MX2022010794A - Sales y formas cristalinas de un agonista del receptor 1 asociado a aminas traza (taar1). - Google Patents
Sales y formas cristalinas de un agonista del receptor 1 asociado a aminas traza (taar1).Info
- Publication number
- MX2022010794A MX2022010794A MX2022010794A MX2022010794A MX2022010794A MX 2022010794 A MX2022010794 A MX 2022010794A MX 2022010794 A MX2022010794 A MX 2022010794A MX 2022010794 A MX2022010794 A MX 2022010794A MX 2022010794 A MX2022010794 A MX 2022010794A
- Authority
- MX
- Mexico
- Prior art keywords
- taar1
- crystalline forms
- salts
- taar1 agonist
- agonist
- Prior art date
Links
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
- A61K31/5375—1,4-Oxazines, e.g. morpholine
- A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/13—Crystalline forms, e.g. polymorphs
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Neurosurgery (AREA)
- Engineering & Computer Science (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Psychiatry (AREA)
- Pain & Pain Management (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Medicinal Preparation (AREA)
Abstract
La presente invención se refiere a formas cristalinas y amorfas de sales farmacéuticamente aceptables del agonista de TAAR1 5-etil-4-metil-N-[4-[(2S) morfolin-2-il]fenil]-1H-pirazol-3-carbox amida. También se describen composiciones farmacéuticas adecuadas para la administración a un mamífero que incluyen el agonista de TAAR1, y métodos para el uso del agonista de TAAR1, solo y en combinación con otros compuestos, para tratar enfermedades o afecciones asociadas con la actividad de TAAR1.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP20164069 | 2020-03-19 | ||
PCT/EP2021/056749 WO2021185878A1 (en) | 2020-03-19 | 2021-03-17 | Salts and crystalline forms of a taar1 agonist |
Publications (1)
Publication Number | Publication Date |
---|---|
MX2022010794A true MX2022010794A (es) | 2022-09-27 |
Family
ID=69846246
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MX2022010794A MX2022010794A (es) | 2020-03-19 | 2021-03-17 | Sales y formas cristalinas de un agonista del receptor 1 asociado a aminas traza (taar1). |
Country Status (12)
Country | Link |
---|---|
US (1) | US20230120311A1 (es) |
EP (1) | EP4121428A1 (es) |
JP (1) | JP2023517729A (es) |
KR (1) | KR20220155575A (es) |
CN (1) | CN115279752A (es) |
AU (1) | AU2021238632A1 (es) |
BR (1) | BR112022016746A2 (es) |
CA (1) | CA3166331A1 (es) |
IL (1) | IL294301A (es) |
MX (1) | MX2022010794A (es) |
TW (1) | TW202140466A (es) |
WO (1) | WO2021185878A1 (es) |
Families Citing this family (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2024033459A1 (en) * | 2022-08-12 | 2024-02-15 | F. Hoffmann-La Roche Ag | Pharmaceutical compositions comprising 5-ethyl-4-methyl- n-[4-[(2 s) morpholin-2-yl]phenyl]-1h-pyrazole-3-carboxamide |
CN117903050B (zh) * | 2024-03-15 | 2024-05-17 | 中国药科大学 | 阿立哌唑共晶及其药物组合物和应用 |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5323907A (en) | 1992-06-23 | 1994-06-28 | Multi-Comp, Inc. | Child resistant package assembly for dispensing pharmaceutical medications |
SG10201913878YA (en) | 2016-03-17 | 2020-03-30 | Hoffmann La Roche | 5-ethyl-4-methyl-pyrazole-3-carboxamide derivative having activity as agonist of taar |
-
2021
- 2021-03-17 JP JP2022555821A patent/JP2023517729A/ja active Pending
- 2021-03-17 MX MX2022010794A patent/MX2022010794A/es unknown
- 2021-03-17 TW TW110109520A patent/TW202140466A/zh unknown
- 2021-03-17 CA CA3166331A patent/CA3166331A1/en active Pending
- 2021-03-17 IL IL294301A patent/IL294301A/en unknown
- 2021-03-17 AU AU2021238632A patent/AU2021238632A1/en active Pending
- 2021-03-17 BR BR112022016746A patent/BR112022016746A2/pt unknown
- 2021-03-17 EP EP21712158.1A patent/EP4121428A1/en active Pending
- 2021-03-17 CN CN202180017438.9A patent/CN115279752A/zh active Pending
- 2021-03-17 KR KR1020227031814A patent/KR20220155575A/ko active Search and Examination
- 2021-03-17 WO PCT/EP2021/056749 patent/WO2021185878A1/en unknown
-
2022
- 2022-09-16 US US17/946,743 patent/US20230120311A1/en active Pending
Also Published As
Publication number | Publication date |
---|---|
JP2023517729A (ja) | 2023-04-26 |
US20230120311A1 (en) | 2023-04-20 |
CN115279752A (zh) | 2022-11-01 |
BR112022016746A2 (pt) | 2022-10-11 |
EP4121428A1 (en) | 2023-01-25 |
IL294301A (en) | 2022-08-01 |
KR20220155575A (ko) | 2022-11-23 |
WO2021185878A1 (en) | 2021-09-23 |
TW202140466A (zh) | 2021-11-01 |
AU2021238632A1 (en) | 2022-07-14 |
CA3166331A1 (en) | 2021-09-23 |
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