JP2022536174A5 - - Google Patents

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Publication number
JP2022536174A5
JP2022536174A5 JP2021573717A JP2021573717A JP2022536174A5 JP 2022536174 A5 JP2022536174 A5 JP 2022536174A5 JP 2021573717 A JP2021573717 A JP 2021573717A JP 2021573717 A JP2021573717 A JP 2021573717A JP 2022536174 A5 JP2022536174 A5 JP 2022536174A5
Authority
JP
Japan
Prior art keywords
pyrazolo
pyridine
fluorophenyl
cyclopropyl
difluoromethyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2021573717A
Other languages
English (en)
Japanese (ja)
Other versions
JP2022536174A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/EP2020/066391 external-priority patent/WO2020249791A1/en
Publication of JP2022536174A publication Critical patent/JP2022536174A/ja
Publication of JP2022536174A5 publication Critical patent/JP2022536174A5/ja
Pending legal-status Critical Current

Links

JP2021573717A 2019-06-14 2020-06-12 置換ピラゾロ[4,3-b]ピリジニル及びGLUN2B受容体調節因子としてのそれらの使用 Pending JP2022536174A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201962861674P 2019-06-14 2019-06-14
US62/861,674 2019-06-14
PCT/EP2020/066391 WO2020249791A1 (en) 2019-06-14 2020-06-12 SUBSTITUTED PYRAZOLO[4,3-b]PYRIDINES AND THEIR USE AS GLUN2B RECEPTOR MODULATORS

Publications (2)

Publication Number Publication Date
JP2022536174A JP2022536174A (ja) 2022-08-12
JP2022536174A5 true JP2022536174A5 (enExample) 2023-06-20

Family

ID=71120146

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2021573717A Pending JP2022536174A (ja) 2019-06-14 2020-06-12 置換ピラゾロ[4,3-b]ピリジニル及びGLUN2B受容体調節因子としてのそれらの使用

Country Status (10)

Country Link
US (2) US20220324860A1 (enExample)
EP (1) EP3983073A1 (enExample)
JP (1) JP2022536174A (enExample)
KR (1) KR20220020917A (enExample)
CN (1) CN113993583A (enExample)
AU (1) AU2020293642A1 (enExample)
BR (1) BR112021025136A2 (enExample)
CA (1) CA3143102A1 (enExample)
MX (1) MX2021015510A (enExample)
WO (1) WO2020249791A1 (enExample)

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AU2020291188A1 (en) 2019-06-14 2022-01-20 Janssen Pharmaceutica Nv Substituted heteroaromatic Pyrazolo-pyridines and their use as GluN2B receptor modulators
SG11202112407PA (en) 2019-06-14 2021-12-30 Janssen Pharmaceutica Nv Substituted pyrazolo-pyridine amides and their use as glun2b receptor modulators
JP7667097B2 (ja) 2019-06-14 2025-04-22 ヤンセン ファーマシューティカ エヌ.ベー. 置換ピラゾロ-ピリジンアミド及びglun2b受容体調節因子としてのその使用
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US20220324860A1 (en) 2019-06-14 2022-10-13 Janssen Pharmaceutica Nv SUBSTITUTED PYRAZOLO[4,3-b]PYRIDINES AND THEIR USE AS GLUN2B RECEPTOR MODULATORS
BR112021025132A2 (pt) 2019-06-14 2022-01-25 Janssen Pharmaceutica Nv Carbamatos de piridina e seu uso como moduladores do receptor glun2b
EP4669318A1 (en) * 2023-02-23 2025-12-31 The Rockefeller University 1-ACYL-3-AMINOINDAZOLES FOR THE TREATMENT OF CYSTIC FIBROSIS

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TW201819376A (zh) * 2016-10-06 2018-06-01 比利時商健生藥品公司 經取代之1H-咪唑並[4,5-b]吡啶-2(3H)-酮及其作為GLUN2B受體調節劑之用途
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EP3774732A4 (en) 2018-04-04 2022-02-09 Janssen Pharmaceutica NV PYRIDINE AND SUBSTITUTED PYRIMIDINES AND THEIR USE AS GLUN2B RECEPTOR MODULATORS
CN110294756A (zh) 2019-06-04 2019-10-01 广州市原子高科同位素医药有限公司 GluN2B亚基靶向型中枢神经系统正电子示踪剂及其制备
AU2020291188A1 (en) 2019-06-14 2022-01-20 Janssen Pharmaceutica Nv Substituted heteroaromatic Pyrazolo-pyridines and their use as GluN2B receptor modulators
US20220324860A1 (en) 2019-06-14 2022-10-13 Janssen Pharmaceutica Nv SUBSTITUTED PYRAZOLO[4,3-b]PYRIDINES AND THEIR USE AS GLUN2B RECEPTOR MODULATORS
EP3983413A1 (en) 2019-06-14 2022-04-20 Janssen Pharmaceutica NV Substituted pyrazolo-pyrazines and their use as glun2b receptor modulators
BR112021025132A2 (pt) 2019-06-14 2022-01-25 Janssen Pharmaceutica Nv Carbamatos de piridina e seu uso como moduladores do receptor glun2b
SG11202112407PA (en) 2019-06-14 2021-12-30 Janssen Pharmaceutica Nv Substituted pyrazolo-pyridine amides and their use as glun2b receptor modulators
AU2020290772A1 (en) 2019-06-14 2022-01-06 Janssen Pharmaceutica Nv Pyrazine carbamates and their use as GluN2B receptor modulators

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