JP2024510504A5 - - Google Patents

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Publication number
JP2024510504A5
JP2024510504A5 JP2023557370A JP2023557370A JP2024510504A5 JP 2024510504 A5 JP2024510504 A5 JP 2024510504A5 JP 2023557370 A JP2023557370 A JP 2023557370A JP 2023557370 A JP2023557370 A JP 2023557370A JP 2024510504 A5 JP2024510504 A5 JP 2024510504A5
Authority
JP
Japan
Prior art keywords
independently selected
nitrogen
sulfur
oxygen
compound according
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2023557370A
Other languages
English (en)
Japanese (ja)
Other versions
JP2024510504A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2022/020527 external-priority patent/WO2022197789A1/en
Publication of JP2024510504A publication Critical patent/JP2024510504A/ja
Publication of JP2024510504A5 publication Critical patent/JP2024510504A5/ja
Pending legal-status Critical Current

Links

JP2023557370A 2021-03-17 2022-03-16 血漿カリクレインの多環式インヒビター Pending JP2024510504A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202163162483P 2021-03-17 2021-03-17
US63/162,483 2021-03-17
PCT/US2022/020527 WO2022197789A1 (en) 2021-03-17 2022-03-16 Polycyclic inhibitors of plasma kallikrein

Publications (2)

Publication Number Publication Date
JP2024510504A JP2024510504A (ja) 2024-03-07
JP2024510504A5 true JP2024510504A5 (enExample) 2025-03-25

Family

ID=81328648

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2023557370A Pending JP2024510504A (ja) 2021-03-17 2022-03-16 血漿カリクレインの多環式インヒビター

Country Status (5)

Country Link
US (1) US20240199613A1 (enExample)
EP (1) EP4308564A1 (enExample)
JP (1) JP2024510504A (enExample)
CN (1) CN117355523A (enExample)
WO (1) WO2022197789A1 (enExample)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP3765459A1 (en) 2018-03-13 2021-01-20 Shire Human Genetic Therapies, Inc. Substituted imidazopyridines as inhibitors of plasma kallikrein and uses thereof
EP4031245A1 (en) 2019-09-18 2022-07-27 Takeda Pharmaceutical Company Limited Heteroaryl plasma kallikrein inhibitors
DK4031547T3 (da) 2019-09-18 2024-09-09 Takeda Pharmaceuticals Co Plasmakallikreininhibitorer og anvendelser deraf
CN118239959A (zh) * 2022-12-23 2024-06-25 上海深势唯思科技有限责任公司 环丙烷类tlr7和8抑制剂及其制备方法和用途

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4911920A (en) 1986-07-30 1990-03-27 Alcon Laboratories, Inc. Sustained release, comfort formulation for glaucoma therapy
FR2588189B1 (fr) 1985-10-03 1988-12-02 Merck Sharp & Dohme Composition pharmaceutique de type a transition de phase liquide-gel
JP2594486B2 (ja) 1991-01-15 1997-03-26 アルコン ラボラトリーズ インコーポレイテッド 局所的眼薬組成物
US5212162A (en) 1991-03-27 1993-05-18 Alcon Laboratories, Inc. Use of combinations gelling polysaccharides and finely divided drug carrier substrates in topical ophthalmic compositions
US6309853B1 (en) 1994-08-17 2001-10-30 The Rockfeller University Modulators of body weight, corresponding nucleic acids and proteins, and diagnostic and therapeutic uses thereof
US6989385B2 (en) * 2000-12-21 2006-01-24 Vertex Pharmaceuticals Incorporated Pyrazole compounds useful as protein kinase inhibitors
EP1750715A1 (en) * 2004-06-04 2007-02-14 Icos Corporation Methods for treating mast cell disorders
KR20080080584A (ko) * 2005-11-30 2008-09-04 버텍스 파마슈티칼스 인코포레이티드 c-Met의 억제제 및 이의 용도
WO2013052526A1 (en) * 2011-10-06 2013-04-11 Merck Sharp & Dohme Corp. Triazolyl pde10 inhibitors
JP6280546B2 (ja) * 2012-06-26 2018-02-14 デル マー ファーマシューティカルズ ジアンヒドロガラクチトール、ジアセチルジアンヒドロガラクチトール、ジブロモズルシトール、又はこれらの類似体若しくは誘導体を用いた、遺伝子多型又はahi1の調節不全若しくは変異を有する患者におけるチロシンキナーゼインヒビター抵抗性悪性腫瘍を処置するための方法
CN104059069B (zh) * 2013-08-22 2016-08-10 北京康立生医药技术开发有限公司 一种替卡格雷的制备方法
EP3134408B1 (en) * 2014-04-22 2020-08-12 Merck Sharp & Dohme Corp. FACTOR XIa INHIBITORS
EP3765459A1 (en) * 2018-03-13 2021-01-20 Shire Human Genetic Therapies, Inc. Substituted imidazopyridines as inhibitors of plasma kallikrein and uses thereof

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