JP2022548602A5 - - Google Patents

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Publication number
JP2022548602A5
JP2022548602A5 JP2022516328A JP2022516328A JP2022548602A5 JP 2022548602 A5 JP2022548602 A5 JP 2022548602A5 JP 2022516328 A JP2022516328 A JP 2022516328A JP 2022516328 A JP2022516328 A JP 2022516328A JP 2022548602 A5 JP2022548602 A5 JP 2022548602A5
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JP
Japan
Prior art keywords
dihydro
pyridazin
acetamide
oxo
ethyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2022516328A
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English (en)
Japanese (ja)
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JP7566888B2 (ja
JP2022548602A (ja
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Priority claimed from PCT/US2020/050823 external-priority patent/WO2021055326A1/en
Publication of JP2022548602A publication Critical patent/JP2022548602A/ja
Publication of JP2022548602A5 publication Critical patent/JP2022548602A5/ja
Application granted granted Critical
Publication of JP7566888B2 publication Critical patent/JP7566888B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2022516328A 2019-09-16 2020-09-15 アゾール縮合ピリダジン-3(2h)-オン誘導体 Active JP7566888B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201962901052P 2019-09-16 2019-09-16
US62/901,052 2019-09-16
PCT/US2020/050823 WO2021055326A1 (en) 2019-09-16 2020-09-15 Azole-fused pyridazin-3(2h)-one derivatives

Publications (3)

Publication Number Publication Date
JP2022548602A JP2022548602A (ja) 2022-11-21
JP2022548602A5 true JP2022548602A5 (https=) 2023-09-25
JP7566888B2 JP7566888B2 (ja) 2024-10-15

Family

ID=72670806

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2022516328A Active JP7566888B2 (ja) 2019-09-16 2020-09-15 アゾール縮合ピリダジン-3(2h)-オン誘導体

Country Status (25)

Country Link
US (1) US12370192B2 (https=)
EP (1) EP4031552B1 (https=)
JP (1) JP7566888B2 (https=)
KR (1) KR102924294B1 (https=)
CN (1) CN114728975A (https=)
AR (1) AR119971A1 (https=)
AU (1) AU2020348675B2 (https=)
BR (1) BR112022004819A2 (https=)
CA (1) CA3150508A1 (https=)
CO (1) CO2022004684A2 (https=)
CR (1) CR20220160A (https=)
DO (1) DOP2022000057A (https=)
EC (1) ECSP22020159A (https=)
ES (1) ES2997267T3 (https=)
HR (1) HRP20250088T1 (https=)
HU (1) HUE069908T2 (https=)
IL (1) IL291181B2 (https=)
JO (1) JOP20220063A1 (https=)
MX (1) MX2022003177A (https=)
PE (1) PE20221341A1 (https=)
PH (1) PH12022550597A1 (https=)
PL (1) PL4031552T3 (https=)
RS (1) RS66463B1 (https=)
TW (1) TWI873185B (https=)
WO (1) WO2021055326A1 (https=)

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CN114149371B (zh) * 2021-11-26 2023-08-22 首都医科大学 四取代吡唑类化合物及其应用
CN116693545A (zh) * 2022-03-01 2023-09-05 上海科技大学 噻吩并含氮杂环类化合物、含其的药物组合物、其制备方法及其应用
CN116693536A (zh) * 2022-03-01 2023-09-05 上海科技大学 吡咯并三嗪酮类化合物、含其的药物组合物、其制备方法及其应用
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CN116063179A (zh) * 2023-02-20 2023-05-05 南京杰运医药科技有限公司 一种4-甲氧基乙酰乙酸甲酯的合成方法
WO2025119351A1 (zh) * 2023-12-08 2025-06-12 深圳湾实验室 Gpr139激动剂
WO2025124544A1 (zh) * 2023-12-14 2025-06-19 华润医药研究院(深圳)有限公司 3,4-二氢-2H-苯并[b][1,4]二氧杂环庚烷类化合物及其制备方法和医药用途
WO2025162441A1 (zh) * 2024-02-02 2025-08-07 上海科技大学 稠杂环类化合物与其制备方法、药物组合物及应用

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