JP2023522023A5 - - Google Patents
Info
- Publication number
- JP2023522023A5 JP2023522023A5 JP2022562632A JP2022562632A JP2023522023A5 JP 2023522023 A5 JP2023522023 A5 JP 2023522023A5 JP 2022562632 A JP2022562632 A JP 2022562632A JP 2022562632 A JP2022562632 A JP 2022562632A JP 2023522023 A5 JP2023522023 A5 JP 2023522023A5
- Authority
- JP
- Japan
- Prior art keywords
- morphology
- shows
- approximately
- water vapor
- eur
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP20170197.6 | 2020-04-17 | ||
| EP20170197 | 2020-04-17 | ||
| PCT/EP2021/059604 WO2021209477A1 (en) | 2020-04-17 | 2021-04-14 | Crystalline forms of 4-[(7-chloro-2-methoxybenzo[b][1,5]naphthyridin-10-yl)amino]-2,6-bis(pyrrolidin-1-ylmethyl)phenol and salts thereof |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2023522023A JP2023522023A (ja) | 2023-05-26 |
| JP2023522023A5 true JP2023522023A5 (https=) | 2025-07-16 |
Family
ID=70333787
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2022562632A Pending JP2023522023A (ja) | 2020-04-17 | 2021-04-14 | 4-[(7-クロロ-2-メトキシベンゾ[b][1,5]ナフチリジン-10-イル)アミノ]-2,6-ビス(ピロリジン-1-イルメチル)フェノールおよびそれらの塩の結晶形態 |
Country Status (8)
| Country | Link |
|---|---|
| US (1) | US20230295156A1 (https=) |
| EP (1) | EP4136087A1 (https=) |
| JP (1) | JP2023522023A (https=) |
| CN (1) | CN115515955A (https=) |
| BR (1) | BR112022018436A2 (https=) |
| CA (1) | CA3175552A1 (https=) |
| PH (1) | PH12022552366A1 (https=) |
| WO (1) | WO2021209477A1 (https=) |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR100975895B1 (ko) * | 2008-04-29 | 2010-08-18 | 강민석 | 피로나리딘의 제조방법 및 이를 위한 중간체 |
| CN101544638B (zh) * | 2009-05-12 | 2012-05-30 | 重庆通天药业有限公司 | 乳酸咯萘啶及其药物组合物 |
| CN103373995B (zh) * | 2012-04-28 | 2016-04-27 | 上海迪赛诺药业有限公司 | 一种制备咯萘啶的方法 |
| ES2902143T3 (es) * | 2014-07-04 | 2022-03-25 | Merck Patent Gmbh | Derivados de azepanilo y composiciones farmacéuticas que los comprenden con actividad antiparasitaria |
| CN105461713A (zh) | 2014-09-25 | 2016-04-06 | 刘力 | 苯并萘啶类的新化合物及其组合物和用途 |
| JP2019530712A (ja) * | 2016-10-13 | 2019-10-24 | エムエムヴィ メディシンズ フォア マラリア ヴェンチャーMmv Medicines For Malaria Venture | 新規抗マラリア薬 |
| HUE069225T2 (hu) * | 2018-04-11 | 2025-02-28 | Merck Patent Gmbh | Kinolin-4-karboxamidok és benzonaftiridin származékok kombinációja maláriaellenes gyógyszer-kombinációként |
| CN112209926A (zh) * | 2019-07-12 | 2021-01-12 | 中国中医科学院中药研究所 | 磷酸咯萘啶的多晶型物及其制备方法、应用 |
| CA3182616A1 (en) * | 2020-06-15 | 2021-12-23 | Lukas Shinji OKITSU | Tlr7/8 antagonists and uses thereof |
-
2021
- 2021-04-14 EP EP21717119.8A patent/EP4136087A1/en active Pending
- 2021-04-14 JP JP2022562632A patent/JP2023522023A/ja active Pending
- 2021-04-14 CA CA3175552A patent/CA3175552A1/en active Pending
- 2021-04-14 CN CN202180028991.2A patent/CN115515955A/zh active Pending
- 2021-04-14 PH PH1/2022/552366A patent/PH12022552366A1/en unknown
- 2021-04-14 WO PCT/EP2021/059604 patent/WO2021209477A1/en not_active Ceased
- 2021-04-14 BR BR112022018436A patent/BR112022018436A2/pt unknown
- 2021-04-14 US US17/995,388 patent/US20230295156A1/en active Pending
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