JP2023543038A5 - - Google Patents

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Publication number
JP2023543038A5
JP2023543038A5 JP2023519291A JP2023519291A JP2023543038A5 JP 2023543038 A5 JP2023543038 A5 JP 2023543038A5 JP 2023519291 A JP2023519291 A JP 2023519291A JP 2023519291 A JP2023519291 A JP 2023519291A JP 2023543038 A5 JP2023543038 A5 JP 2023543038A5
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JP
Japan
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group
pharmaceutically acceptable
acceptable salt
hydrogen atom
compound
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JP2023519291A
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English (en)
Japanese (ja)
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JP7824282B2 (ja
JP2023543038A (ja
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Priority claimed from PCT/US2021/052025 external-priority patent/WO2022067082A1/en
Publication of JP2023543038A publication Critical patent/JP2023543038A/ja
Publication of JP2023543038A5 publication Critical patent/JP2023543038A5/ja
Application granted granted Critical
Publication of JP7824282B2 publication Critical patent/JP7824282B2/ja
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JP2023519291A 2020-09-28 2021-09-24 縮合ヘテロアリール化合物およびCaMKII阻害剤としてのその使用 Active JP7824282B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202063084217P 2020-09-28 2020-09-28
US63/084,217 2020-09-28
PCT/US2021/052025 WO2022067082A1 (en) 2020-09-28 2021-09-24 Fused heteroaryl compounds and their use as camkii inhibitors

Publications (3)

Publication Number Publication Date
JP2023543038A JP2023543038A (ja) 2023-10-12
JP2023543038A5 true JP2023543038A5 (enExample) 2024-10-01
JP7824282B2 JP7824282B2 (ja) 2026-03-04

Family

ID=80821052

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2023519291A Active JP7824282B2 (ja) 2020-09-28 2021-09-24 縮合ヘテロアリール化合物およびCaMKII阻害剤としてのその使用

Country Status (14)

Country Link
US (2) US11795172B2 (enExample)
EP (1) EP4216948A4 (enExample)
JP (1) JP7824282B2 (enExample)
KR (1) KR20230107551A (enExample)
CN (1) CN116940354A (enExample)
AU (1) AU2021350015A1 (enExample)
CA (1) CA3196946A1 (enExample)
CL (1) CL2023000894A1 (enExample)
CO (1) CO2023005189A2 (enExample)
IL (1) IL301480A (enExample)
MX (1) MX2023003610A (enExample)
PE (1) PE20240148A1 (enExample)
TW (1) TW202229273A (enExample)
WO (1) WO2022067082A1 (enExample)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP7824282B2 (ja) * 2020-09-28 2026-03-04 カーデュリオン・ファーマシューティカルズ・インコーポレイテッド 縮合ヘテロアリール化合物およびCaMKII阻害剤としてのその使用
WO2023134692A1 (zh) * 2022-01-13 2023-07-20 浙江同源康医药股份有限公司 多环类化合物及其用途
CN115160235B (zh) * 2022-08-10 2023-12-15 宜宾学院 一种2,3-二氢喹唑啉-4(1h)-酮类化合物及其超声合成方法
US20250145630A1 (en) * 2023-11-07 2025-05-08 Cardurion Pharmaceuticals, Inc. Polymorphs of a pyridinylimidazo[1,2-b]pyridazine

Family Cites Families (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1317266A2 (en) 2000-08-08 2003-06-11 Ortho-McNeil Pharmaceutical, Inc. Neuroprotective 2-pyridinamine compositions and related methods
HK1054393B (en) 2000-09-20 2009-08-28 Ortho-Mcneil Pharmaceutical, Inc. Pyrazine derivatives as modulators of tyrosine kinases
US20030187026A1 (en) * 2001-12-13 2003-10-02 Qun Li Kinase inhibitors
JP2007504229A (ja) 2003-09-02 2007-03-01 メルク エンド カムパニー インコーポレーテッド 代謝調節型グルタミン酸受容体−5のモジュレーターとしてのビピリジルアミン類およびエーテル類
US7776857B2 (en) 2007-04-05 2010-08-17 Amgen Inc. Aurora kinase modulators and method of use
US9216173B2 (en) 2011-10-05 2015-12-22 Merck Sharp & Dohme Corp. 2-Pyridyl carboxamide-containing spleen tyrosine kinase (SYK) inhibitors
HRP20180037T1 (hr) 2012-04-17 2018-03-23 Fujifilm Corporation Heterociklični spoj koji sadrži dušik ili njegovu sol
CA2894126A1 (en) 2012-12-21 2014-06-26 Epizyme, Inc. Prmt5 inhibitors and uses thereof
CN107074856A (zh) * 2014-09-05 2017-08-18 阿略斯泰罗斯医疗公司 CaMKII抑制剂及其用途
AR110252A1 (es) 2016-11-30 2019-03-13 Gilead Sciences Inc Compuestos heterocíclicos fusionados como inhibidores de la quinasa cam
CN110799190B (zh) 2017-03-27 2024-04-19 卡都瑞恩医药有限公司 杂环化合物
JP7447098B2 (ja) 2018-09-25 2024-03-11 カーデュリオン・ファーマシューティカルズ・インコーポレイテッド アミノピリミジン化合物
WO2020068846A1 (en) * 2018-09-25 2020-04-02 Heterocyclic Compound Heterocyclic compound
US20230000842A1 (en) 2019-01-17 2023-01-05 Samumed, Llc Methods of treating cartilage disorders through inhibition of clk and dyrk
JP7824282B2 (ja) * 2020-09-28 2026-03-04 カーデュリオン・ファーマシューティカルズ・インコーポレイテッド 縮合ヘテロアリール化合物およびCaMKII阻害剤としてのその使用

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