JP2024528986A5 - - Google Patents

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Publication number
JP2024528986A5
JP2024528986A5 JP2024506668A JP2024506668A JP2024528986A5 JP 2024528986 A5 JP2024528986 A5 JP 2024528986A5 JP 2024506668 A JP2024506668 A JP 2024506668A JP 2024506668 A JP2024506668 A JP 2024506668A JP 2024528986 A5 JP2024528986 A5 JP 2024528986A5
Authority
JP
Japan
Application number
JP2024506668A
Other languages
Japanese (ja)
Other versions
JP2024528986A (ja
JPWO2023015199A5 (https=
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2022/074455 external-priority patent/WO2023015199A1/en
Publication of JP2024528986A publication Critical patent/JP2024528986A/ja
Publication of JP2024528986A5 publication Critical patent/JP2024528986A5/ja
Publication of JPWO2023015199A5 publication Critical patent/JPWO2023015199A5/ja
Pending legal-status Critical Current

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JP2024506668A 2021-08-03 2022-08-03 Hpk1アンタゴニスト及びその使用 Pending JP2024528986A (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US202163203890P 2021-08-03 2021-08-03
US63/203,890 2021-08-03
US202163264749P 2021-12-01 2021-12-01
US63/264,749 2021-12-01
PCT/US2022/074455 WO2023015199A1 (en) 2021-08-03 2022-08-03 Hpk1 antagonists and uses thereof

Publications (3)

Publication Number Publication Date
JP2024528986A JP2024528986A (ja) 2024-08-01
JP2024528986A5 true JP2024528986A5 (https=) 2025-08-13
JPWO2023015199A5 JPWO2023015199A5 (https=) 2025-08-13

Family

ID=85156431

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2024506668A Pending JP2024528986A (ja) 2021-08-03 2022-08-03 Hpk1アンタゴニスト及びその使用

Country Status (4)

Country Link
US (1) US20250011331A1 (https=)
EP (1) EP4380565A4 (https=)
JP (1) JP2024528986A (https=)
WO (1) WO2023015199A1 (https=)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20250236619A1 (en) * 2022-02-23 2025-07-24 Chia Tai Tianqing Pharmaceutical Group Co., Ltd. Fused bicyclic compound containing pyrrolinone
JP2025519624A (ja) * 2022-06-10 2025-06-26 貝達薬業股▲ふん▼有限公司 Hpk1阻害剤およびその医薬における使用
WO2024078448A1 (zh) * 2022-10-10 2024-04-18 珠海宇繁生物科技有限责任公司 一种hpk1激酶抑制剂及其制备方法和应用
WO2025021181A1 (zh) * 2023-07-26 2025-01-30 正大天晴药业集团股份有限公司 取代的吡咯啉酮化合物
WO2025096666A1 (en) * 2023-10-30 2025-05-08 Nimbus Saturn, Inc. Solid forms of hpk1 antagonists
WO2026072991A1 (en) * 2024-09-26 2026-04-02 Arvinas Operations, Inc. Hpk1 targeting compounds and uses thereof

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPWO2008047831A1 (ja) * 2006-10-17 2010-02-25 協和発酵キリン株式会社 Jak阻害剤
KR101846475B1 (ko) * 2015-04-27 2018-04-09 주식회사 녹십자 TNIK, IKKε 및 TBK1 억제제로서의 화합물 및 이를 포함하는 약학적 조성물
RS61919B1 (sr) * 2015-06-25 2021-06-30 Univ Health Network Inhibitori hpk1 i postupci za njihovo korišćenje
WO2018167147A1 (en) * 2017-03-15 2018-09-20 F. Hoffmann-La Roche Ag Azaindoles as inhibitors of hpk1
JP7167146B2 (ja) * 2017-11-06 2022-11-08 ブリストル-マイヤーズ スクイブ カンパニー Hpk1阻害剤として有用なイソフラノン化合物
US11453681B2 (en) * 2019-05-23 2022-09-27 Gilead Sciences, Inc. Substituted eneoxindoles and uses thereof
CN114945366B (zh) * 2019-09-13 2025-01-07 林伯士萨顿公司 Hpk1拮抗剂和其用途
WO2021262684A1 (en) * 2020-06-22 2021-12-30 Pmv Pharmaceuticals, Inc. METHODS AND COMPOUNDS FOR RESTORING MUTANT p53 FUNCTION

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