EA200800147A1 - Способ получения олмесартан медоксомила - Google Patents
Способ получения олмесартан медоксомилаInfo
- Publication number
- EA200800147A1 EA200800147A1 EA200800147A EA200800147A EA200800147A1 EA 200800147 A1 EA200800147 A1 EA 200800147A1 EA 200800147 A EA200800147 A EA 200800147A EA 200800147 A EA200800147 A EA 200800147A EA 200800147 A1 EA200800147 A1 EA 200800147A1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- olmesartan
- medoksomil
- obtaining
- hypertension
- medicament
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
Abstract
Настоящее изобретение относится к улучшенному способу получения олмесартана и его фармацевтически приемлемых солей и эфиров в качестве активного ингредиента лекарственного средства для лечения гипертонии и связанных с ней болезней и состояний.
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
SI200500221A SI22092A (sl) | 2005-07-29 | 2005-07-29 | Postopek za pripravo olmesartan medoksomila |
EP06002388A EP1816131A1 (en) | 2006-02-06 | 2006-02-06 | Process for the preparation of olmesartan medoxomil |
PCT/EP2006/007453 WO2007017135A2 (en) | 2005-07-29 | 2006-07-27 | Process for the preparation of olmesartan medoxomil |
Publications (2)
Publication Number | Publication Date |
---|---|
EA200800147A1 true EA200800147A1 (ru) | 2008-06-30 |
EA014026B1 EA014026B1 (ru) | 2010-08-30 |
Family
ID=36979539
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EA200800147A EA014026B1 (ru) | 2005-07-29 | 2006-07-27 | Способ получения олмесартан медоксомила |
Country Status (5)
Country | Link |
---|---|
US (1) | US7943779B2 (ru) |
EP (1) | EP1910343B1 (ru) |
CA (1) | CA2616466A1 (ru) |
EA (1) | EA014026B1 (ru) |
WO (1) | WO2007017135A2 (ru) |
Families Citing this family (28)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP1801111B1 (en) * | 2005-12-20 | 2014-07-16 | LEK Pharmaceuticals d.d. | Novel polymorph forms of olmesartan medoxomil |
EP1891952B1 (en) * | 2006-05-04 | 2011-10-05 | LEK Pharmaceuticals d.d. | Pharmaceutical composition of olmesartan medoxomil |
WO2007148344A2 (en) * | 2006-06-19 | 2007-12-27 | Matrix Laboratories Limited | Process for the preparation of olmesartan medoxomil |
KR101458369B1 (ko) * | 2006-10-09 | 2014-11-05 | 씨아이피엘에이 엘티디. | 트리틸 올메사탄 메독소밀 및 올메사탄 메독소밀의 제조방법 |
CA2681591A1 (en) * | 2007-03-23 | 2008-10-02 | Daiichi Sankyo Company, Limited | Pulverized crystals of olmesartan medoxomil |
CN101311168B (zh) * | 2007-05-21 | 2010-12-08 | 上海医药工业研究院 | 4-(1-羟基-1-甲基乙基)-2-丙基咪唑-5-羧酸酯的制备方法 |
GB0710680D0 (en) * | 2007-06-05 | 2007-07-11 | Generics Uk Ltd | Novel crystalline form of olmesartan medoxmil |
GB0710905D0 (en) * | 2007-06-07 | 2007-07-18 | Generics Uk Ltd | Amorphous olmesartan medoxomil |
EP2022790A1 (en) * | 2007-08-08 | 2009-02-11 | LEK Pharmaceuticals D.D. | A process for the preparation or purification of olmesartan medoxomil |
CA2707365A1 (en) | 2007-08-08 | 2009-02-12 | Lek Pharmaceuticals D.D. | A process for the preparation of olmesartan medoxomil |
EP2036904A1 (en) * | 2007-08-08 | 2009-03-18 | LEK Pharmaceuticals D.D. | A process for the preparation of olmesartan medoxomil |
CN102083823B (zh) | 2008-06-09 | 2015-10-07 | 第一三共株式会社 | 1-联苯甲基咪唑化合物的制备方法 |
MY158090A (en) | 2009-04-28 | 2016-08-30 | Daiichi Sankyo Co Ltd | Novel solvate crystals |
ES2527686T3 (es) | 2009-04-28 | 2015-01-28 | Daiichi Sankyo Company, Limited | Procedimiento de producción de olmesartán medoxomil |
