JP2023536911A5 - - Google Patents

Info

Publication number
JP2023536911A5
JP2023536911A5 JP2023507579A JP2023507579A JP2023536911A5 JP 2023536911 A5 JP2023536911 A5 JP 2023536911A5 JP 2023507579 A JP2023507579 A JP 2023507579A JP 2023507579 A JP2023507579 A JP 2023507579A JP 2023536911 A5 JP2023536911 A5 JP 2023536911A5
Authority
JP
Japan
Prior art keywords
crystalline
anhydrous
ray powder
powder diffraction
compound
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2023507579A
Other languages
English (en)
Japanese (ja)
Other versions
JP7789056B2 (ja
JP2023536911A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2021/044341 external-priority patent/WO2022031701A1/en
Publication of JP2023536911A publication Critical patent/JP2023536911A/ja
Publication of JP2023536911A5 publication Critical patent/JP2023536911A5/ja
Application granted granted Critical
Publication of JP7789056B2 publication Critical patent/JP7789056B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2023507579A 2020-08-03 2021-08-03 O-糖タンパク質-2-アセトアミド-2-デオキシ-3-d-グルコピラノシダーゼ阻害剤の結晶形態 Active JP7789056B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202063060281P 2020-08-03 2020-08-03
US63/060,281 2020-08-03
PCT/US2021/044341 WO2022031701A1 (en) 2020-08-03 2021-08-03 Crystaline forms of an o-glycoprotein-2-acetamido-2-deoxy-3-d-glucopyranosidase inhibitor

Publications (3)

Publication Number Publication Date
JP2023536911A JP2023536911A (ja) 2023-08-30
JP2023536911A5 true JP2023536911A5 (https=) 2024-08-13
JP7789056B2 JP7789056B2 (ja) 2025-12-19

Family

ID=77640732

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2023507579A Active JP7789056B2 (ja) 2020-08-03 2021-08-03 O-糖タンパク質-2-アセトアミド-2-デオキシ-3-d-グルコピラノシダーゼ阻害剤の結晶形態

Country Status (18)

Country Link
US (1) US20230286972A1 (https=)
EP (1) EP4188925A1 (https=)
JP (1) JP7789056B2 (https=)
KR (1) KR20230061395A (https=)
CN (1) CN116917284A (https=)
AR (1) AR123132A1 (https=)
AU (1) AU2021322186A1 (https=)
BR (1) BR112023002013A2 (https=)
CA (1) CA3188250A1 (https=)
CL (1) CL2023000327A1 (https=)
CO (1) CO2023002543A2 (https=)
CR (1) CR20230118A (https=)
IL (1) IL300365A (https=)
MX (1) MX2023001469A (https=)
PE (1) PE20231168A1 (https=)
TW (1) TW202220984A (https=)
UY (1) UY39366A (https=)
WO (1) WO2022031701A1 (https=)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB2602139B (en) * 2020-12-18 2024-07-24 Nexeon Ltd Electroactive materials for metal-ion batteries
WO2025184490A1 (en) 2024-03-01 2025-09-04 Biogen Ma Inc. N-[4-fluor-5-[[(2s, 4 r)-4-[(6-methoxy-4-pyrimidinyl)oxy]- 2-methyl-1-pyrrolidinyl] methyl ]-2-thiazolyl]acetamid for use in the treatment of alzheimer disease

