JP2024506382A5 - - Google Patents
Info
- Publication number
- JP2024506382A5 JP2024506382A5 JP2023548868A JP2023548868A JP2024506382A5 JP 2024506382 A5 JP2024506382 A5 JP 2024506382A5 JP 2023548868 A JP2023548868 A JP 2023548868A JP 2023548868 A JP2023548868 A JP 2023548868A JP 2024506382 A5 JP2024506382 A5 JP 2024506382A5
- Authority
- JP
- Japan
- Prior art keywords
- approximately
- pharmaceutical composition
- less
- decanoate
- pharmaceutically acceptable
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US202163149550P | 2021-02-15 | 2021-02-15 | |
| US63/149,550 | 2021-02-15 | ||
| PCT/US2022/016278 WO2022174134A1 (en) | 2021-02-15 | 2022-02-14 | Abiraterone prodrugs |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2024506382A JP2024506382A (ja) | 2024-02-13 |
| JP2024506382A5 true JP2024506382A5 (enExample) | 2025-02-19 |
Family
ID=80625499
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2023548868A Pending JP2024506382A (ja) | 2021-02-15 | 2022-02-14 | アビラテロンプロドラッグ |
Country Status (6)
| Country | Link |
|---|---|
| US (3) | US11957696B2 (enExample) |
| EP (1) | EP4291159A1 (enExample) |
| JP (1) | JP2024506382A (enExample) |
| CN (1) | CN117120034A (enExample) |
| CA (1) | CA3207282A1 (enExample) |
| WO (1) | WO2022174134A1 (enExample) |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP3577109A4 (en) | 2017-01-31 | 2020-11-18 | Arvinas Operations, Inc. | CEREMONY LIGANDS AND BIFUNCTIONAL COMPOUNDS CONTAINING THEM |
| JP7644713B2 (ja) | 2019-03-06 | 2025-03-12 | プロペラ セラピューティクス インコーポレイテッド | アビラテロンプロドラッグ |
| EP4077309A1 (en) | 2019-12-19 | 2022-10-26 | Arvinas Operations, Inc. | Compounds and methods for the targeted degradation of androgen receptor |
| JP7850366B2 (ja) * | 2020-09-02 | 2026-04-23 | アステラス ユーエス エルエルシー | アビラテロンプロドラッグ |
| CA3207282A1 (en) * | 2021-02-15 | 2022-08-18 | Matthew J. Sharp | Abiraterone prodrugs |
| CN118215466A (zh) * | 2021-09-08 | 2024-06-18 | 普洛佩拉治疗公司 | 口服阿比特龙制剂 |
| KR20240167653A (ko) | 2022-03-01 | 2024-11-27 | 프로펠라 쎄라퓨틱스, 인크. | 아비라테론 데카노에이트 프로드러그 및 요법에서의 용도 |
| US20240180900A1 (en) * | 2022-10-24 | 2024-06-06 | Arvinas Operations, Inc. | Compounds and methods for the targeted degradation of androgen receptor |
| WO2024107928A1 (en) | 2022-11-16 | 2024-05-23 | Propella Therapeutics, Inc. | Abiraterone decanoate composition and use in therapy |
| CN116046950A (zh) * | 2023-01-18 | 2023-05-02 | 河北省药品医疗器械检验研究院(河北省化妆品检验研究中心) | 一种检测醋酸阿比特龙中5种杂质的方法 |
| WO2024186523A2 (en) * | 2023-03-07 | 2024-09-12 | Board Of Regents, The University Of Texas System | Glucocorticoid receptor antagonists for cancer treatment |
