15 | 2025-03-17 | Evah Atlantic Inc | Dihydroisoxazole compound for use in reducing ectoparasite infestations on fish |
| CN117486869A (zh) * | 2023-11-06 | 2024-02-02 | 北京康立生医药技术开发有限公司 | 一种眼科治疗药物新的制备方法 |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2747354C (en) | 2008-12-19 | 2016-12-06 | Novartis Ag | Isoxazoline derivatives and their use as pesticide |
| AU2011220041A1 (en) | 2010-02-25 | 2012-08-23 | Syngenta Limited | Process for the preparation of isoxazoline derivatives |
| JP6075563B2 (ja) | 2011-11-08 | 2017-02-08 | 日産化学工業株式会社 | 光学活性イソキサゾリン化合物の触媒的不斉合成方法及び光学活性イソキサゾリン化合物 |
| WO2013079407A1 (en) | 2011-11-29 | 2013-06-06 | Novartis Ag | Aryl derivatives for controlling ectoparasites |
| JP2015505560A (ja) | 2012-02-03 | 2015-02-23 | ゾエティス・エルエルシー | 抗寄生虫薬としてのキラルイソオキサゾリンアゼチジン誘導体の製造法 |
| MX368078B (es) | 2012-11-21 | 2019-09-17 | Zoetis Llc | Sintesis de derivados de isoxazolina espirociclicos. |
| WO2014090918A1 (en) * | 2012-12-13 | 2014-06-19 | Novartis Ag | Process for the enantiomeric enrichment of diaryloxazoline derivatives |
| EP3018129A1 (en) | 2014-11-10 | 2016-05-11 | Novartis Tiergesundheit AG | Diaryl isoxazoline compound |
| DK3440062T3 (da) | 2016-04-06 | 2022-01-03 | Boehringer Ingelheim Animal Health Usa Inc | Fremgangsmåde til fremstillingen af enantiomerisk berigede isoxazolinforbindelser - krystallinsk toluensolvat af (s)-afoxolaner |
-
2022
- 2022-08-10 AU AU2022326468A patent/AU2022326468A1/en active Pending
- 2022-08-10 WO PCT/US2022/039965 patent/WO2023018806A1/en not_active Ceased
- 2022-08-10 EP EP22764943.1A patent/EP4384514A1/en active Pending
- 2022-08-10 CA CA3224701A patent/CA3224701A1/en active Pending
- 2022-08-10 MX MX2023014962A patent/MX2023014962A/es unknown
- 2022-08-10 BR BR112023026362A patent/BR112023026362A2/pt unknown
- 2022-08-10 KR KR1020237042100A patent/KR20240046112A/ko active Pending
- 2022-08-10 US US18/576,593 patent/US20240308993A1/en active Pending
- 2022-08-10 JP JP2024503432A patent/JP2024531064A/ja active Pending
- 2022-08-11 TW TW111130189A patent/TW202312880A/zh unknown
Also Published As
| Publication number | Publication date |
|---|---|
| US20240308993A1 (en) | 2024-09-19 |
| WO2023018806A1 (en) | 2023-02-16 |
| JP2024531064A (ja) | 2024-08-29 |
| EP4384514A1 (en) | 2024-06-19 |
| BR112023026362A2 (pt) | 2024-03-05 |
| KR20240046112A (ko) | 2024-04-08 |
| AU2022326468A1 (en) | 2023-11-30 |
| MX2023014962A (es) | 2024-02-13 |
| TW202312880A (zh) | 2023-04-01 |
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