JP2023511152A5 - - Google Patents
Info
- Publication number
- JP2023511152A5 JP2023511152A5 JP2022544247A JP2022544247A JP2023511152A5 JP 2023511152 A5 JP2023511152 A5 JP 2023511152A5 JP 2022544247 A JP2022544247 A JP 2022544247A JP 2022544247 A JP2022544247 A JP 2022544247A JP 2023511152 A5 JP2023511152 A5 JP 2023511152A5
- Authority
- JP
- Japan
- Prior art keywords
- group
- substituted
- compound
- unsubstituted
- halogen
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CN202010075139.8 | 2020-01-22 | ||
| CN202010075139.8A CN113149977A (zh) | 2020-01-22 | 2020-01-22 | 一类呼吸道合胞病毒抑制剂的合成与用途 |
| PCT/CN2021/073042 WO2021147947A1 (zh) | 2020-01-22 | 2021-01-21 | 一类呼吸道合胞病毒抑制剂的合成与用途 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2023511152A JP2023511152A (ja) | 2023-03-16 |
| JP2023511152A5 true JP2023511152A5 (https=) | 2024-01-30 |
| JP7726487B2 JP7726487B2 (ja) | 2025-08-20 |
Family
ID=76881779
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2022544247A Active JP7726487B2 (ja) | 2020-01-22 | 2021-01-21 | 呼吸器合胞体ウイルス阻害剤の合成及び使用 |
Country Status (6)
| Country | Link |
|---|---|
| US (1) | US12582661B2 (https=) |
| EP (1) | EP4095136A4 (https=) |
| JP (1) | JP7726487B2 (https=) |
| KR (1) | KR20220130761A (https=) |
| CN (2) | CN113149977A (https=) |
| WO (1) | WO2021147947A1 (https=) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN113149977A (zh) * | 2020-01-22 | 2021-07-23 | 苏州爱科百发生物医药技术有限公司 | 一类呼吸道合胞病毒抑制剂的合成与用途 |
| CN116425754A (zh) * | 2021-12-30 | 2023-07-14 | 苏州爱科百发生物医药技术有限公司 | 芳杂双环化合物及其抗病毒用途 |
| CN120794971A (zh) * | 2024-04-10 | 2025-10-17 | 广州医科大学 | 二氨基嘧啶化合物及其用途 |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5760230A (en) * | 1996-10-11 | 1998-06-02 | Bayer Aktiengesellschaft | 4, 4'-bridged bis-2, 4-diaminoquinazolines |
| US8871756B2 (en) | 2011-08-11 | 2014-10-28 | Hoffmann-La Roche Inc. | Compounds for the treatment and prophylaxis of Respiratory Syncytial Virus disease |
| NO3004079T3 (https=) | 2013-06-04 | 2018-06-16 | ||
| AR099134A1 (es) * | 2014-01-24 | 2016-06-29 | Hoffmann La Roche | Procedimiento para la preparación de n-[(3-aminooxetán-3-il)metil]-2-(1,1-dioxo-3,5-dihidro-1,4-benzotiazepín-4-il)-6-metil-quinazolín-4-amina |
| EP3322704B1 (en) * | 2015-07-16 | 2019-11-27 | H. Hoffnabb-La Roche Ag | Crystalline form of n-[(3-amino-3-oxetanyl)methyl]-2-(2,3-dihydro-1,1-dioxido-1,4-benzothiazepin-4(5h)-yl)-6-methyl-4-quinazolinamine for the treatment of respiratory syncytial virus (rsv) infections |
| DK3324977T3 (da) | 2015-07-22 | 2022-10-17 | Enanta Pharm Inc | Benzodiazepinderivater som rsv-inhibitorer |
| CN113149977A (zh) | 2020-01-22 | 2021-07-23 | 苏州爱科百发生物医药技术有限公司 | 一类呼吸道合胞病毒抑制剂的合成与用途 |
-
2020
- 2020-01-22 CN CN202010075139.8A patent/CN113149977A/zh not_active Withdrawn
-
2021
- 2021-01-21 KR KR1020227028783A patent/KR20220130761A/ko not_active Withdrawn
- 2021-01-21 EP EP21744323.3A patent/EP4095136A4/en active Pending
- 2021-01-21 CN CN202180010637.7A patent/CN115023423B/zh active Active
- 2021-01-21 US US17/790,987 patent/US12582661B2/en active Active
- 2021-01-21 WO PCT/CN2021/073042 patent/WO2021147947A1/zh not_active Ceased
- 2021-01-21 JP JP2022544247A patent/JP7726487B2/ja active Active
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