JP2023514725A5 - - Google Patents

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Publication number
JP2023514725A5
JP2023514725A5 JP2022550164A JP2022550164A JP2023514725A5 JP 2023514725 A5 JP2023514725 A5 JP 2023514725A5 JP 2022550164 A JP2022550164 A JP 2022550164A JP 2022550164 A JP2022550164 A JP 2022550164A JP 2023514725 A5 JP2023514725 A5 JP 2023514725A5
Authority
JP
Japan
Prior art keywords
carboxamide
oxy
naphthyridine
alkylene
dimethoxy
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
JP2022550164A
Other languages
English (en)
Japanese (ja)
Other versions
JP2023514725A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2021/019294 external-priority patent/WO2021173591A1/en
Publication of JP2023514725A publication Critical patent/JP2023514725A/ja
Publication of JP2023514725A5 publication Critical patent/JP2023514725A5/ja
Withdrawn legal-status Critical Current

Links

JP2022550164A 2020-02-24 2021-02-23 化合物および使用方法 Withdrawn JP2023514725A (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US202062980954P 2020-02-24 2020-02-24
US62/980,954 2020-02-24
US202063121418P 2020-12-04 2020-12-04
US63/121,418 2020-12-04
PCT/US2021/019294 WO2021173591A1 (en) 2020-02-24 2021-02-23 Compounds and methods of use

Publications (2)

Publication Number Publication Date
JP2023514725A JP2023514725A (ja) 2023-04-07
JP2023514725A5 true JP2023514725A5 (https=) 2024-03-01

Family

ID=74885066

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2022550164A Withdrawn JP2023514725A (ja) 2020-02-24 2021-02-23 化合物および使用方法

Country Status (7)

Country Link
US (1) US20230151003A1 (https=)
EP (1) EP4110779A1 (https=)
JP (1) JP2023514725A (https=)
CN (1) CN115605478A (https=)
AU (1) AU2021226747A1 (https=)
CA (1) CA3171473A1 (https=)
WO (1) WO2021173591A1 (https=)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2022551422A (ja) 2019-09-26 2022-12-09 エグゼリクシス, インコーポレイテッド ピリドン化合物およびタンパク質キナーゼの調節における使用の方法
CA3211063A1 (en) 2021-02-19 2022-08-25 Exelixis, Inc. Pyridone compounds and methods of use
CN117343046A (zh) * 2023-09-25 2024-01-05 辽宁大学 一种新型3-氧代-4-取代芳基-3,4-二氢吡嗪-2-甲酰胺类化合物及其应用
CN118878515B (zh) * 2024-06-19 2025-10-28 河北科技大学 一种取代苯胺嘧啶类化合物及其制备方法和用途

Family Cites Families (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3845770A (en) 1972-06-05 1974-11-05 Alza Corp Osmatic dispensing device for releasing beneficial agent
US4326525A (en) 1980-10-14 1982-04-27 Alza Corporation Osmotic device that improves delivery properties of agent in situ
US5364620A (en) 1983-12-22 1994-11-15 Elan Corporation, Plc Controlled absorption diltiazem formulation for once daily administration
US5023252A (en) 1985-12-04 1991-06-11 Conrex Pharmaceutical Corporation Transdermal and trans-membrane delivery of drugs
US5001139A (en) 1987-06-12 1991-03-19 American Cyanamid Company Enchancers for the transdermal flux of nivadipine
US4992445A (en) 1987-06-12 1991-02-12 American Cyanamid Co. Transdermal delivery of pharmaceuticals
US4902514A (en) 1988-07-21 1990-02-20 Alza Corporation Dosage form for administering nilvadipine for treating cardiovascular symptoms
JO2787B1 (en) * 2005-04-27 2014-03-15 امجين إنك, Alternative amide derivatives and methods of use
CN104072480B (zh) * 2013-03-27 2016-12-28 沈阳药科大学 喹啉类化合物及其制备方法和应用
TWI649308B (zh) * 2013-07-24 2019-02-01 小野藥品工業股份有限公司 喹啉衍生物
CN105461687B (zh) * 2014-08-26 2020-06-19 北京京奉医药科技有限公司 含二氢哒嗪酮的喹啉类化合物及其用途
ES2749726T3 (es) * 2014-12-25 2020-03-23 Ono Pharmaceutical Co Derivado de quinolina
CN109896997A (zh) * 2017-12-08 2019-06-18 中国药科大学 N-酰基苯胺类c-Met激酶抑制剂的制备方法及其用途
CN110330479A (zh) * 2019-07-19 2019-10-15 南京华威医药科技集团有限公司 一种用作axl抑制剂的抗肿瘤化合物及其用途

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