JP2024524215A5 - - Google Patents

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Publication number
JP2024524215A5
JP2024524215A5 JP2023578919A JP2023578919A JP2024524215A5 JP 2024524215 A5 JP2024524215 A5 JP 2024524215A5 JP 2023578919 A JP2023578919 A JP 2023578919A JP 2023578919 A JP2023578919 A JP 2023578919A JP 2024524215 A5 JP2024524215 A5 JP 2024524215A5
Authority
JP
Japan
Prior art keywords
group
protected
piperidine
groups
independently selected
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2023578919A
Other languages
English (en)
Japanese (ja)
Other versions
JP2024524215A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/EP2022/067126 external-priority patent/WO2022268935A2/en
Publication of JP2024524215A publication Critical patent/JP2024524215A/ja
Publication of JP2024524215A5 publication Critical patent/JP2024524215A5/ja
Pending legal-status Critical Current

Links

JP2023578919A 2021-06-23 2022-06-23 Nlrp3阻害剤を調製するための方法 Pending JP2024524215A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
IN202141028180 2021-06-23
IN202141028180 2021-06-23
PCT/EP2022/067126 WO2022268935A2 (en) 2021-06-23 2022-06-23 Novel process

Publications (2)

Publication Number Publication Date
JP2024524215A JP2024524215A (ja) 2024-07-05
JP2024524215A5 true JP2024524215A5 (enExample) 2025-06-27

Family

ID=82458485

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2023578919A Pending JP2024524215A (ja) 2021-06-23 2022-06-23 Nlrp3阻害剤を調製するための方法

Country Status (12)

Country Link
US (1) US20240150291A1 (enExample)
EP (1) EP4359385A2 (enExample)
JP (1) JP2024524215A (enExample)
KR (1) KR20240024842A (enExample)
CN (1) CN118019727A (enExample)
AR (1) AR126215A1 (enExample)
AU (1) AU2022300325A1 (enExample)
CA (1) CA3219597A1 (enExample)
IL (1) IL308071A (enExample)
MX (1) MX2023014547A (enExample)
TW (1) TW202317514A (enExample)
WO (1) WO2022268935A2 (enExample)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2023220628A1 (en) * 2022-02-15 2024-05-23 F. Hoffmann-La Roche Ag Processes for the preparation of 1,2,3,5,6,7-hexahydro-s-indacene derivatives
WO2024133610A1 (en) * 2022-12-23 2024-06-27 F. Hoffmann-La Roche Ag Proccesses for the preparation of an nlrp3 inhibitor
WO2025036914A1 (en) 2023-08-16 2025-02-20 F. Hoffmann-La Roche Ag Process for the preparation of preparing 1-ethyl-n-((1,2,3,5,6,7-hexahydro-s-indacen-4-yl)carbamoyl)piperidine-4-sulfonamide
WO2025153532A1 (en) 2024-01-16 2025-07-24 NodThera Limited Nlrp3 inhibitors and glp-1 agonists combination therapies

Family Cites Families (22)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZA917435B (en) * 1990-09-26 1992-05-27 Takeda Chemical Industries Ltd Herbicides
CA2059450A1 (en) * 1991-01-24 1992-07-25 Nobuyuki Sakashita Subsituted pyridinesulfonamide compound or its salt, process for preparing the same, and herbicide containing the same
JP2001518069A (ja) * 1997-05-02 2001-10-09 ドクター・レディーズ・リサーチ・ファウンデーション 低脂質性、抗高血圧性特性を有する新規な抗糖尿病化合物、それらの製造方法及びそれらを含有する薬学的組成物
ATE342266T1 (de) * 2000-11-16 2006-11-15 Sankyo Co 1-methylcarbapenemderivate
US7199147B2 (en) * 2001-06-12 2007-04-03 Dainippon Sumitomo Pharma Co., Ltd. Rho kinase inhibitors
MXPA04010172A (es) * 2002-04-18 2005-02-03 Schering Corp 1-(4-piperidinil)benzimidazolonas como antagonistas de histamina h3).
US7759387B2 (en) * 2003-10-08 2010-07-20 Piramal Life Sciences Limited Fibrinogen receptor antagonists and their use
DOP2006000009A (es) * 2005-01-13 2006-08-15 Arena Pharm Inc Procedimiento para preparar eteres de pirazolo [3,4-d] pirimidina
US8614215B2 (en) * 2007-02-22 2013-12-24 Merck Serono Sa Quinoxaline inhibitors of phosphoinositide-3-kinases (PI3Ks)
US20120196889A1 (en) * 2009-02-25 2012-08-02 H. Lundbeck A/S Catecholamine derivatives and prodrugs thereof
JP5898962B2 (ja) * 2012-01-11 2016-04-06 東京応化工業株式会社 レジスト組成物及びレジストパターン形成方法
EP3383853B1 (en) * 2015-12-01 2020-11-04 Merck Sharp & Dohme Corp. Homobispiperidinyl derivatives as liver x receptor (lxr) beta agonists for treating e.g. alzheimer's disease
KR102669722B1 (ko) * 2017-07-07 2024-05-29 인플라좀 리미티드 신규한 설폰아마이드 카복스아마이드 화합물
GB201712282D0 (en) * 2017-07-31 2017-09-13 Nodthera Ltd Selective inhibitors of NLRP3 inflammasome
SG11202001164SA (en) * 2017-08-15 2020-03-30 Inflazome Ltd Novel sulfonamide carboxamide compounds
KR20210018199A (ko) * 2018-03-26 2021-02-17 씨4 테라퓨틱스, 인코포레이티드 이카로스의 분해를 위한 세레블론 결합제
MA52489A (fr) * 2018-05-04 2021-03-10 Inflazome Ltd Nouveaux composés
CA3113573A1 (en) * 2018-09-21 2020-03-26 Novartis Ag Isoxazole carboxamide compounds and uses thereof
GB201817038D0 (en) 2018-10-19 2018-12-05 Inflazome Ltd Novel processes
GB201819083D0 (en) * 2018-11-23 2019-01-09 Inflazome Ltd Novel compounds
WO2020157069A1 (en) * 2019-01-28 2020-08-06 NodThera Limited Amino heterocyclic compounds and uses thereof
CN111393415B (zh) * 2020-04-30 2020-11-20 苏州信诺维医药科技有限公司 一种杂芳腈类化合物及其应用

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