JP2024520646A5 - - Google Patents

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Publication number
JP2024520646A5
JP2024520646A5 JP2023574378A JP2023574378A JP2024520646A5 JP 2024520646 A5 JP2024520646 A5 JP 2024520646A5 JP 2023574378 A JP2023574378 A JP 2023574378A JP 2023574378 A JP2023574378 A JP 2023574378A JP 2024520646 A5 JP2024520646 A5 JP 2024520646A5
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pharmaceutically acceptable
acceptable salt
compound according
compound
pain
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Pending
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JP2023574378A
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English (en)
Japanese (ja)
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JP2024520646A (ja
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Priority claimed from PCT/US2022/032202 external-priority patent/WO2022256679A1/en
Publication of JP2024520646A publication Critical patent/JP2024520646A/ja
Publication of JP2024520646A5 publication Critical patent/JP2024520646A5/ja
Pending legal-status Critical Current

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JP2023574378A 2021-06-04 2022-06-03 ナトリウムチャネルのモジュレーターとしてのn-(ヒドロキシアルキル(ヘテロ)アリール)テトラヒドロフランカルボキサミド類似体 Pending JP2024520646A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202163196970P 2021-06-04 2021-06-04
US63/196,970 2021-06-04
PCT/US2022/032202 WO2022256679A1 (en) 2021-06-04 2022-06-03 N-(hydroxyalkyl (hetero)aryl) tetrahydrofuran carboxamide analogs as modulators of sodium channels

Publications (2)

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JP2024520646A JP2024520646A (ja) 2024-05-24
JP2024520646A5 true JP2024520646A5 (enExample) 2025-06-11

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JP2023574378A Pending JP2024520646A (ja) 2021-06-04 2022-06-03 ナトリウムチャネルのモジュレーターとしてのn-(ヒドロキシアルキル(ヘテロ)アリール)テトラヒドロフランカルボキサミド類似体

Country Status (7)

Country Link
US (1) US20240400544A1 (enExample)
EP (1) EP4347584A1 (enExample)
JP (1) JP2024520646A (enExample)
CN (1) CN117794919A (enExample)
AU (1) AU2022286438A1 (enExample)
CA (1) CA3221939A1 (enExample)
WO (1) WO2022256679A1 (enExample)

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CN120040429B (zh) * 2024-02-23 2026-03-31 山东盛迪医药有限公司 一种取代四氢呋喃衍生物的结晶形式及其用途
CN120040430A (zh) * 2024-02-23 2025-05-27 山东盛迪医药有限公司 一种取代四氢呋喃衍生物的可药用盐、其结晶形式及用途
WO2025176204A1 (zh) * 2024-02-23 2025-08-28 江苏恒瑞医药股份有限公司 一种吡啶-n-氧化物衍生物的结晶形式、盐及其用途
CN120774914A (zh) * 2024-04-03 2025-10-14 武汉人福创新药物研发中心有限公司 作为Nav1.8抑制剂的四氢呋喃吡啶酮类化合物
WO2025218764A1 (zh) * 2024-04-19 2025-10-23 广州市联瑞制药有限公司 作为电压门控钠通道抑制剂的化合物及其应用
WO2025223429A1 (zh) * 2024-04-22 2025-10-30 晶新医药研发(上海)有限公司 一种五元杂环类化合物、药物组合物及其应用
WO2025223430A1 (zh) * 2024-04-22 2025-10-30 晶新医药研发(上海)有限公司 一种五元杂环类化合物、药物组合物及其应用
CN118388466A (zh) * 2024-04-23 2024-07-26 安润医药科技(苏州)有限公司 作钠通道调节剂的酰胺衍生物及其用途
WO2025252109A1 (zh) * 2024-06-04 2025-12-11 成都苑东生物制药股份有限公司 一种取代四氢呋喃类衍生物、其制备方法及用途
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