JP2023523770A5 - - Google Patents

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Publication number
JP2023523770A5
JP2023523770A5 JP2022566012A JP2022566012A JP2023523770A5 JP 2023523770 A5 JP2023523770 A5 JP 2023523770A5 JP 2022566012 A JP2022566012 A JP 2022566012A JP 2022566012 A JP2022566012 A JP 2022566012A JP 2023523770 A5 JP2023523770 A5 JP 2023523770A5
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JP
Japan
Prior art keywords
pharmaceutically acceptable
acceptable salt
compound according
alkyl
cycloalkyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2022566012A
Other languages
English (en)
Japanese (ja)
Other versions
JP2023523770A (ja
JP7661361B2 (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/IB2021/053517 external-priority patent/WO2021220183A1/en
Publication of JP2023523770A publication Critical patent/JP2023523770A/ja
Publication of JP2023523770A5 publication Critical patent/JP2023523770A5/ja
Application granted granted Critical
Publication of JP7661361B2 publication Critical patent/JP7661361B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2022566012A 2020-04-30 2021-04-28 Il-17のモジュレーターとしてのイミダゾピリミジン Active JP7661361B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202063017679P 2020-04-30 2020-04-30
US63/017,679 2020-04-30
PCT/IB2021/053517 WO2021220183A1 (en) 2020-04-30 2021-04-28 Imidazopyrimidines as modulators of il-17

Publications (3)

Publication Number Publication Date
JP2023523770A JP2023523770A (ja) 2023-06-07
JP2023523770A5 true JP2023523770A5 (enExample) 2024-04-15
JP7661361B2 JP7661361B2 (ja) 2025-04-14

Family

ID=75769661

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2022566012A Active JP7661361B2 (ja) 2020-04-30 2021-04-28 Il-17のモジュレーターとしてのイミダゾピリミジン

Country Status (12)

Country Link
US (1) US12559496B2 (enExample)
EP (1) EP4143193B1 (enExample)
JP (1) JP7661361B2 (enExample)
KR (1) KR20230018387A (enExample)
CN (1) CN115867348B (enExample)
AU (1) AU2021262588A1 (enExample)
BR (1) BR112022021957A2 (enExample)
CA (1) CA3181793A1 (enExample)
ES (1) ES3071556T3 (enExample)
IL (1) IL297734A (enExample)
MX (1) MX2022013650A (enExample)
WO (1) WO2021220183A1 (enExample)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB201909190D0 (en) * 2019-06-26 2019-08-07 Ucb Biopharma Sprl Therapeutic agents
WO2023025783A1 (en) 2021-08-23 2023-03-02 Leo Pharma A/S Small molecule modulators of il-17
WO2023111181A1 (en) 2021-12-16 2023-06-22 Leo Pharma A/S Small molecule modulators of il-17
EP4486737A1 (en) 2022-03-04 2025-01-08 LEO Pharma A/S Small molecule modulators of il-17
TW202430165A (zh) 2022-12-02 2024-08-01 丹麥商理奧藥品公司 Il-17之小分子調節劑
EP4688156A1 (en) * 2023-03-28 2026-02-11 Janssen Pharmaceutica NV Lactam-containing imidazopyridazine il-17 inhibitor compounds

Family Cites Families (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2809660B1 (en) * 2012-02-02 2016-01-20 Ensemble Therapeutics Corporation Macrocyclic compounds for modulating il-17
GB201321736D0 (en) 2013-12-09 2014-01-22 Ucb Pharma Sa Therapeutic agents
ES2702126T3 (es) 2013-12-10 2019-02-27 Bristol Myers Squibb Co Compuestos de imidazopiridazina útiles como moduladores de respuestas a IL-12, IL-23 y/o IFN alfa
MA40759A (fr) * 2014-09-26 2017-08-01 Pfizer Modulateurs de rorc2 de type pyrrolopyridine substitué par un méthyle et trifluorométhyle et leurs procédés d'utilisation
US10152431B2 (en) 2015-03-16 2018-12-11 Honeywell International Inc. System and method for remote set-up and adjustment of peripherals
KR102782807B1 (ko) * 2015-11-18 2025-03-14 브리스톨-마이어스 스큅 컴퍼니 Il-12, il-23 및/또는 ifn 알파 반응의 조정제로서 유용한 이미다조피리다진 화합물
GB201709456D0 (en) 2017-06-14 2017-07-26 Ucb Biopharma Sprl Therapeutic agents
CN111601799B (zh) 2018-01-15 2023-06-09 Ucb生物制药有限责任公司 作为Il-17调节剂的稠合咪唑衍生物
WO2019223718A1 (zh) 2018-05-22 2019-11-28 成都先导药物开发股份有限公司 一种免疫调节剂
US11993574B2 (en) 2018-06-15 2024-05-28 Reata Pharmaceuticals, Inc Pyrazole and imidazole compounds for inhibition of IL-17 and RORgamma
WO2020011731A1 (en) 2018-07-12 2020-01-16 UCB Biopharma SRL Spirocyclic indane analogues as il-17 modulators
JP7664947B2 (ja) 2020-04-30 2025-04-18 ヤンセン ファーマシューティカ エヌ.ベー. Il-17の調節因子としてのイミダゾリダジン
KR20230017211A (ko) 2020-04-30 2023-02-03 얀센 파마슈티카 엔.브이. Il-17 경로의 조절인자를 식별하는 방법
WO2021219784A1 (en) 2020-04-30 2021-11-04 Janssen Pharmaceutica Nv New triazinoindole compounds

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