JP2022553056A5 - - Google Patents

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Publication number
JP2022553056A5
JP2022553056A5 JP2022523585A JP2022523585A JP2022553056A5 JP 2022553056 A5 JP2022553056 A5 JP 2022553056A5 JP 2022523585 A JP2022523585 A JP 2022523585A JP 2022523585 A JP2022523585 A JP 2022523585A JP 2022553056 A5 JP2022553056 A5 JP 2022553056A5
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JP
Japan
Prior art keywords
compound according
group
sirna
formula
sirna28
Prior art date
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Granted
Application number
JP2022523585A
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English (en)
Japanese (ja)
Other versions
JP2022553056A (ja
JP7668032B2 (ja
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Priority claimed from PCT/US2020/057185 external-priority patent/WO2021081420A2/en
Publication of JP2022553056A publication Critical patent/JP2022553056A/ja
Publication of JP2022553056A5 publication Critical patent/JP2022553056A5/ja
Application granted granted Critical
Publication of JP7668032B2 publication Critical patent/JP7668032B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2022523585A 2019-10-24 2020-10-23 先端巨大症を処置するためのコンジュゲート及び方法 Active JP7668032B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201962925659P 2019-10-24 2019-10-24
US62/925,659 2019-10-24
PCT/US2020/057185 WO2021081420A2 (en) 2019-10-24 2020-10-23 Conjugates and methods for treating acromegaly

Publications (3)

Publication Number Publication Date
JP2022553056A JP2022553056A (ja) 2022-12-21
JP2022553056A5 true JP2022553056A5 (https=) 2023-10-27
JP7668032B2 JP7668032B2 (ja) 2025-04-24

Family

ID=75620892

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2022523585A Active JP7668032B2 (ja) 2019-10-24 2020-10-23 先端巨大症を処置するためのコンジュゲート及び方法

Country Status (9)

Country Link
US (1) US20220288214A1 (https=)
EP (1) EP4048801A4 (https=)
JP (1) JP7668032B2 (https=)
CN (1) CN114616339A (https=)
AU (1) AU2020371736A1 (https=)
BR (1) BR112022007725A2 (https=)
CA (1) CA3158917A1 (https=)
IL (1) IL292391A (https=)
WO (1) WO2021081420A2 (https=)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA3020585A1 (en) * 2016-04-11 2017-10-19 Arbutus Biopharma Corporation Targeted nucleic acid conjugate compositions

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2322651A1 (en) * 2004-05-14 2011-05-18 Rosetta Genomics Ltd MicroRNAs and uses thereof
CA2917229A1 (en) * 2013-07-02 2015-01-08 Isis Pharmaceuticals, Inc. Modulators of growth hormone receptor
BR112016022742B1 (pt) * 2014-05-01 2022-06-14 Ionis Pharmaceuticals, Inc Composto químico, composição compreendendo o composto e uso dos mesmos
WO2015179693A1 (en) * 2014-05-22 2015-11-26 Isis Pharmaceuticals, Inc. Conjugated antisense compounds and their use
EP3151839A4 (en) * 2014-06-06 2018-02-28 Ionis Pharmaceuticals, Inc. Compositions and methods for enhanced intestinal absorption of conjugated oligomeric compounds
EP3228326A1 (en) 2016-04-05 2017-10-11 Silence Therapeutics GmbH Nucleic acid linked to a trivalent glycoconjugate
DK3607069T3 (da) 2017-04-05 2022-11-21 Silence Therapeutics Gmbh Produkter og sammensætninger
WO2018185253A1 (en) * 2017-04-05 2018-10-11 Silence Therapeutics Gmbh Ligand modified double-stranded nucleic acids
JP7406793B2 (ja) * 2017-06-23 2023-12-28 ユニバーシティー オブ マサチューセッツ 2テイル自己デリバリー型siRNAおよび関連方法
EP3775209A1 (en) * 2018-04-05 2021-02-17 Silence Therapeutics GmbH Sirnas with at least two ligands at different ends

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