|
US7956064B2
(en)
*
|
2006-09-01 |
2011-06-07 |
Cylene Pharmaceuticals, Inc. |
Fused tricyclic compounds as serine-threonine protein kinase and PARP modulators
|
|
PT2268618E
(pt)
|
2008-03-03 |
2015-10-12 |
Novartis Ag |
Compostos e composições moduladores da actividade tlr
|
|
US20100173013A1
(en)
*
|
2009-01-08 |
2010-07-08 |
Denis Drygin |
Treatment of neoplastic disorders using combination therapies
|
|
BRPI1016185A2
(pt)
*
|
2009-04-17 |
2016-04-19 |
Cylene Pharmaceuticals Inc |
processo para o tratamento de distúrbios associados à atividade da proteína quinase ck2
|
|
US9968574B2
(en)
*
|
2009-05-15 |
2018-05-15 |
The University Of Kentucky Research Foundation |
Treatment of MCI and Alzheimer's disease
|
|
CN102596969A
(zh)
*
|
2009-08-26 |
2012-07-18 |
赛林药物股份有限公司 |
用作蛋白激酶调节剂的稠合喹啉类化合物
|
|
JP5567137B2
(ja)
*
|
2009-09-03 |
2014-08-06 |
ブリストル−マイヤーズ スクイブ カンパニー |
Jak2阻害剤、ならびに骨髄増殖性疾患および癌の治療のためのそれらの使用
|
|
MX2012003316A
(es)
*
|
2009-09-16 |
2012-07-23 |
Cylene Pharmaceuticals Inc |
Compuestos triciclicos y usos farmaceuticos de los mismos.
|
|
WO2011049625A1
(en)
|
2009-10-20 |
2011-04-28 |
Mansour Samadpour |
Method for aflatoxin screening of products
|
|
PH12012500901A1
(en)
|
2009-11-05 |
2016-08-05 |
Rhizen Pharmaceuticals Sa |
Novel benzopyran kinase modulators
|
|
WO2011063398A1
(en)
*
|
2009-11-23 |
2011-05-26 |
Cylene Pharamaceuticals, Inc. |
Polymorphs and salts of a kinase inhibitor
|
|
US9109227B2
(en)
|
2010-01-05 |
2015-08-18 |
Institut National De La Sante Et De La Recherche Medicale (Inserm) |
FLT3 receptor antagonists for the treatment or the prevention of pain disorders
|
|
US10106798B2
(en)
|
2010-01-05 |
2018-10-23 |
Institut National De La Sante Et De La Recherche Medicale (Inserm) |
FLT3 receptor antagonists for the treatment or the prevention of pain disorders
|
|
TWI503323B
(zh)
*
|
2010-03-29 |
2015-10-11 |
Oncotherapy Science Inc |
三環化合物以及含此化合物之pbk抑制劑
|
|
HRP20190128T1
(hr)
|
2011-05-04 |
2019-03-08 |
Rhizen Pharmaceuticals S.A. |
Novi spojevi kao modulatori protein kinaza
|
|
CN102731431A
(zh)
*
|
2012-06-20 |
2012-10-17 |
盛世泰科生物医药技术(苏州)有限公司 |
一种5-溴噻唑-4-甲酸的制备方法
|
|
CN109970742A
(zh)
|
2012-07-04 |
2019-07-05 |
理森制药股份公司 |
选择性PI3Kδ抑制剂
|
|
JP6437452B2
(ja)
|
2013-01-14 |
2018-12-12 |
インサイト・ホールディングス・コーポレイションIncyte Holdings Corporation |
Pimキナーゼ阻害剤として有用な二環式芳香族カルボキサミド化合物
|
|
RS60244B1
(sr)
|
2013-01-15 |
2020-06-30 |
Incyte Holdings Corp |
Jedinjenja tiazolkarboksamida i piridinkarboksamida korisna kao inhibitori pim kinaze
|
|
CN105764501A
(zh)
|
2013-07-26 |
2016-07-13 |
现代化制药公司 |
改善比生群治疗效益的组合物
|
|
CN105658653A
(zh)
|
2013-08-23 |
2016-06-08 |
因赛特公司 |
可用作pim激酶抑制剂的呋喃并-和噻吩并-吡啶甲酰胺化合物
|
|
WO2016010897A1
(en)
|
2014-07-14 |
2016-01-21 |
Incyte Corporation |
Bicyclic heteroaromatic carboxamide compounds useful as pim kinase inhibitors
|
|
US9580418B2
(en)
|
2014-07-14 |
2017-02-28 |
Incyte Corporation |
Bicyclic aromatic carboxamide compounds useful as Pim kinase inhibitors
|
|
WO2016196244A1
(en)
|
2015-05-29 |
2016-12-08 |
Incyte Corporation |
Pyridineamine compounds useful as pim kinase inhibitors
|
|
TWI734699B
(zh)
|
2015-09-09 |
2021-08-01 |
美商英塞特公司 |
Pim激酶抑制劑之鹽
|
|
US9920032B2
(en)
|
2015-10-02 |
2018-03-20 |
Incyte Corporation |
Heterocyclic compounds useful as pim kinase inhibitors
|
|
CN108341774B
(zh)
*
|
2017-01-25 |
2022-07-19 |
首药控股(北京)股份有限公司 |
取代的喹啉酮类抑制剂
|
|
