JP2022526675A5 - - Google Patents
Info
- Publication number
- JP2022526675A5 JP2022526675A5 JP2021560231A JP2021560231A JP2022526675A5 JP 2022526675 A5 JP2022526675 A5 JP 2022526675A5 JP 2021560231 A JP2021560231 A JP 2021560231A JP 2021560231 A JP2021560231 A JP 2021560231A JP 2022526675 A5 JP2022526675 A5 JP 2022526675A5
- Authority
- JP
- Japan
- Prior art keywords
- sub
- formula
- dichlorophenyl
- glucitol
- deoxy
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP19382273.1 | 2019-04-11 | ||
| EP19382273 | 2019-04-11 | ||
| PCT/EP2020/057683 WO2020207753A1 (en) | 2019-04-11 | 2020-03-19 | Process for preparing 1-deoxy-1-methylamino-d-glucitol 2-(3,5-dichlorophenyl)-6-benzoxazolecarboxylate |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2022526675A JP2022526675A (ja) | 2022-05-25 |
| JP2022526675A5 true JP2022526675A5 (enExample) | 2023-03-27 |
| JP7622338B2 JP7622338B2 (ja) | 2025-01-28 |
Family
ID=66240025
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2021560231A Active JP7622338B2 (ja) | 2019-04-11 | 2020-03-19 | 2-(3,5-ジクロロフェニル)-6-ベンズオキサゾールカルボン酸1-デオキシ-1-メチルアミノ-d-グルシトールの製造方法 |
Country Status (10)
| Country | Link |
|---|---|
| US (1) | US12116352B2 (enExample) |
| EP (1) | EP3953339B1 (enExample) |
| JP (1) | JP7622338B2 (enExample) |
| CN (1) | CN113874359B (enExample) |
| AR (1) | AR118647A1 (enExample) |
| ES (1) | ES2991081T3 (enExample) |
| HR (1) | HRP20241374T1 (enExample) |
| HU (1) | HUE068975T2 (enExample) |
| PL (1) | PL3953339T3 (enExample) |
| WO (1) | WO2020207753A1 (enExample) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN113372290A (zh) * | 2021-05-21 | 2021-09-10 | 遵义医科大学 | 一种药物Tafamidis的合成方法 |
| CN113277993B (zh) * | 2021-06-06 | 2023-07-21 | 湖南第一师范学院 | 一种Tafamidis及其衍生物的合成方法 |
| CN113735792B (zh) * | 2021-09-22 | 2024-10-18 | 上海新礼泰药业有限公司 | 氯苯唑酸葡胺及其中间体的制备方法 |
| KR102657823B1 (ko) * | 2022-03-10 | 2024-04-16 | 고려대학교 산학협력단 | 타파미디스의 신규 합성법 |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2800237C (en) * | 2002-12-19 | 2016-05-17 | The Scripps Research Institute | Compositions and methods for stabilizing transthyretin and inhibiting transthyretin misfolding |
| JP2006513250A (ja) | 2003-01-28 | 2006-04-20 | 中国科学院上海薬物研究所 | アラニン系化合物、その製造方法及び用途 |
| RU2586330C2 (ru) | 2011-09-16 | 2016-06-10 | Пфайзер Инк. | Твердые формы ингибитора диссоциации транстиретина |
| US9499527B2 (en) * | 2012-05-10 | 2016-11-22 | Cellix Bio Private Limited | Compositions and methods for the treatment of familial amyloid polyneuropathy |
| PT4349406T (pt) * | 2014-09-08 | 2026-02-04 | Pfizer | Formas sólidas cristalinas de 6-carboxi-2-(3,5-diclorofenil)-benzoxazol para utilização como medicamento |
| CN107344927A (zh) | 2016-05-05 | 2017-11-14 | 苏州晶云药物科技有限公司 | Tafamidis葡甲胺盐的晶型E及其制备方法和用途 |
-
2020
- 2020-03-19 US US17/601,946 patent/US12116352B2/en active Active
- 2020-03-19 ES ES20710987T patent/ES2991081T3/es active Active
- 2020-03-19 HU HUE20710987A patent/HUE068975T2/hu unknown
- 2020-03-19 JP JP2021560231A patent/JP7622338B2/ja active Active
- 2020-03-19 WO PCT/EP2020/057683 patent/WO2020207753A1/en not_active Ceased
- 2020-03-19 HR HRP20241374TT patent/HRP20241374T1/hr unknown
- 2020-03-19 CN CN202080035225.4A patent/CN113874359B/zh active Active
- 2020-03-19 PL PL20710987.7T patent/PL3953339T3/pl unknown
- 2020-03-19 EP EP20710987.7A patent/EP3953339B1/en active Active
- 2020-04-09 AR ARP200101020A patent/AR118647A1/es unknown
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