JP2024512497A5 - - Google Patents

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Publication number
JP2024512497A5
JP2024512497A5 JP2023557369A JP2023557369A JP2024512497A5 JP 2024512497 A5 JP2024512497 A5 JP 2024512497A5 JP 2023557369 A JP2023557369 A JP 2023557369A JP 2023557369 A JP2023557369 A JP 2023557369A JP 2024512497 A5 JP2024512497 A5 JP 2024512497A5
Authority
JP
Japan
Prior art keywords
compound
independently selected
compound according
sulfur
nitrogen
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2023557369A
Other languages
English (en)
Japanese (ja)
Other versions
JP2024512497A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2022/020491 external-priority patent/WO2022197763A1/en
Publication of JP2024512497A publication Critical patent/JP2024512497A/ja
Publication of JP2024512497A5 publication Critical patent/JP2024512497A5/ja
Pending legal-status Critical Current

Links

JP2023557369A 2021-03-17 2022-03-16 血漿カリクレインの阻害剤 Pending JP2024512497A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202163162487P 2021-03-17 2021-03-17
US63/162,487 2021-03-17
PCT/US2022/020491 WO2022197763A1 (en) 2021-03-17 2022-03-16 Inhibitors of plasma kallikrein

Publications (2)

Publication Number Publication Date
JP2024512497A JP2024512497A (ja) 2024-03-19
JP2024512497A5 true JP2024512497A5 (enExample) 2025-03-24

Family

ID=81326196

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2023557369A Pending JP2024512497A (ja) 2021-03-17 2022-03-16 血漿カリクレインの阻害剤

Country Status (5)

Country Link
US (1) US20240226106A1 (enExample)
EP (1) EP4308229A1 (enExample)
JP (1) JP2024512497A (enExample)
CN (1) CN117396469A (enExample)
WO (1) WO2022197763A1 (enExample)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP3765459A1 (en) 2018-03-13 2021-01-20 Shire Human Genetic Therapies, Inc. Substituted imidazopyridines as inhibitors of plasma kallikrein and uses thereof
EP4031245A1 (en) 2019-09-18 2022-07-27 Takeda Pharmaceutical Company Limited Heteroaryl plasma kallikrein inhibitors
DK4031547T3 (da) 2019-09-18 2024-09-09 Takeda Pharmaceuticals Co Plasmakallikreininhibitorer og anvendelser deraf

Family Cites Families (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4911920A (en) 1986-07-30 1990-03-27 Alcon Laboratories, Inc. Sustained release, comfort formulation for glaucoma therapy
FR2588189B1 (fr) 1985-10-03 1988-12-02 Merck Sharp & Dohme Composition pharmaceutique de type a transition de phase liquide-gel
JP2594486B2 (ja) 1991-01-15 1997-03-26 アルコン ラボラトリーズ インコーポレイテッド 局所的眼薬組成物
US5212162A (en) 1991-03-27 1993-05-18 Alcon Laboratories, Inc. Use of combinations gelling polysaccharides and finely divided drug carrier substrates in topical ophthalmic compositions
US6309853B1 (en) 1994-08-17 2001-10-30 The Rockfeller University Modulators of body weight, corresponding nucleic acids and proteins, and diagnostic and therapeutic uses thereof
JP2003509428A (ja) * 1999-09-17 2003-03-11 アボツト・ゲー・エム・ベー・ハー・ウント・コンパニー・カーゲー 治療薬としてのピラゾロピリミジン
CN1486302A (zh) * 2000-12-07 2004-03-31 CV���ƹ�˾ 作为抗冠状动脉疾病或动脉硬化的abca-1加强化合物的取代1,3,5-三嗪和嘧啶
TW201103904A (en) * 2009-06-11 2011-02-01 Hoffmann La Roche Janus kinase inhibitor compounds and methods
WO2014074715A1 (en) * 2012-11-07 2014-05-15 Genentech, Inc. Cyclopropyl amide derivatives
ES2693718T3 (es) * 2013-11-06 2018-12-13 Bristol-Myers Squibb Company Derivados de piridina sustituidos útiles como inhibidores de GSK-3
EP3134408B1 (en) * 2014-04-22 2020-08-12 Merck Sharp & Dohme Corp. FACTOR XIa INHIBITORS
ES2735924T3 (es) * 2015-04-17 2019-12-20 Dow Agrosciences Llc Moléculas que tienen utilidad plaguicida e intermediarios, composiciones y procesos, relacionados con ellas
JP6629958B2 (ja) * 2015-07-29 2020-01-15 ブリストル−マイヤーズ スクイブ カンパニーBristol−Myers Squibb Company アルキルまたはシクロアルキルP2’基を担持する大員環の第XIa因子阻害剤
EP3601259B1 (en) * 2017-03-30 2022-02-23 F. Hoffmann-La Roche AG Isoquinolines as inhibitors of hpk1
AU2018244935A1 (en) * 2017-03-30 2019-08-15 F. Hoffmann-La Roche Ag Naphthyridines as inhibitors of HPK1
EA202091269A1 (ru) * 2017-11-21 2020-08-07 Бристол-Маерс Сквибб Компани Сульфон-, пиридин-, алкил-, амид-замещенные гетероарильные соединения
EP3765459A1 (en) 2018-03-13 2021-01-20 Shire Human Genetic Therapies, Inc. Substituted imidazopyridines as inhibitors of plasma kallikrein and uses thereof
TW202116753A (zh) * 2019-07-11 2021-05-01 大陸商南京征祥醫藥有限公司 以噌啉作為hpk1的抑制劑
CN114573575B (zh) * 2020-04-28 2023-08-04 江南大学 一类含氧五元杂环化合物、合成方法、药物组合物及用途

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