Family Cites Families (42)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4432987A (en) * | 1982-04-23 | 1984-02-21 | Pfizer Inc. | Crystalline benzenesulfonate salts of sultamicillin |
| US5604213A (en) | 1992-03-31 | 1997-02-18 | British Technology Group Limited | 17-substituted steroids useful in cancer treatment |
| DE60045751D1 (de) * | 1999-09-30 | 2011-04-28 | Harbor Biosciences Inc | Therapeutische Behandlung androgenrezeptorbedingter Leiden |
| JP2004002321A (ja) * | 2002-03-11 | 2004-01-08 | Takeda Chem Ind Ltd | 性ホルモン依存性疾患治療剤 |
| GB0418900D0 (en) | 2004-08-24 | 2004-09-29 | Btg Int Ltd | Novel salt forms |
| US20080051380A1 (en) | 2006-08-25 | 2008-02-28 | Auerbach Alan H | Methods and compositions for treating cancer |
| US20090124587A1 (en) | 2007-07-12 | 2009-05-14 | Auerbach Alan H | METHODS FOR TREATING CANCER USING 17alpha-HYDROXYLASE/C17,20-LYASE INHIBITORS |
| WO2010091306A1 (en) | 2009-02-05 | 2010-08-12 | Tokai Pharmaceuticals | Novel prodrugs of steroidal cyp17 inhibitors/antiandrogens |
| EP2506855A4 (en) | 2009-11-30 | 2014-07-30 | Harbor Biosciences Inc | ANTICARCINOMA COMPOUNDS AND SCREENING METHODS |
| CA2819515A1 (en) | 2010-12-16 | 2012-06-21 | Biomarin Pharmaceutical Inc. | Cyp11b, cyp17, and/or cyp21 inhibitors |
| JP6091510B2 (ja) | 2011-10-10 | 2017-03-08 | ザック システム | １７−置換ステロイドの製造方法 |
| US20140079636A1 (en) | 2012-04-16 | 2014-03-20 | Dinesh U. Chimmanamada | Targeted therapeutics |
| CA2871314A1 (en) | 2012-04-23 | 2013-10-31 | Alphora Research Inc. | Process for preparation of 17-substituted steroids |
| WO2014009434A1 (en) | 2012-07-11 | 2014-01-16 | Sandoz Ag | Self-microemulsifying drug delivery system of abiraterone or abiraterone acetate |
| US20140011992A1 (en) | 2012-12-20 | 2014-01-09 | Crystal Pharma, S.A.U. | Synthesis of abiraterone and related compounds |
| DK2945628T3 (da) * | 2013-01-15 | 2020-05-04 | Aragon Pharmaceuticals Inc | Androgen receptormodulator i kombination med abirateronacetat og prednison til behandling af prostatacancer |
| US20150337003A1 (en) | 2013-01-18 | 2015-11-26 | Cortendo Ab (Publ) | Abiraterone and analogs thereof for the treatment of diseases associated with cortisol overproduction |
| EP2969227B1 (en) | 2013-03-15 | 2019-05-08 | Iceutica Inc. | Abiraterone acetate formulation |
| US20150246060A1 (en) | 2013-03-15 | 2015-09-03 | Iceutica Inc. | Abiraterone Acetate Formulation and Methods of Use |
| EP3035938B1 (en) | 2013-09-10 | 2020-08-19 | Madrigal Pharmaceuticals, Inc. | Targeted therapeutics |
| US20150157646A1 (en) | 2013-09-27 | 2015-06-11 | Iceutica Inc. | Abiraterone Steroid Formulation |
| CN106456795A (zh) | 2014-03-03 | 2017-02-22 | 辛塔医药品有限公司 | 靶向治疗学 |
