JP2023036007A5 - - Google Patents
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- Publication number
- JP2023036007A5 JP2023036007A5 JP2022136673A JP2022136673A JP2023036007A5 JP 2023036007 A5 JP2023036007 A5 JP 2023036007A5 JP 2022136673 A JP2022136673 A JP 2022136673A JP 2022136673 A JP2022136673 A JP 2022136673A JP 2023036007 A5 JP2023036007 A5 JP 2023036007A5
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- alkoxy
- group
- pharmaceutically acceptable
- acceptable salt
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2024074339A JP2024112817A (ja) | 2021-08-31 | 2024-05-01 | 6-アミノピラゾロピリミジン化合物及びその医薬用途 |
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2021141253 | 2021-08-31 | ||
| JP2021141253 | 2021-08-31 | ||
| JP2022068967 | 2022-04-19 | ||
| JP2022068967 | 2022-04-19 |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2024074339A Division JP2024112817A (ja) | 2021-08-31 | 2024-05-01 | 6-アミノピラゾロピリミジン化合物及びその医薬用途 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2023036007A JP2023036007A (ja) | 2023-03-13 |
| JP2023036007A5 true JP2023036007A5 (enExample) | 2024-01-11 |
| JP7483810B2 JP7483810B2 (ja) | 2024-05-15 |
Family
ID=85411220
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2022136673A Active JP7483810B2 (ja) | 2021-08-31 | 2022-08-30 | 6-アミノピラゾロピリミジン化合物及びその医薬用途 |
| JP2024074339A Withdrawn JP2024112817A (ja) | 2021-08-31 | 2024-05-01 | 6-アミノピラゾロピリミジン化合物及びその医薬用途 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2024074339A Withdrawn JP2024112817A (ja) | 2021-08-31 | 2024-05-01 | 6-アミノピラゾロピリミジン化合物及びその医薬用途 |
Country Status (15)
| Country | Link |
|---|---|
| US (1) | US20240287079A1 (enExample) |
| EP (1) | EP4397663A4 (enExample) |
| JP (2) | JP7483810B2 (enExample) |
| KR (1) | KR20240055035A (enExample) |
| AR (1) | AR126912A1 (enExample) |
| AU (1) | AU2022340126A1 (enExample) |
| CA (1) | CA3229401A1 (enExample) |
| CL (1) | CL2024000581A1 (enExample) |
| CO (1) | CO2024002515A2 (enExample) |
| IL (1) | IL310062A (enExample) |
| MX (1) | MX2024002609A (enExample) |
| PE (1) | PE20240882A1 (enExample) |
| TW (1) | TW202328134A (enExample) |
| WO (1) | WO2023032987A1 (enExample) |
| ZA (1) | ZA202400656B (enExample) |
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AR130318A1 (es) * | 2022-08-29 | 2024-11-27 | Japan Tobacco Inc | Compuestos de pirazolopirimidina y su uso médico |
| EP4671246A1 (en) * | 2023-02-24 | 2025-12-31 | Japan Tobacco Inc. | COMPOSITE OF 6-ALCOXYPYRAZOLOPYRIMIDINE AND ITS PHARMACEUTICAL USE |
| TW202448887A (zh) * | 2023-02-24 | 2024-12-16 | 日商日本煙草產業股份有限公司 | 取代吡唑并嘧啶化合物及其醫藥用途 |
| KR20250170647A (ko) | 2023-04-14 | 2025-12-05 | 다케다 야쿠힌 고교 가부시키가이샤 | Nlrp3 억제제로서의 피라졸로피리미딘 유도체 |
| AU2024280075A1 (en) | 2023-06-02 | 2025-12-11 | Merck Sharp & Dohme Llc | 5,6-Unsaturated Bicyclic Heterocycles Useful as Inhibitors of Nod-Like Receptor Protein 3 |
| TW202535370A (zh) * | 2023-12-14 | 2025-09-16 | 美商默沙東有限責任公司 | 作為nod樣受體蛋白3抑制劑之吲唑衍生物 |
| US20250223290A1 (en) * | 2023-12-14 | 2025-07-10 | Merck Sharp & Dohme Llc | Azaindazole derivatives useful as inhibitors of nod-like receptor protein 3 |
| WO2025140708A1 (zh) * | 2023-12-31 | 2025-07-03 | 杭州百新生物医药科技有限公司 | 吡唑并嘧啶类化合物及其医药用途 |
| TW202545527A (zh) | 2024-01-16 | 2025-12-01 | 英商諾得瑟拉公司 | Nlrp3及glp-1a組合療法 |
| WO2026164254A1 (ja) * | 2025-01-31 | 2026-08-06 | 塩野義製薬株式会社 | ピラゾロピリミジン化合物の製造方法及びその合成中間体 |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU2012244550C1 (en) * | 2011-04-21 | 2017-06-22 | Origenis Gmbh | Pyrazolo [4, 3-d] pyrimidines useful as kinase inhibitors |
| WO2017205766A1 (en) * | 2016-05-27 | 2017-11-30 | Pharmacyclics Llc | Inhibitors of interleukin-1 receptor-associated kinase |
| KR102815870B1 (ko) * | 2019-01-14 | 2025-05-30 | 인네이트 튜머 이뮤니티, 인코포레이티드 | 암의 치료에 사용하기 위한 헤테로시클릭 nlrp3 조정제 |
| CN113286786A (zh) * | 2019-01-14 | 2021-08-20 | 先天肿瘤免疫公司 | Nlrp3调节剂 |
-
2022
- 2022-08-30 KR KR1020247010356A patent/KR20240055035A/ko active Pending
- 2022-08-30 TW TW111132739A patent/TW202328134A/zh unknown
- 2022-08-30 AR ARP220102331A patent/AR126912A1/es unknown
- 2022-08-30 CA CA3229401A patent/CA3229401A1/en active Pending
- 2022-08-30 WO PCT/JP2022/032606 patent/WO2023032987A1/ja not_active Ceased
- 2022-08-30 IL IL310062A patent/IL310062A/en unknown
- 2022-08-30 US US18/566,623 patent/US20240287079A1/en active Pending
- 2022-08-30 PE PE2024000332A patent/PE20240882A1/es unknown
- 2022-08-30 MX MX2024002609A patent/MX2024002609A/es unknown
- 2022-08-30 JP JP2022136673A patent/JP7483810B2/ja active Active
- 2022-08-30 AU AU2022340126A patent/AU2022340126A1/en active Pending
- 2022-08-30 EP EP22864569.3A patent/EP4397663A4/en active Pending
-
2024
- 2024-01-18 ZA ZA2024/00656A patent/ZA202400656B/en unknown
- 2024-02-26 CL CL2024000581A patent/CL2024000581A1/es unknown
- 2024-02-28 CO CONC2024/0002515A patent/CO2024002515A2/es unknown
- 2024-05-01 JP JP2024074339A patent/JP2024112817A/ja not_active Withdrawn
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