JP2023522166A5 - - Google Patents

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Publication number
JP2023522166A5
JP2023522166A5 JP2022561040A JP2022561040A JP2023522166A5 JP 2023522166 A5 JP2023522166 A5 JP 2023522166A5 JP 2022561040 A JP2022561040 A JP 2022561040A JP 2022561040 A JP2022561040 A JP 2022561040A JP 2023522166 A5 JP2023522166 A5 JP 2023522166A5
Authority
JP
Japan
Prior art keywords
inhibitor
menin
pharmaceutical combination
combination according
cyp3a4
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2022561040A
Other languages
English (en)
Japanese (ja)
Other versions
JP2023522166A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2021/026141 external-priority patent/WO2021207335A1/en
Publication of JP2023522166A publication Critical patent/JP2023522166A/ja
Publication of JP2023522166A5 publication Critical patent/JP2023522166A5/ja
Pending legal-status Critical Current

Links

JP2022561040A 2020-04-07 2021-04-07 メニン阻害剤とcyp3a4阻害剤との組合せ、およびその使用方法 Pending JP2023522166A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202063006574P 2020-04-07 2020-04-07
US63/006,574 2020-04-07
PCT/US2021/026141 WO2021207335A1 (en) 2020-04-07 2021-04-07 Combinations of menin inhibitors and cyp3a4 inhibitors and methods of use thereof

Publications (2)

Publication Number Publication Date
JP2023522166A JP2023522166A (ja) 2023-05-29
JP2023522166A5 true JP2023522166A5 (enExample) 2024-04-16

Family

ID=78023861

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2022561040A Pending JP2023522166A (ja) 2020-04-07 2021-04-07 メニン阻害剤とcyp3a4阻害剤との組合せ、およびその使用方法

Country Status (10)

Country Link
US (1) US12564590B2 (enExample)
EP (1) EP4132932A4 (enExample)
JP (1) JP2023522166A (enExample)
KR (1) KR20230007359A (enExample)
CN (3) CN120393025A (enExample)
AU (1) AU2021252552A1 (enExample)
CA (1) CA3178691A1 (enExample)
IL (1) IL297039A (enExample)
MX (1) MX2022012471A (enExample)
WO (1) WO2021207335A1 (enExample)

Families Citing this family (9)

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WO2017214367A1 (en) 2016-06-10 2017-12-14 Vitae Pharmaceuticals, Inc. Inhibitors of the menin-mll interaction
TW202525813A (zh) 2019-12-19 2025-07-01 比利時商健生藥品公司 經取代之直鏈螺環接衍生物
EP4132932A4 (en) 2020-04-07 2024-04-17 Syndax Pharmaceuticals, Inc. COMBINATIONS OF MENIN INHIBITORS AND CYP3A4 INHIBITORS AND METHODS OF USE THEREOF
IL308476A (en) 2021-05-14 2024-01-01 Syndax Pharmaceuticals Inc Inhibitors of the menin-mil interaction
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US20250295661A1 (en) * 2022-05-09 2025-09-25 Syndax Pharmaceuticals, Inc. Menin-mll inhibitors for the treatment of cancer
CN120456907A (zh) * 2022-11-02 2025-08-08 库拉肿瘤学公司 急性白血病的治疗方法
CN120529900A (zh) 2022-11-24 2025-08-22 奥莱松基因组股份有限公司 用于治疗癌症的LSD1抑制剂和Menin抑制剂的组合
WO2025106862A1 (en) * 2023-11-17 2025-05-22 Kura Oncology, Inc. Methods of treating kit positive cancers with a menin inhibitor

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CN118234497A (zh) 2021-12-15 2024-06-21 丹娜-法伯癌症研究所 通过破坏menin-mll表观遗传复合体靶向治疗胃肠道间质瘤(gist)
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