JP2022527630A5 - - Google Patents

Info

Publication number
JP2022527630A5
JP2022527630A5 JP2021560228A JP2021560228A JP2022527630A5 JP 2022527630 A5 JP2022527630 A5 JP 2022527630A5 JP 2021560228 A JP2021560228 A JP 2021560228A JP 2021560228 A JP2021560228 A JP 2021560228A JP 2022527630 A5 JP2022527630 A5 JP 2022527630A5
Authority
JP
Japan
Prior art keywords
approximately
pharmaceutical composition
composition according
sucralose
citric acid
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2021560228A
Other languages
English (en)
Japanese (ja)
Other versions
JP2022527630A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2020/026696 external-priority patent/WO2020206336A1/en
Publication of JP2022527630A publication Critical patent/JP2022527630A/ja
Publication of JP2022527630A5 publication Critical patent/JP2022527630A5/ja
Pending legal-status Critical Current

Links

JP2021560228A 2019-04-05 2020-04-03 鎌状赤血球症を治療するためのpde9阻害剤 Pending JP2022527630A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201962829784P 2019-04-05 2019-04-05
US62/829,784 2019-04-05
PCT/US2020/026696 WO2020206336A1 (en) 2019-04-05 2020-04-03 Pde9 inhibitors for treating sickle cell disease

Publications (2)

Publication Number Publication Date
JP2022527630A JP2022527630A (ja) 2022-06-02
JP2022527630A5 true JP2022527630A5 (https=) 2023-04-10

Family

ID=72666968

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2021560228A Pending JP2022527630A (ja) 2019-04-05 2020-04-03 鎌状赤血球症を治療するためのpde9阻害剤

Country Status (9)

Country Link
US (1) US20220023302A1 (https=)
EP (1) EP3946348A4 (https=)
JP (1) JP2022527630A (https=)
CN (1) CN114302724A (https=)
BR (1) BR112021019876A2 (https=)
CA (1) CA3136128A1 (https=)
IL (1) IL286976A (https=)
WO (1) WO2020206336A1 (https=)
ZA (1) ZA202107544B (https=)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PT3865484T (pt) 2015-07-07 2024-01-30 H Lundbeck As Inibidor da pde9 com esqueleto de imidazo pirazinona para tratamento de doenças periféricas
CA3100988A1 (en) 2018-05-25 2019-11-28 Imara Inc. Monohydrate and crystalline forms of 6-[(3s,4s)-4-methyl-1-(pyrimidin-2-ylmethyl)pyrrolidin-3-yl]-3-tetrahydropyran-4-yl-7h-imidazo[1,5-a]pyrazin-8-one
CA3110680A1 (en) 2018-08-31 2020-03-05 Imara Inc. Pde9 inhibitors for treating sickle cell disease

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2009507032A (ja) * 2005-09-02 2009-02-19 アボット・ラボラトリーズ 新規なイミダゾ系複素環
JP4941977B2 (ja) * 2007-04-11 2012-05-30 大蔵製薬株式会社 ベンズイソキサゾール誘導体の経口ゼリー状医薬組成物
BR112015007731B1 (pt) * 2011-10-10 2022-05-31 H. Lundbeck A/S Composto, composição farmacêutica que o compreende e uso do mesmo
EP2868319A4 (en) * 2012-06-29 2016-02-24 Maruishi Pharma ORAL PHARMACEUTICAL ARIPIPRAZONE PREPARATION
PT3865484T (pt) * 2015-07-07 2024-01-30 H Lundbeck As Inibidor da pde9 com esqueleto de imidazo pirazinona para tratamento de doenças periféricas
US10045991B2 (en) * 2016-04-04 2018-08-14 Loxo Oncology, Inc. Methods of treating pediatric cancers
MX2018016127A (es) * 2016-07-06 2019-05-30 Imara Inc Inhibidores de pde9 para el tratamiento de enfermedades perifericas.
CN115746003B (zh) * 2017-05-26 2024-08-09 卡都瑞恩医药公司 制备和使用pde9抑制剂的方法
EP3965768A1 (en) * 2019-05-07 2022-03-16 Imara Inc. Pde9 inhibitors for treating thalassemia

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