JP2022538795A5 - - Google Patents

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Publication number
JP2022538795A5
JP2022538795A5 JP2021573885A JP2021573885A JP2022538795A5 JP 2022538795 A5 JP2022538795 A5 JP 2022538795A5 JP 2021573885 A JP2021573885 A JP 2021573885A JP 2021573885 A JP2021573885 A JP 2021573885A JP 2022538795 A5 JP2022538795 A5 JP 2022538795A5
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JP
Japan
Prior art keywords
methyl
pyrazine
fluorophenyl
difluoromethoxy
oxazolidine
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
JP2021573885A
Other languages
English (en)
Japanese (ja)
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JP2022538795A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/EP2020/066396 external-priority patent/WO2020249796A1/en
Publication of JP2022538795A publication Critical patent/JP2022538795A/ja
Publication of JP2022538795A5 publication Critical patent/JP2022538795A5/ja
Withdrawn legal-status Critical Current

Links

JP2021573885A 2019-06-14 2020-06-12 ピラジンカルバメート及びGluN2B受容体調節因子としての使用 Withdrawn JP2022538795A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201962861642P 2019-06-14 2019-06-14
US62/861,642 2019-06-14
PCT/EP2020/066396 WO2020249796A1 (en) 2019-06-14 2020-06-12 Pyrazine carbamates and their use as glun2b receptor modulators

Publications (2)

Publication Number Publication Date
JP2022538795A JP2022538795A (ja) 2022-09-06
JP2022538795A5 true JP2022538795A5 (enExample) 2023-06-21

Family

ID=71108570

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2021573885A Withdrawn JP2022538795A (ja) 2019-06-14 2020-06-12 ピラジンカルバメート及びGluN2B受容体調節因子としての使用

Country Status (10)

Country Link
US (1) US11459336B2 (enExample)
EP (1) EP3983072A1 (enExample)
JP (1) JP2022538795A (enExample)
KR (1) KR20220020915A (enExample)
CN (1) CN113950357A (enExample)
AU (1) AU2020290772A1 (enExample)
BR (1) BR112021023562A2 (enExample)
CA (1) CA3142998A1 (enExample)
MX (1) MX2021015511A (enExample)
WO (1) WO2020249796A1 (enExample)

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MX2021015511A (es) 2019-06-14 2022-01-31 Janssen Pharmaceutica Nv Carbamatos de pirazina y sus usos como moduladores del receptor glun2b.
CA3143103A1 (en) 2019-06-14 2020-12-17 Janssen Pharmaceutica Nv Pyridine carbamates and their use as glun2b receptor modulators
AU2020293642A1 (en) 2019-06-14 2022-01-20 Janssen Pharmaceutica Nv Substituted pyrazolo[4,3-b]pyridines and their use as GluN2B receptor modulators
TW202112774A (zh) 2019-06-14 2021-04-01 比利時商健生藥品公司 經取代之吡唑并-吡啶醯胺及其作為glun2b受體調節劑之用途
JP7667097B2 (ja) 2019-06-14 2025-04-22 ヤンセン ファーマシューティカ エヌ.ベー. 置換ピラゾロ-ピリジンアミド及びglun2b受容体調節因子としてのその使用
BR112021025141A2 (pt) 2019-06-14 2022-01-25 Janssen Pharmaceutica Nv Pirazolo-piridinas heteroaromáticas substituídas e seu uso como moduladores do receptor glun2b
CN114008052A (zh) 2019-06-14 2022-02-01 詹森药业有限公司 取代的吡唑并-吡嗪以及它们作为GluN2B受体调节剂的用途

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TW202112774A (zh) 2019-06-14 2021-04-01 比利時商健生藥品公司 經取代之吡唑并-吡啶醯胺及其作為glun2b受體調節劑之用途
MX2021015511A (es) 2019-06-14 2022-01-31 Janssen Pharmaceutica Nv Carbamatos de pirazina y sus usos como moduladores del receptor glun2b.
BR112021025141A2 (pt) 2019-06-14 2022-01-25 Janssen Pharmaceutica Nv Pirazolo-piridinas heteroaromáticas substituídas e seu uso como moduladores do receptor glun2b
CN114008052A (zh) 2019-06-14 2022-02-01 詹森药业有限公司 取代的吡唑并-吡嗪以及它们作为GluN2B受体调节剂的用途
AU2020293642A1 (en) 2019-06-14 2022-01-20 Janssen Pharmaceutica Nv Substituted pyrazolo[4,3-b]pyridines and their use as GluN2B receptor modulators
CA3143103A1 (en) 2019-06-14 2020-12-17 Janssen Pharmaceutica Nv Pyridine carbamates and their use as glun2b receptor modulators

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