JP2022552445A5 - - Google Patents
Info
- Publication number
- JP2022552445A5 JP2022552445A5 JP2022546591A JP2022546591A JP2022552445A5 JP 2022552445 A5 JP2022552445 A5 JP 2022552445A5 JP 2022546591 A JP2022546591 A JP 2022546591A JP 2022546591 A JP2022546591 A JP 2022546591A JP 2022552445 A5 JP2022552445 A5 JP 2022552445A5
- Authority
- JP
- Japan
- Prior art keywords
- optionally substituted
- alkyl
- group
- pharmaceutically acceptable
- occurrence
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201962911653P | 2019-10-07 | 2019-10-07 | |
| US62/911,653 | 2019-10-07 | ||
| PCT/US2020/054373 WO2021071821A1 (en) | 2019-10-07 | 2020-10-06 | Arylmethylene aromatic compounds as kv1.3 potassium shaker channel blockers |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2022552445A JP2022552445A (ja) | 2022-12-15 |
| JP2022552445A5 true JP2022552445A5 (cg-RX-API-DMAC10.html) | 2024-09-06 |
| JP7697954B2 JP7697954B2 (ja) | 2025-06-24 |
Family
ID=75438313
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2022546591A Active JP7697954B2 (ja) | 2019-10-07 | 2020-10-06 | Ｋｖ１．３カリウムシェーカーチャネル遮断薬としてのアリールメチレン芳香族化合物 |
Country Status (11)
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN116782894A (zh) | 2020-10-06 | 2023-09-19 | D.E.肖研究有限责任公司 | 作为Kv1.3钾Shaker通道阻断剂的内酰胺化合物 |
| EP4253383A4 (en) * | 2020-12-31 | 2024-07-17 | Tsinghua University | PYRIDINE-2-AMINE DERIVATIVE, PHARMACEUTICAL COMPOSITION AND ASSOCIATED USE |
| EP4308095A4 (en) | 2021-03-15 | 2025-02-19 | Maze Therapeutics, Inc. | GLYCOGEN SYNTHASE 1 (GYS1) INHIBITORS AND METHODS OF USE THEREOF |
| CN115703734B (zh) * | 2021-08-05 | 2024-08-09 | 重庆文理学院 | 二芳基甲基吡啶类化合物及其制备方法和应用 |
| TW202345806A (zh) | 2022-03-31 | 2023-12-01 | 美商艾伯維有限公司 | 噻唑并〔５，４－ｂ〕吡啶ｍａｌｔ－１抑制劑 |
| CN120202194A (zh) | 2022-11-16 | 2025-06-24 | 巴斯夫欧洲公司 | 作为杀真菌剂的取代的四氢苯并二氮杂䓬 |
| EP4619392A1 (en) | 2022-11-16 | 2025-09-24 | Basf Se | Substituted benzodiazepines as fungicides |
| JP2026509904A (ja) | 2023-03-17 | 2026-03-25 | ビーエーエスエフ ソシエタス・ヨーロピア | 植物病原真菌を駆除するための置換ピリジル／ピラジジルジヒドロベンゾチアゼピン化合物 |
| WO2025029769A1 (en) | 2023-07-31 | 2025-02-06 | Eli Lilly And Company | Solid forms of a kv1.3 potassium shaker channel blockers and method of using the same |
| WO2026057374A1 (en) | 2024-09-11 | 2026-03-19 | Basf Se | Fungicidal mixture comprising substituted pyridyl/pyrazidyl dihydrobenzothiazepine compounds |
Family Cites Families (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CH540009A (de) * | 1970-07-23 | 1973-09-28 | Ciba Geigy Ag | Verwendung von Monohydroxyphenylcarbinolen zum antimikrobiellen Ausrüsten bzw. zum Schützen von textilen Materialien gegen schädliche Mikroorganismen |
| JPH07309837A (ja) * | 1993-04-28 | 1995-11-28 | Takeda Chem Ind Ltd | ピリジン誘導体、その製造法および剤 |
| JPH09278757A (ja) * | 1996-04-15 | 1997-10-28 | Takeda Chem Ind Ltd | ヒドラゾン誘導体および剤 |
| TW467902B (en) * | 1996-07-31 | 2001-12-11 | Bristol Myers Squibb Co | Diphenyl heterocycles as potassium channel modulators |
| EP1056730A4 (en) * | 1998-01-29 | 2003-01-02 | Bristol Myers Squibb Co | Diaryl-1,3,4-oxadiazolone benzoate |
| EP1838690A2 (en) * | 2004-12-21 | 2007-10-03 | Devgen N.V. | Compounds with kv4 ion channel activity |
| AU2008307075B2 (en) * | 2007-10-04 | 2012-05-17 | Bionomics Limited | Novel aryl potassium channel blockers and uses thereof |
| GB0815784D0 (en) * | 2008-08-29 | 2008-10-08 | Xention Ltd | Novel potassium channel blockers |
| GB0909672D0 (en) * | 2009-06-04 | 2009-07-22 | Xention Discovery Ltd | Compounds |
| KR20130100300A (ko) * | 2010-08-27 | 2013-09-10 | 그뤼넨탈 게엠베하 | Ｋｃｎｑ２／３ 조절제로서의 치환된 ２-옥시-퀴놀린-３-카복스아미드 |
| EP2970153B1 (en) * | 2013-03-13 | 2018-02-21 | The United States of America, as represented by The Secretary of The Army, on behalf of Walter Reed Army Institute of Research | Triazine compounds and compositions thereof and methods for treating malaria and chemoprophylaxis |
| HRP20210472T1 (hr) * | 2015-08-27 | 2021-05-14 | Pfizer Inc. | Biciklički kondenzirani heteroarilni ili arilni spojevi kao modulatori irak4 |
| EP3490542A4 (en) * | 2016-07-26 | 2020-07-08 | Flagship Pioneering Innovations V, Inc. | NEUROMODULATION COMPOSITIONS AND RELATED THERAPEUTIC METHODS FOR THE TREATMENT OF CANCER BY MODULATION OF AN ANTI-CANCER RESPONSE |
-
2020
- 2020-10-06 KR KR1020227013504A patent/KR20220079879A/ko not_active Withdrawn
- 2020-10-06 WO PCT/US2020/054373 patent/WO2021071821A1/en not_active Ceased
- 2020-10-06 BR BR112022006242A patent/BR112022006242A2/pt not_active IP Right Cessation
- 2020-10-06 CA CA3157026A patent/CA3157026A1/en active Pending
- 2020-10-06 AU AU2020363366A patent/AU2020363366A1/en not_active Abandoned
- 2020-10-06 US US17/766,879 patent/US20230131535A1/en not_active Abandoned
- 2020-10-06 EP EP20875222.0A patent/EP4041230A4/en active Pending
- 2020-10-06 JP JP2022546591A patent/JP7697954B2/ja active Active
- 2020-10-06 CN CN202080084417.4A patent/CN114727992A/zh active Pending
- 2020-10-06 MX MX2022004168A patent/MX2022004168A/es unknown
-
2022
- 2022-03-27 IL IL291733A patent/IL291733A/en unknown