JP2022513215A5 - - Google Patents
Info
- Publication number
- JP2022513215A5 JP2022513215A5 JP2021533641A JP2021533641A JP2022513215A5 JP 2022513215 A5 JP2022513215 A5 JP 2022513215A5 JP 2021533641 A JP2021533641 A JP 2021533641A JP 2021533641 A JP2021533641 A JP 2021533641A JP 2022513215 A5 JP2022513215 A5 JP 2022513215A5
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- independently
- group
- pharmaceutically acceptable
- compound according
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201862779960P | 2018-12-14 | 2018-12-14 | |
| US62/779,960 | 2018-12-14 | ||
| PCT/US2019/066414 WO2020124060A1 (en) | 2018-12-14 | 2019-12-14 | Organophosphorus-substituted compounds as c-met inhibitors and therapeutic uses thereof |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2022513215A JP2022513215A (ja) | 2022-02-07 |
| JP2022513215A5 true JP2022513215A5 (https=) | 2022-11-24 |
Family
ID=71077551
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2021533641A Pending JP2022513215A (ja) | 2018-12-14 | 2019-12-14 | C-met阻害剤としての有機リン置換化合物およびその治療用途 |
Country Status (15)
| Country | Link |
|---|---|
| US (1) | US12258365B2 (https=) |
| EP (1) | EP3893872B1 (https=) |
| JP (1) | JP2022513215A (https=) |
| KR (1) | KR20210111779A (https=) |
| CN (1) | CN113412112B (https=) |
| AU (1) | AU2019395282A1 (https=) |
| BR (1) | BR112021011547A2 (https=) |
| CA (1) | CA3122575A1 (https=) |
| EA (1) | EA202191541A1 (https=) |
| IL (1) | IL283589A (https=) |
| MX (1) | MX2021006982A (https=) |
| SG (1) | SG11202105872RA (https=) |
| TW (1) | TW202039500A (https=) |
| WO (1) | WO2020124060A1 (https=) |
| ZA (1) | ZA202104000B (https=) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN116969955B (zh) * | 2023-09-25 | 2023-12-19 | 中国药科大学 | 一种[1,2,4]三唑[4,3-b]哒嗪类化合物及其制法与应用 |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| HRP20170103T1 (hr) | 2005-12-21 | 2017-03-24 | Janssen Pharmaceutica N.V. | Triazolopiridazini kao modulatori tirozin kinaze |
| NL2000613C2 (nl) * | 2006-05-11 | 2007-11-20 | Pfizer Prod Inc | Triazoolpyrazinederivaten. |
| US20110039856A1 (en) * | 2007-11-29 | 2011-02-17 | Pfizer Inc. | Polymorphs of a c-met/hgfr inhibitor |
| UY32049A (es) | 2008-08-14 | 2010-03-26 | Takeda Pharmaceutical | Inhibidores de cmet |
| EA030141B1 (ru) | 2009-12-31 | 2018-06-29 | Хатчисон Медифарма Лимитед | Определенные триазолопиридины и триазолопиразины, их композиции и способы их применения |
| ES2598530T3 (es) | 2010-07-14 | 2017-01-27 | Betta Pharmaceuticals Co., Ltd. | Nuevos derivados heterocíclicos condensados útiles como inhibidores de la tirosina quinasa c-Met |
| TWI520962B (zh) * | 2012-06-29 | 2016-02-11 | As the c-Met tyrosine kinase inhibitors novel fused pyridine derivatives | |
| CN103122000B (zh) * | 2012-09-03 | 2013-12-25 | 中美冠科生物技术(太仓)有限公司 | 用作抗肿瘤药物的高选择性的c-Met激酶抑制剂 |
| ES2877799T3 (es) * | 2015-12-31 | 2021-11-17 | Shanghai Pharmaceuticals Holding Co Ltd | Sal de derivado de quinolina, formas polimórficas de la misma, métodos de preparación de la misma, composición y aplicaciones |
-
2019
- 2019-12-14 EA EA202191541A patent/EA202191541A1/ru unknown
- 2019-12-14 BR BR112021011547-1A patent/BR112021011547A2/pt not_active IP Right Cessation
- 2019-12-14 AU AU2019395282A patent/AU2019395282A1/en not_active Abandoned
- 2019-12-14 JP JP2021533641A patent/JP2022513215A/ja active Pending
- 2019-12-14 SG SG11202105872RA patent/SG11202105872RA/en unknown
- 2019-12-14 CA CA3122575A patent/CA3122575A1/en not_active Abandoned
- 2019-12-14 US US17/312,669 patent/US12258365B2/en active Active
- 2019-12-14 MX MX2021006982A patent/MX2021006982A/es unknown
- 2019-12-14 EP EP19897455.2A patent/EP3893872B1/en active Active
- 2019-12-14 CN CN201980091722.3A patent/CN113412112B/zh active Active
- 2019-12-14 WO PCT/US2019/066414 patent/WO2020124060A1/en not_active Ceased
- 2019-12-14 KR KR1020217022048A patent/KR20210111779A/ko not_active Withdrawn
- 2019-12-16 TW TW108146055A patent/TW202039500A/zh unknown
-
2021
- 2021-05-31 IL IL283589A patent/IL283589A/en unknown
- 2021-06-10 ZA ZA2021/04000A patent/ZA202104000B/en unknown
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