JP2023517729A5 - - Google Patents

Info

Publication number
JP2023517729A5
JP2023517729A5 JP2022555821A JP2022555821A JP2023517729A5 JP 2023517729 A5 JP2023517729 A5 JP 2023517729A5 JP 2022555821 A JP2022555821 A JP 2022555821A JP 2022555821 A JP2022555821 A JP 2022555821A JP 2023517729 A5 JP2023517729 A5 JP 2023517729A5
Authority
JP
Japan
Prior art keywords
process according
disorders
pharmaceutical composition
monohydrochloride salt
crystalline
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2022555821A
Other languages
English (en)
Japanese (ja)
Other versions
JP2023517729A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/EP2021/056749 external-priority patent/WO2021185878A1/en
Publication of JP2023517729A publication Critical patent/JP2023517729A/ja
Publication of JP2023517729A5 publication Critical patent/JP2023517729A5/ja
Priority to JP2025132332A priority Critical patent/JP2025166092A/ja
Pending legal-status Critical Current

Links

JP2022555821A 2020-03-19 2021-03-17 Taar1アゴニストの塩形態および結晶形態 Pending JP2023517729A (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2025132332A JP2025166092A (ja) 2020-03-19 2025-08-07 Taar1アゴニストの塩形態および結晶形態

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP20164069 2020-03-19
EP20164069.5 2020-03-19
PCT/EP2021/056749 WO2021185878A1 (en) 2020-03-19 2021-03-17 Salts and crystalline forms of a taar1 agonist

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2025132332A Division JP2025166092A (ja) 2020-03-19 2025-08-07 Taar1アゴニストの塩形態および結晶形態

Publications (2)

Publication Number Publication Date
JP2023517729A JP2023517729A (ja) 2023-04-26
JP2023517729A5 true JP2023517729A5 (https=) 2024-03-26

Family

ID=69846246

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2022555821A Pending JP2023517729A (ja) 2020-03-19 2021-03-17 Taar1アゴニストの塩形態および結晶形態
JP2025132332A Pending JP2025166092A (ja) 2020-03-19 2025-08-07 Taar1アゴニストの塩形態および結晶形態

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2025132332A Pending JP2025166092A (ja) 2020-03-19 2025-08-07 Taar1アゴニストの塩形態および結晶形態

Country Status (13)

Country Link
US (1) US20230120311A1 (https=)
EP (1) EP4121428B1 (https=)
JP (2) JP2023517729A (https=)
KR (1) KR20220155575A (https=)
CN (1) CN115279752A (https=)
AU (1) AU2021238632A1 (https=)
BR (1) BR112022016746A2 (https=)
CA (1) CA3166331A1 (https=)
ES (1) ES3044409T3 (https=)
IL (1) IL294301A (https=)
MX (1) MX2022010794A (https=)
TW (1) TWI874616B (https=)
WO (1) WO2021185878A1 (https=)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP4731191A1 (en) * 2022-08-12 2026-04-29 F. Hoffmann-La Roche AG Pharmaceutical compositions comprising 5-ethyl-4-methyl- n-[4-[(2 s) morpholin-2-yl]phenyl]-1h-pyrazole-3-carboxamide
WO2024222860A1 (zh) * 2023-04-28 2024-10-31 江苏豪森药业集团有限公司 一种吗啉杂环类化合物的盐及其制备方法和应用
CN117903050B (zh) * 2024-03-15 2024-05-17 中国药科大学 阿立哌唑共晶及其药物组合物和应用

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5323907A (en) 1992-06-23 1994-06-28 Multi-Comp, Inc. Child resistant package assembly for dispensing pharmaceutical medications
CN108713019B (zh) * 2016-03-17 2021-06-15 豪夫迈·罗氏有限公司 具有作为taar的激动剂的活性的5-乙基-4-甲基-吡唑-3-甲酰胺衍生物

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