| EP3131586A4 (en) | 2014-03-18 | 2017-10-25 | Madrigal Pharmaceuticals, Inc. | Targeted therapeutics |
| CN104017045B (zh) | 2014-06-23 | 2016-01-13 | 广州艾格生物科技有限公司 | 甾体cyp17抑制剂的新型药物前体及其应用、制备方法 |
| US9937259B2 (en) | 2014-06-27 | 2018-04-10 | Zhuhai Beihai Biotech Co., Ltd. | Abiraterone derivatives and non-covalent complexes with albumin |
| BR112017003219A2 (pt) | 2014-09-18 | 2017-11-28 | Iceutica Inc | formulação de acetato de abiraterona e métodos de uso |
| CN104356191A (zh) | 2014-09-29 | 2015-02-18 | 上海延安药业（湖北）有限公司 | 阿比特龙单琥珀酸酯及其制备方法 |
| WO2016082792A1 (zh) | 2014-11-28 | 2016-06-02 | 四川海思科制药有限公司 | 一种阿比特龙衍生物及其制备方法和医药用途 |
| CN104710499A (zh) | 2015-02-15 | 2015-06-17 | 重庆医药工业研究院有限责任公司 | 一种丙酸阿比特龙的晶型及其制备方法 |
| CA3008909C (en) | 2015-12-23 | 2023-10-03 | The University Of British Columbia | Lipid-linked prodrugs |
| JP6842474B2 (ja) | 2016-02-02 | 2021-03-17 | 深▲セン▼市塔吉瑞生物医▲薬▼有限公司Ｓｈｅｎｚｈｅｎ ＴａｒｇｅｔＲｘ，Ｉｎｃ． | ステロイド系化合物、当該化合物を含む組成物及びその使用 |
| CN109922809B (zh) | 2016-10-11 | 2021-08-13 | 珠海贝海生物技术有限公司 | 阿比特龙衍生物及其制剂 |
| CN106977577A (zh) | 2017-04-21 | 2017-07-25 | 湖南师范大学 | 两类阿比特龙衍生物的合成 |
| US20190105332A1 (en) * | 2017-10-11 | 2019-04-11 | Janssen Oncology, Inc. | Methods of treating prostate cancer |
| CN118684633A (zh) | 2018-10-18 | 2024-09-24 | 埃萨制药股份有限公司 | 雄激素受体调节剂及其使用方法 |
| CN113473974A (zh) | 2019-01-25 | 2021-10-01 | 深圳市药欣生物科技有限公司 | 药物组合物 |
| JP7644713B2 (ja) * | 2019-03-06 | 2025-03-12 | プロペラ セラピューティクス インコーポレイテッド | アビラテロンプロドラッグ |
| EP3941478A4 (en) * | 2019-03-18 | 2022-12-28 | Dispersol Technologies, LLC | PHARMACEUTICAL FORMULATIONS OF ABIRATERON CYCLIC OLIGOMERS AND METHODS OF PREPARATION AND ADMINISTRATION THEREOF |
| JP7850366B2 (ja) * | 2020-09-02 | 2026-04-23 | アステラス ユーエス エルエルシー | アビラテロンプロドラッグ |
| CN113929727A (zh) | 2020-09-28 | 2022-01-14 | 南京易腾药物研究院有限公司 | 阿比特龙酯类衍生物及其制备方法和应用 |
| CA3207282A1 (en) | 2021-02-15 | 2022-08-18 | Matthew J. Sharp | Abiraterone prodrugs |
| CN118215466A (zh) | 2021-09-08 | 2024-06-18 | 普洛佩拉治疗公司 | 口服阿比特龙制剂 |
-
2022
- 2022-02-14 CA CA3207282A patent/CA3207282A1/en active Pending
- 2022-02-14 JP JP2023548868A patent/JP2024506382A/ja active Pending
- 2022-02-14 WO PCT/US2022/016278 patent/WO2022174134A1/en not_active Ceased
- 2022-02-14 US US17/670,712 patent/US11957696B2/en active Active
- 2022-02-14 CN CN202280028179.4A patent/CN117120034A/zh active Pending
- 2022-02-14 EP EP22707562.9A patent/EP4291159A1/en active Pending
-
2023
- 2023-07-26 US US18/226,339 patent/US20240139212A1/en active Pending
-
2025
- 2025-09-17 US US19/331,393 patent/US20260014172A1/en active Pending
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