JP2023021316A5 - - Google Patents

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Publication number
JP2023021316A5
JP2023021316A5 JP2022199375A JP2022199375A JP2023021316A5 JP 2023021316 A5 JP2023021316 A5 JP 2023021316A5 JP 2022199375 A JP2022199375 A JP 2022199375A JP 2022199375 A JP2022199375 A JP 2022199375A JP 2023021316 A5 JP2023021316 A5 JP 2023021316A5
Authority
JP
Japan
Prior art keywords
alkyl
pyridyl
trifluoromethyl
phenyl
pyridin
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
JP2022199375A
Other languages
English (en)
Japanese (ja)
Other versions
JP2023021316A (ja
Filing date
Publication date
Priority claimed from JP2020510114A external-priority patent/JP7201260B2/ja
Application filed filed Critical
Publication of JP2023021316A publication Critical patent/JP2023021316A/ja
Publication of JP2023021316A5 publication Critical patent/JP2023021316A5/ja
Ceased legal-status Critical Current

Links

JP2022199375A 2017-08-23 2022-12-14 ピリジンアミン-ピリドンおよびピリミジンアミン-ピリドン化合物 Ceased JP2023021316A (ja)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
EP17187560 2017-08-23
EP17187560.2 2017-08-23
JP2020510114A JP7201260B2 (ja) 2017-08-23 2018-08-23 ピリジンアミン-ピリドンおよびピリミジンアミン-ピリドン化合物
PCT/EP2018/072790 WO2019038389A1 (en) 2017-08-23 2018-08-23 PYRIDINAMINE-PYRIDONE AND PYRIMIDINAMINE-PYRIDONE COMPOUNDS

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
JP2020510114A Division JP7201260B2 (ja) 2017-08-23 2018-08-23 ピリジンアミン-ピリドンおよびピリミジンアミン-ピリドン化合物

Publications (2)

Publication Number Publication Date
JP2023021316A JP2023021316A (ja) 2023-02-10
JP2023021316A5 true JP2023021316A5 (enExample) 2023-09-26

Family

ID=59686885

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2020510114A Active JP7201260B2 (ja) 2017-08-23 2018-08-23 ピリジンアミン-ピリドンおよびピリミジンアミン-ピリドン化合物
JP2022199375A Ceased JP2023021316A (ja) 2017-08-23 2022-12-14 ピリジンアミン-ピリドンおよびピリミジンアミン-ピリドン化合物

Family Applications Before (1)

Application Number Title Priority Date Filing Date
JP2020510114A Active JP7201260B2 (ja) 2017-08-23 2018-08-23 ピリジンアミン-ピリドンおよびピリミジンアミン-ピリドン化合物

Country Status (21)

Country Link
US (2) US11208423B2 (enExample)
EP (2) EP3672948B1 (enExample)
JP (2) JP7201260B2 (enExample)
KR (1) KR102730753B1 (enExample)
CN (3) CN111094271B (enExample)
AU (2) AU2018320418B2 (enExample)
CA (1) CA3073129A1 (enExample)
DK (1) DK3672948T3 (enExample)
ES (1) ES2929424T3 (enExample)
FI (1) FI3672948T3 (enExample)
HR (1) HRP20221454T1 (enExample)
HU (1) HUE060805T2 (enExample)
IL (3) IL302293A (enExample)
LT (1) LT3672948T (enExample)
PL (1) PL3672948T3 (enExample)
PT (1) PT3672948T (enExample)
RS (1) RS63795B1 (enExample)
SI (1) SI3672948T1 (enExample)
SM (1) SMT202200493T1 (enExample)
TW (2) TW202325302A (enExample)
WO (1) WO2019038389A1 (enExample)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2929424T3 (es) * 2017-08-23 2022-11-29 Sprint Bioscience Ab Compuestos de piridinamina-piridona y pirimidinamina-piridona
EP3728230A1 (en) 2017-12-22 2020-10-28 Ravenna Pharmaceuticals, Inc. Aryl-bipyridine amine derivatives as phosphatidylinositol phosphate kinase inhibitors
AU2020398215A1 (en) * 2019-12-04 2022-06-16 Chdi Foundation, Inc. ATM kinase inhibitors and compositions and methods of use thereof
WO2022115562A1 (en) 2020-11-25 2022-06-02 Deciphera Pharmaceuticals, Llc Morpholino derivatives as vsp34 inhibitors for use in the treatment of a viral infection
US20220184093A1 (en) * 2020-11-25 2022-06-16 Deciphera Pharmaceuticals, Llc Anti-viral activity of vps34 inhibitors
WO2022115546A1 (en) 2020-11-25 2022-06-02 Deciphera Pharmaceuticals, Llc Anti-viral activity of vps34 inhibitors
US20240277852A1 (en) * 2021-05-20 2024-08-22 Dana-Farber Cancer Institute, Inc. Inhibitors and degraders of pip4k protein
US20250127790A1 (en) * 2021-08-13 2025-04-24 Deciphera Pharmaceuticals, Llc Combination therapy using vps34 inhibitors
AU2023255558A1 (en) * 2022-04-22 2024-10-31 Vertex Pharmaceuticals Incorporated Heteroaryl compounds for the treatment of pain
US20250236609A1 (en) * 2023-12-13 2025-07-24 Deciphera Pharmaceuticals, Llc Vps34 inhibitors and methods of use thereof

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP4606161B2 (ja) * 2002-05-21 2011-01-05 アムジエン・インコーポレーテツド 置換複素環式化合物および使用方法
EA201390917A1 (ru) * 2010-12-21 2013-12-30 Новартис Аг Дигетероарильные соединения в качестве ингибиторов vps34
HUE024504T2 (en) 2010-12-23 2016-01-28 Sanofi Sa Pyrimidine derivatives, a process for their preparation and their use in medicine
GB201120317D0 (en) 2011-11-24 2012-01-04 Queen Mary & Westfield College Screening method
FR2992314B1 (fr) 2012-06-22 2015-10-16 Sanofi Sa Nouveaux derives de 2,3-dihydro-1h-imidazo{1,2-a}pyrimidin-5-one et 1,2,3,4-tetrahydro-pyrimido{1,2-a}pyrimidin-6-one comportant une morpholine substituee, leur preparation et leur utilisation pharmaceutique
JP2017502092A (ja) 2014-01-14 2017-01-19 ミレニアム ファーマシューティカルズ, インコーポレイテッドMillennium Pharmaceuticals, Inc. ヘテロアリール及びその使用
TN2016000270A1 (en) 2014-01-14 2017-10-06 Millennium Pharm Inc Heteroaryls and uses thereof.
MA39822A (fr) 2014-04-03 2018-02-06 Janssen Pharmaceutica Nv Dérivés de pyrimidine bicycle
MA39823A (fr) 2014-04-03 2018-01-09 Janssen Pharmaceutica Nv Dérivés de pyridine macrocyclique
WO2016001789A1 (en) 2014-06-30 2016-01-07 Pfizer Inc. Pyrimidine derivatives as pi3k inhibitors for use in the treatment of cancer
CA3015045A1 (en) 2016-02-19 2017-08-24 Sprint Bioscience Ab 6-aryl-4-morpholin-1-ylpyridone compounds useful for the treatment of cancer and diabetes
US11179399B2 (en) 2016-02-19 2021-11-23 Sprint Bioscience Ab 6-heterocyclyl-4-morpholin-4-ylpyridine-2-one compounds useful for the treatment of cancer and diabetes
ES2929424T3 (es) * 2017-08-23 2022-11-29 Sprint Bioscience Ab Compuestos de piridinamina-piridona y pirimidinamina-piridona

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