JP2023082086A5 - - Google Patents

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Publication number
JP2023082086A5
JP2023082086A5 JP2023052465A JP2023052465A JP2023082086A5 JP 2023082086 A5 JP2023082086 A5 JP 2023082086A5 JP 2023052465 A JP2023052465 A JP 2023052465A JP 2023052465 A JP2023052465 A JP 2023052465A JP 2023082086 A5 JP2023082086 A5 JP 2023082086A5
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JP
Japan
Prior art keywords
crystalline form
powder
ray diffraction
pharmaceutical composition
composition
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JP2023052465A
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English (en)
Japanese (ja)
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JP7763203B2 (ja
JP2023082086A (ja
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Priority claimed from JP2019538551A external-priority patent/JP7253491B2/ja
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JP2023052465A 2016-09-29 2023-03-28 キナーゼ阻害剤化合物の結晶多形、それを含む医薬組成物及びその製造方法と応用 Active JP7763203B2 (ja)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
CN201610866253 2016-09-29
CN201610866253.6 2016-09-29
JP2019538551A JP7253491B2 (ja) 2016-09-29 2017-09-29 キナーゼ阻害剤化合物の結晶多形、それを含む医薬組成物及びその製造方法と応用
PCT/CN2017/104506 WO2018059556A1 (zh) 2016-09-29 2017-09-29 激酶抑制剂化合物的多晶型、含其的药物组合物及其制备方法和应用

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
JP2019538551A Division JP7253491B2 (ja) 2016-09-29 2017-09-29 キナーゼ阻害剤化合物の結晶多形、それを含む医薬組成物及びその製造方法と応用

Publications (3)

Publication Number Publication Date
JP2023082086A JP2023082086A (ja) 2023-06-13
JP2023082086A5 true JP2023082086A5 (enExample) 2023-07-28
JP7763203B2 JP7763203B2 (ja) 2025-10-31

Family

ID=61763329

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2019538551A Active JP7253491B2 (ja) 2016-09-29 2017-09-29 キナーゼ阻害剤化合物の結晶多形、それを含む医薬組成物及びその製造方法と応用
JP2023052465A Active JP7763203B2 (ja) 2016-09-29 2023-03-28 キナーゼ阻害剤化合物の結晶多形、それを含む医薬組成物及びその製造方法と応用

Family Applications Before (1)

Application Number Title Priority Date Filing Date
JP2019538551A Active JP7253491B2 (ja) 2016-09-29 2017-09-29 キナーゼ阻害剤化合物の結晶多形、それを含む医薬組成物及びその製造方法と応用

Country Status (17)

Country Link
US (3) US11053224B2 (enExample)
EP (1) EP3502105B8 (enExample)
JP (2) JP7253491B2 (enExample)
KR (1) KR102289684B1 (enExample)
CN (1) CN108884080B (enExample)
AU (1) AU2017336889B2 (enExample)
CA (2) CA3253105A1 (enExample)
EA (1) EA201990688A1 (enExample)
ES (1) ES2914294T3 (enExample)
IL (2) IL265266B2 (enExample)
MY (1) MY194364A (enExample)
PH (1) PH12019500681A1 (enExample)
PL (1) PL3502105T3 (enExample)
SG (1) SG11201901962QA (enExample)
TW (1) TWI647224B (enExample)
WO (1) WO2018059556A1 (enExample)
ZA (1) ZA201901717B (enExample)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA3253105A1 (en) * 2016-09-29 2025-07-08 Equinox Sciences, Llc. POLYMORPHIC FORM OF A KINASE INHIBITOR COMPOUND, PHARMACEUTICAL COMPOSITION, CONTAINER, PREPARATION PROCESS AND USE
KR102195348B1 (ko) 2018-11-15 2020-12-24 에이치케이이노엔 주식회사 단백질 키나제 억제제로서의 신규 화합물 및 이를 포함하는 약제학적 조성물
TW202202138A (zh) 2020-03-25 2022-01-16 美商歐克萊製藥公司 含有酪胺酸激酶抑制劑之眼用植入物
WO2022056392A1 (en) 2020-09-14 2022-03-17 EyePoint Pharmaceuticals, Inc. Bioerodible ocular drug delivery insert and therapeutic method
CA3212253A1 (en) * 2021-03-16 2022-09-22 Young Ju Kim Crystalline form of heterocyclic compound as protein kinase inhibitor
JP7138982B1 (ja) 2021-09-24 2022-09-20 東海物産株式会社 アンセリンの結晶及びその製造方法
JP2025508127A (ja) 2022-03-11 2025-03-21 アイポイント ファーマシューティカルズ, インコーポレイテッド 眼薬物送達インサートを投与することによる加齢黄斑変性症の予防方法
IL315333A (en) 2022-03-11 2024-10-01 Eyepoint Pharmaceuticals Inc A continuous dosing regimen to treat the condition of the eye
WO2023173095A1 (en) 2022-03-11 2023-09-14 EyePoint Pharmaceuticals, Inc. Method of treating wet age-related macular degeneration
CN120897764A (zh) 2023-04-11 2025-11-04 视尔普斯眼科公司 包含阿西替尼多晶型物iv的眼部植入物
CN117143083B (zh) * 2023-08-30 2026-02-27 沈阳药科大学 VEGFR抑制剂Vorolanib的合成方法

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1434774A1 (en) * 2001-10-10 2004-07-07 Sugen, Inc. 3-(4-substituted heterocyclyl)-pyrrol-2-ylmethylidene)-2-indolinone derivatives as protein kinase inhibitors
KR101507375B1 (ko) 2006-09-15 2015-04-07 엑스커버리 홀딩 컴퍼니 엘엘씨 키나아제 억제제 화합물
US20110026367A1 (en) * 2007-05-07 2011-02-03 Baumer Electric Ag Acoustic Transducer
US20100256392A1 (en) * 2007-11-21 2010-10-07 Teva Pharmaceutical Industries Ltd. Polymorphs of sunitinib base and processes for preparation thereof
US8466190B2 (en) * 2008-04-16 2013-06-18 Natco Pharma Limited Polymorphic forms of Sunitinib base
RU2468022C2 (ru) 2008-05-23 2012-11-27 Шанхай Инститьют Оф Фармасьютикал Индастри Производные дигидроиндолона
EP2186809A1 (en) 2008-11-13 2010-05-19 LEK Pharmaceuticals D.D. New crystal form of sunitinib malate
EP2264027A1 (en) 2009-05-27 2010-12-22 Ratiopharm GmbH Process for the preparation of N-[2-(Diethylamino)ethyl]-5-[(5-fluoro-1,2-dihydro-2-oxo-3H-indol-3-ylidene) methyl]-2,4-dimethyl-1H-pyrrole-3-carboxamide
CN106928114B (zh) * 2015-12-31 2020-07-28 韶远科技(上海)有限公司 含有脲基的环状手性氨基类化合物及其可放大工艺和用途
CA3253105A1 (en) * 2016-09-29 2025-07-08 Equinox Sciences, Llc. POLYMORPHIC FORM OF A KINASE INHIBITOR COMPOUND, PHARMACEUTICAL COMPOSITION, CONTAINER, PREPARATION PROCESS AND USE

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