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2780014A4 (en) 2011-11-18 2015-07-01 Constellation Pharmaceuticals Inc MODULATORS OF METHYL MODIFYING ENZYMES, COMPOSITIONS AND USES THEREOF
US9051269B2 (en) 2011-11-18 2015-06-09 Constellation Pharmaceuticals, Inc. Modulators of methyl modifying enzymes, compositions and uses thereof
WO2013078320A1 (en) 2011-11-21 2013-05-30 Constellation Pharmaceuticals Modulators of methyl modifying enzymes, compositions and uses thereof
JP5989805B2 (ja) 2012-02-10 2016-09-07 コンステレーション・ファーマシューティカルズ・インコーポレイテッドConstellation Pharmaceuticals,Inc. メチル基変更酵素の調節物質、組成物及びその使用
MA38341B1 (fr) 2013-02-11 2018-11-30 Constellation Pharmaceuticals Inc Modulateurs d'enzymes de modification par méthylation, compositions et utilisations associées
US9745305B2 (en) 2013-03-15 2017-08-29 Constellation Pharmaceuticals, Inc. Modulators of methyl modifying enzymes, compositions and uses thereof
US9969716B2 (en) 2013-08-15 2018-05-15 Constellation Pharmaceuticals, Inc. Indole derivatives as modulators of methyl modifying enzymes, compositions and uses thereof
EP3555087A1 (en) 2016-12-16 2019-10-23 Janssen Pharmaceutica NV Monocyclic oga inhibitor compounds
TWI654978B (zh) 2017-01-27 2019-04-01 美商美國禮來大藥廠 5-甲基-1,2,4-二唑-3-基化合物
WO2018154133A1 (en) 2017-02-27 2018-08-30 Janssen Pharmaceutica Nv [1,2,4]-triazolo [1,5-a]-pyrimidinyl derivatives substituted with piperidine, morpholine or piperazine as oga inhibitors
US12180205B2 (en) * 2018-09-19 2024-12-31 Biogen Ma Inc. O-glycoprotein-2-acetamido-2-deoxy-3-d-glucopyranosidase inhibitors

Similar Documents

Publication Publication Date Title
JP2005503386A5 (https=)
DE69720719T2 (de) Mesylat des trihydrats des 5-(2-(4-(1,2-benzothiazol-3-yl)-1-piperazinyl)ethyl)-6-chlor-1,3-dihydro-2(1h)-indol-2-ons (=ziprasidon), seine herstellung und seine anwendung als dopamin d2 antagonist
JPWO2022138988A5 (https=)
ES2466221T3 (es) Monohidrato de mesilato de N-[5-aminosulfonil)-4-metil-1,3-tiazol-2-il]-N-metil-2-[4-(2-piridinil)fenil]acetamida
KR101612642B1 (ko) 테노포비어 알라펜아미드 헤미푸마레이트
JP2023036708A5 (https=)
JP2023536911A5 (https=)
JP2010516681A5 (https=)
JP2023511105A5 (https=)
JP2009534468A5 (https=)
JP2017527578A5 (https=)
JP2020143129A5 (https=)
RU2019100065A (ru) Кристаллы анилинпиримидинового соединения, действующего в качестве ингибитора EGFR
JP2020510661A5 (https=)
JP6832946B2 (ja) キナーゼ阻害剤およびその中間体の調製方法
JP2004516278A (ja) 一酸化窒素合成酵素阻害物質であるリン酸塩
HUP0003230A2 (hu) Egy N-fenil-(2-piridil)-amin-származék kristálymódosulata, valamint előállítási eljárásai és alkalmazása
WO1997042191A1 (en) Mesylate dihydrate salts of 5-(2-(4-(1,2-benzisothiazol-3-yl)-1-piperazinyl)-ethyl)-6-chloro-1,3-dihydro-2(1h)-indol-2-one (=ziprasidone), its preparation and its use as dopamine d2 antagonist
JP2022523368A5 (https=)
SK16702002A3 (sk) Polymorfná forma V 5-chlór-3-(4-metánsulfonylfenyl)-6'-metyl- [2,3']bipyridinylu, spôsob jej výroby, farmaceutický prostriedok s jej obsahom a jej použitie
JP2021535111A5 (https=)
US12428414B2 (en) Methods for purifying isavuconazonium sulfate
JP2022507795A5 (https=)
JP2022553833A5 (https=)
CN102131803A (zh) (1r,2s,3r)-1-(2-(异噁唑-3-基)-1h-咪唑-4-基)丁烷-1,2,3,4-四醇的固体形式及其使用方法