WO2011007368A2 (en) | 2009-07-14 | 2011-01-20 | Cadila Healthcare Limited | An improved process for preparation of olmesartan |
WO2011014611A2 (en) * | 2009-07-30 | 2011-02-03 | Dr. Reddy's Laboratories Ltd. | Preparation of olmesartan medoxomil |
WO2011083112A2 (en) | 2010-01-05 | 2011-07-14 | Ratiopharm Gmbh | Solid oral dosage form containing olmesartan medoxomil |
AR083523A1 (es) | 2010-10-29 | 2013-03-06 | Interquim Sa | Procedimiento de obtencion del olmesartan medoxomilo |
MX2014001298A (es) * | 2011-08-05 | 2014-09-01 | Lupin Ltd | Procedimiento para la preparacion de olmesartan medoxomilo. |
CN102351849B (zh) * | 2011-10-26 | 2013-10-02 | 齐鲁天和惠世制药有限公司 | 一种奥美沙坦酯的制备方法 |
US20150225380A1 (en) | 2012-08-22 | 2015-08-13 | Lupin Limited | Novel Method to Obtain Olmesartan Medoxomil With Reduced Particle Size |
KR101418871B1 (ko) * | 2012-08-28 | 2014-07-17 | 한국과학기술연구원 | 올메사탄 메독소밀의 정제방법 |
US10835714B2 (en) | 2016-03-21 | 2020-11-17 | Edwards Lifesciences Corporation | Multi-direction steerable handles for steering catheters |
US10973638B2 (en) | 2016-07-07 | 2021-04-13 | Edwards Lifesciences Corporation | Device and method for treating vascular insufficiency |
US11224511B2 (en) | 2017-04-18 | 2022-01-18 | Edwards Lifesciences Corporation | Heart valve sealing devices and delivery devices therefor |
CN107311990B (zh) * | 2017-07-25 | 2021-09-03 | 浙江华海致诚药业有限公司 | 一种奥美沙坦酯的制备方法 |
US10105222B1 (en) | 2018-01-09 | 2018-10-23 | Edwards Lifesciences Corporation | Native valve repair devices and procedures |
US10945844B2 (en) | 2018-10-10 | 2021-03-16 | Edwards Lifesciences Corporation | Heart valve sealing devices and delivery devices therefor |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
IE920540A1 (en) * | 1991-02-21 | 1992-08-26 | Sankyo Co | 1-biphenylmethylimidazole derivatives, their preparation and¹their therapetuic use |
ATE194603T1 (de) * | 1994-01-28 | 2000-07-15 | Takeda Chemical Industries Ltd | Ein verfahren zur herstellung von tetrazolyl- verbindungen |
JP3671266B2 (ja) | 1996-03-21 | 2005-07-13 | 東洋化成工業株式会社 | 5−置換テトラゾール類の製造方法 |
CN1197866C (zh) | 2003-03-21 | 2005-04-20 | 上海医药工业研究院 | 4,6-二氢呋喃并[3,4-d]咪唑-6-酮衍生物及其盐和制备方法 |
CN1271068C (zh) | 2003-03-25 | 2006-08-23 | 上海医药工业研究院 | 一种奥美沙坦酯的制备方法 |
ITMI20032338A1 (it) * | 2003-11-28 | 2005-05-29 | Dinamite Dipharma S P A In Forma A Bbreviata Diph | Composti feniltetrazolici. |
CN1976926A (zh) | 2004-09-02 | 2007-06-06 | 特瓦制药工业有限公司 | 奥美沙坦酯的制备 |
-
2006
- 2006-07-27 CA CA002616466A patent/CA2616466A1/en not_active Abandoned
- 2006-07-27 WO PCT/EP2006/007453 patent/WO2007017135A2/en active Application Filing
- 2006-07-27 EP EP06776466.2A patent/EP1910343B1/en active Active
- 2006-07-27 EA EA200800147A patent/EA014026B1/ru not_active IP Right Cessation
- 2006-07-27 US US11/997,133 patent/US7943779B2/en not_active Expired - Fee Related
Also Published As
Publication number | Publication date |
---|---|
EA014026B1 (ru) | 2010-08-30 |
EP1910343A2 (en) | 2008-04-16 |
WO2007017135A3 (en) | 2007-04-12 |
US7943779B2 (en) | 2011-05-17 |
EP1910343B1 (en) | 2014-10-29 |
US20090131680A1 (en) | 2009-05-21 |
WO2007017135A2 (en) | 2007-02-15 |
CA2616466A1 (en) | 2007-02-15 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
MM4A | Lapse of a eurasian patent due to non-payment of renewal fees within the time limit in the following designated state(s) |
Designated state(s): AM AZ BY KZ KG MD TJ TM |