US11319320B2
(en)
|
2017-11-06 |
2022-05-03 |
Snap Bio, Inc. |
PIM kinase inhibitor compositions, methods, and uses thereof
|
|
AR113922A1
(es)
|
2017-12-08 |
2020-07-01 |
Incyte Corp |
Terapia de combinación de dosis baja para el tratamiento de neoplasias mieloproliferativas
|
|
ES2971712T3
(es)
|
2017-12-22 |
2024-06-06 |
Hibercell Inc |
Derivados de cromenopiridina como inhibidores de la fosfatidilinositol fosfato cinasa
|
|
US11071727B2
(en)
|
2018-01-26 |
2021-07-27 |
Northwestern University |
Therapeutic targeting of proteolytic cleavage of the mixed lineage leukemia gene product (MLL1) by taspase1 using kinase inhibitors
|
|
WO2019191896A1
(en)
*
|
2018-04-03 |
2019-10-10 |
3Sm Biotron Inc. |
Fms-like tyrosine kinase inhibitors
|
|
MA54243A
(fr)
*
|
2018-11-15 |
2021-09-22 |
Nippon Shinyaku Co Ltd |
Composé de 1,3,4-oxadiazolone et médicament
|
|
CN109369526A
(zh)
*
|
2018-12-19 |
2019-02-22 |
桂林理工大学 |
一种两面针碱衍生物的合成方法及其抗肿瘤应用
|
|
GB201902759D0
(en)
|
2019-02-28 |
2019-04-17 |
Benevolentai Bio Ltd |
Compositions and uses thereof
|
|
TW202112784A
(zh)
|
2019-06-17 |
2021-04-01 |
美商佩特拉製藥公司 |
作為磷脂酸肌醇磷酸激酶抑制劑之𠳭唏并嘧啶衍生物
|
|
CN111320605A
(zh)
*
|
2020-03-09 |
2020-06-23 |
吉林工程技术师范学院 |
一种银催化的含氟菲啶衍生物的制备方法
|
|
CN113444085B
(zh)
*
|
2020-03-26 |
2022-04-08 |
东南大学 |
一种具有克服顺铂耐药的抗肿瘤化合物及其制备与应用
|
|
CN113444084A
(zh)
*
|
2020-03-26 |
2021-09-28 |
东南大学 |
一类抗肿瘤化合物及其制备与用途
|
|
BR112022019554A2
(pt)
*
|
2020-03-30 |
2022-12-06 |
Senhwa Biosciences Inc |
Método e composição farmacêutica para tratar uma infecção viral por ácido ribonucleico, e, uso de um composto
|
|
EP3967307A1
(en)
|
2020-09-15 |
2022-03-16 |
Instytut Hematologii I Transfuzologii |
Use of pim kinase inhibitors to augment the efficacy of anti-cd20 antibody-based therapies in hematologic malignancies and non-malignant conditions
|
|
EP4230628B1
(en)
*
|
2020-10-16 |
2025-10-15 |
Shanghai de Novo Pharmatech Co., Ltd. |
Triheterocyclic derivative, and pharmaceutical composition and application thereof
|
|
GB202102895D0
(en)
*
|
2021-03-01 |
2021-04-14 |
Cambridge Entpr Ltd |
Novel compounds, compositions and therapeutic uses thereof
|
|
WO2023126951A1
(en)
*
|
2022-01-03 |
2023-07-06 |
Yeda Research And Development Co. Ltd. |
Inhibitors of autophagy-related protein-protein interactions
|
|
WO2023225586A2
(en)
*
|
2022-05-19 |
2023-11-23 |
4M Therapeutics Inc. |
Novel azaphenantrhene derivatives as inhibitors of glycogen synthase kinase 3 for therapeutic use
|
|
JP2026504483A
(ja)
*
|
2023-02-03 |
2026-02-05 |
ミラティ セラピューティクス, インコーポレイテッド |
置換三環式化合物
|
|
US11987581B1
(en)
|
2023-12-19 |
2024-05-21 |
King Faisal University |
Imidazo[1,2-c]pyrido[3,4-e]pyrimidine-2-carboxylic acids as CK2 inhibitors
|
|
US12024518B1
(en)
|
2023-12-20 |
2024-07-02 |
King Faisal University |
Pyrazolo[4,3-C][1,6]naphthyridines as CK2 inhibitors
|
|
US12012414B1
(en)
|
2024-01-04 |
2024-06-18 |
King Faisal University |
Imidazo[1,5-a]pyrido[4,3-e]pyrimidines as CK2 inhibitors
|
|
US11964974B1
(en)
|
2024-01-08 |
2024-04-23 |
King Faisal University |
Imidazo[1,2-c]pyrido[3,4-e]pyrimidine-3-carboxylic acids as CK2 inhibitors
|
|
US11981676B1
(en)
|
2024-01-16 |
2024-05-14 |
King Faisal University |
Pyrazolo[4,3-c][2,6]naphthyridines as CK2 inhibitors
|
|
US12187726B1
(en)
|
2024-02-06 |
2025-01-07 |
King Faisal University |
Imidazo[1,5-a]pyrido[4,3-e]pyrazines as CK2 inhibitors
|