JP2023021277A5 - - Google Patents

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Publication number
JP2023021277A5
JP2023021277A5 JP2022198545A JP2022198545A JP2023021277A5 JP 2023021277 A5 JP2023021277 A5 JP 2023021277A5 JP 2022198545 A JP2022198545 A JP 2022198545A JP 2022198545 A JP2022198545 A JP 2022198545A JP 2023021277 A5 JP2023021277 A5 JP 2023021277A5
Authority
JP
Japan
Prior art keywords
pyridin
pyrrolo
trifluoromethyl
alkyl
phenyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
JP2022198545A
Other languages
English (en)
Japanese (ja)
Other versions
JP2023021277A (ja
Filing date
Publication date
Priority claimed from PCT/EP2018/072785 external-priority patent/WO2019038384A1/en
Application filed filed Critical
Publication of JP2023021277A publication Critical patent/JP2023021277A/ja
Publication of JP2023021277A5 publication Critical patent/JP2023021277A5/ja
Ceased legal-status Critical Current

Links

JP2022198545A 2017-08-23 2022-12-13 アザインドリルピリドンおよびジアザインドリルピリドン化合物 Ceased JP2023021277A (ja)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
EP17187519.8 2017-08-23
EP17187519 2017-08-23
PCT/EP2018/072785 WO2019038384A1 (en) 2017-08-23 2018-08-23 AZAINDOLYLPYRIDONE AND DIAZAINDOLYLPYRIDONE COMPOUNDS
JP2020510099A JP7199738B2 (ja) 2017-08-23 2018-08-23 アザインドリルピリドンおよびジアザインドリルピリドン化合物

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
JP2020510099A Division JP7199738B2 (ja) 2017-08-23 2018-08-23 アザインドリルピリドンおよびジアザインドリルピリドン化合物

Publications (2)

Publication Number Publication Date
JP2023021277A JP2023021277A (ja) 2023-02-10
JP2023021277A5 true JP2023021277A5 (enExample) 2023-09-25

Family

ID=59686871

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2020510099A Active JP7199738B2 (ja) 2017-08-23 2018-08-23 アザインドリルピリドンおよびジアザインドリルピリドン化合物
JP2022198545A Ceased JP2023021277A (ja) 2017-08-23 2022-12-13 アザインドリルピリドンおよびジアザインドリルピリドン化合物

Family Applications Before (1)

Application Number Title Priority Date Filing Date
JP2020510099A Active JP7199738B2 (ja) 2017-08-23 2018-08-23 アザインドリルピリドンおよびジアザインドリルピリドン化合物

Country Status (20)

Country Link
US (2) US11498919B2 (enExample)
EP (2) EP4001278A1 (enExample)
JP (2) JP7199738B2 (enExample)
KR (1) KR102731945B1 (enExample)
CN (3) CN116589462A (enExample)
AU (1) AU2018321135B2 (enExample)
CY (1) CY1124818T1 (enExample)
DK (1) DK3672967T3 (enExample)
ES (1) ES2902346T3 (enExample)
HR (1) HRP20211999T1 (enExample)
HU (1) HUE057818T2 (enExample)
IL (3) IL302355A (enExample)
LT (1) LT3672967T (enExample)
PL (1) PL3672967T3 (enExample)
PT (1) PT3672967T (enExample)
RS (1) RS62785B1 (enExample)
SI (1) SI3672967T1 (enExample)
SM (1) SMT202100718T1 (enExample)
TW (2) TWI785101B (enExample)
WO (1) WO2019038384A1 (enExample)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PT3672967T (pt) * 2017-08-23 2021-12-28 Sprint Bioscience Ab Compostos de azaindolilpiridona e diazaindolilpiridona
EP4251156A1 (en) 2020-11-25 2023-10-04 Deciphera Pharmaceuticals, LLC Anti-viral activity of vps34 inhibitors
CA3199999A1 (en) 2020-11-25 2022-06-02 Deciphera Pharmaceuticals, Llc Morpholino derivatives as vsp34 inhibitors for use in the treatment of a viral infection

Family Cites Families (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1154024B (it) * 1982-09-22 1987-01-21 Lepetit Spa Derivati pridinici e procedimento per la loro produzione
US8921376B2 (en) 2005-05-20 2014-12-30 Vertex Pharmaceuticals Incorporated Pyrrolopyridines useful as inhibitors of protein kinase
EP2320895A2 (en) * 2008-07-03 2011-05-18 Exelixis, Inc. Cdk modulators
ES2488219T3 (es) * 2010-04-19 2014-08-26 Abbvie Inc. Pirrolopiridinas como inhibidores de quinasas
CN103270026A (zh) 2010-12-21 2013-08-28 诺瓦提斯公司 作为vps34抑制剂的联-杂芳基化合物
PL2655375T3 (pl) 2010-12-23 2015-05-29 Sanofi Sa Pochodne pirymidynonu, ich wytwarzanie i ich farmaceutyczne zastosowanie
GB201120317D0 (en) 2011-11-24 2012-01-04 Queen Mary & Westfield College Screening method
CN103450152B (zh) 2012-06-04 2015-11-18 济南海乐医药技术开发有限公司 基于吲唑、吲哚或氮杂吲唑、氮杂吲哚的双芳基脲类结构抗肿瘤药物
FR2992314B1 (fr) 2012-06-22 2015-10-16 Sanofi Sa Nouveaux derives de 2,3-dihydro-1h-imidazo{1,2-a}pyrimidin-5-one et 1,2,3,4-tetrahydro-pyrimido{1,2-a}pyrimidin-6-one comportant une morpholine substituee, leur preparation et leur utilisation pharmaceutique
US10202373B2 (en) * 2014-01-14 2019-02-12 Millennium Pharmaceuticals, Inc. Heteroaryls and uses thereof
WO2015108861A1 (en) 2014-01-14 2015-07-23 Millennium Pharmaceuticals, Inc. Heteroaryls and uses thereof
MA39823A (fr) 2014-04-03 2018-01-09 Janssen Pharmaceutica Nv Dérivés de pyridine macrocyclique
MA39822A (fr) 2014-04-03 2018-02-06 Janssen Pharmaceutica Nv Dérivés de pyrimidine bicycle
WO2017140841A1 (en) 2016-02-19 2017-08-24 Sprint Bioscience Ab 6-aryl-4-morpholin-1-ylpyridone compounds useful for the treatment of cancer and diabetes
SMT202000529T1 (it) 2016-02-19 2020-11-10 Sprint Bioscience Ab Composti di 6-eterociclil-4-morfolina-4-ilpiridin-2-one utili per il trattamento di cancro e diabete
PT3672967T (pt) * 2017-08-23 2021-12-28 Sprint Bioscience Ab Compostos de azaindolilpiridona e diazaindolilpiridona

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