JP2023533982A5 - - Google Patents

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Publication number
JP2023533982A5
JP2023533982A5 JP2023501137A JP2023501137A JP2023533982A5 JP 2023533982 A5 JP2023533982 A5 JP 2023533982A5 JP 2023501137 A JP2023501137 A JP 2023501137A JP 2023501137 A JP2023501137 A JP 2023501137A JP 2023533982 A5 JP2023533982 A5 JP 2023533982A5
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JP
Japan
Prior art keywords
alkyl
pharmaceutically acceptable
acceptable salt
heteroaryl
compound according
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JP2023501137A
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English (en)
Japanese (ja)
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JP2023533982A (ja
JP7758369B2 (ja
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Priority claimed from PCT/US2021/015263 external-priority patent/WO2022010537A1/en
Publication of JP2023533982A publication Critical patent/JP2023533982A/ja
Publication of JP2023533982A5 publication Critical patent/JP2023533982A5/ja
Application granted granted Critical
Publication of JP7758369B2 publication Critical patent/JP7758369B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2023501137A 2020-07-10 2021-01-27 Gas41阻害剤及びその使用方法 Active JP7758369B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202063050303P 2020-07-10 2020-07-10
US63/050,303 2020-07-10
PCT/US2021/015263 WO2022010537A1 (en) 2020-07-10 2021-01-27 Gas41 inhibitors and methods of use thereof

Publications (3)

Publication Number Publication Date
JP2023533982A JP2023533982A (ja) 2023-08-07
JP2023533982A5 true JP2023533982A5 (enExample) 2024-02-02
JP7758369B2 JP7758369B2 (ja) 2025-10-22

Family

ID=79291969

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2023501137A Active JP7758369B2 (ja) 2020-07-10 2021-01-27 Gas41阻害剤及びその使用方法

Country Status (7)

Country Link
US (1) US11858925B2 (enExample)
EP (1) EP4178571A4 (enExample)
JP (1) JP7758369B2 (enExample)
CN (1) CN116113406B (enExample)
AU (1) AU2021304826A1 (enExample)
CA (1) CA3185209A1 (enExample)
WO (1) WO2022010537A1 (enExample)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
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EP4284804A1 (en) 2021-01-26 2023-12-06 Schrödinger, Inc. Tricyclic compounds useful in the treatment of cancer, autoimmune and inflammatory disorders
CN115974864B (zh) * 2022-12-29 2025-09-16 苏州汉德创宏生化科技有限公司 一种2-(3-氮杂环丁基)噻唑盐的合成方法
CN116143763B (zh) * 2023-03-01 2025-09-23 清华大学 靶向gas41的化合物、gas41抑制剂和药物组合物及其用途
CN119307620A (zh) * 2024-12-19 2025-01-14 上海交通大学医学院附属上海儿童医学中心 预后标志物H4K5la在神经母细胞瘤预后评估中的应用

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