JP2022508523A5 - - Google Patents
Info
- Publication number
- JP2022508523A5 JP2022508523A5 JP2021542086A JP2021542086A JP2022508523A5 JP 2022508523 A5 JP2022508523 A5 JP 2022508523A5 JP 2021542086 A JP2021542086 A JP 2021542086A JP 2021542086 A JP2021542086 A JP 2021542086A JP 2022508523 A5 JP2022508523 A5 JP 2022508523A5
- Authority
- JP
- Japan
- Prior art keywords
- pyridine
- thieno
- trifluoromethyl
- methylcarbamoyl
- piperidine
- Prior art date
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201862739405P | 2018-10-01 | 2018-10-01 | |
| US62/739,405 | 2018-10-01 | ||
| PCT/US2019/054085 WO2020072504A1 (en) | 2018-10-01 | 2019-10-01 | Thieno[3,2-b]pyridine derivatives as udp glycosyltransferase inhibitors and methods of use |
Publications (4)
| Publication Number | Publication Date |
|---|---|
| JP2022508523A JP2022508523A (ja) | 2022-01-19 |
| JP2022508523A5 true JP2022508523A5 (https=) | 2022-09-07 |
| JPWO2020072504A5 JPWO2020072504A5 (https=) | 2022-09-07 |
| JP7545979B2 JP7545979B2 (ja) | 2024-09-05 |
Family
ID=68296740
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2021542086A Active JP7545979B2 (ja) | 2018-10-01 | 2019-10-01 | ＵＤＰグリコシルトランスフェラーゼ阻害剤としてのチエノ［３，２－ｂ］ピリジン誘導体および使用の方法 |
Country Status (15)
| Country | Link |
|---|---|
| US (1) | US11098056B2 (https=) |
| EP (1) | EP3861000A1 (https=) |
| JP (1) | JP7545979B2 (https=) |
| KR (1) | KR102903997B1 (https=) |
| CN (1) | CN113423711B (https=) |
| AU (1) | AU2019355870B2 (https=) |
| BR (1) | BR112021005914A2 (https=) |
| CA (1) | CA3114722A1 (https=) |
| CO (1) | CO2021005738A2 (https=) |
| IL (1) | IL281811B2 (https=) |
| MA (1) | MA53043B2 (https=) |
| MX (1) | MX2021003794A (https=) |
| SG (1) | SG11202102987VA (https=) |
| TW (1) | TWI821426B (https=) |
| WO (1) | WO2020072504A1 (https=) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TW202302565A (zh) * | 2021-02-19 | 2023-01-16 | 英商卡爾維斯塔製藥有限公司 | 酶抑制劑 |
| EP4483954A1 (en) * | 2023-06-29 | 2025-01-01 | Masarykova Univerzita | Substituted thieno [3,2-b]pyridines as inhibitors of protein kinases |
Family Cites Families (15)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3763156A (en) * | 1970-01-28 | 1973-10-02 | Boehringer Sohn Ingelheim | 2-heterocyclic amino-4-morpholinothieno(3,2-d)pyrimidines |
| US7375125B2 (en) * | 1999-08-04 | 2008-05-20 | Ore Pharmaceuticals, Inc. | Melanocortin-4 receptor binding compounds and methods of use thereof |
| MXPA02001160A (es) | 1999-08-04 | 2002-07-02 | Millennium Pharm Inc | Compuestos que se unen a los receptores para melanocortina-4, y metodo de uso de estos. |
| FR2821356A1 (fr) * | 2001-02-23 | 2002-08-30 | Cerep | Nouveaux derives d'arylcarbamates et d'arylurees, preparations et utilisations |
| EP3109249A1 (en) * | 2007-11-15 | 2016-12-28 | YM BioSciences Australia Pty Ltd | N-containing heterocyclic compounds |
| MX2011008276A (es) * | 2009-02-06 | 2011-12-14 | Elan Pharm Inc | Inhibidores de quinasa jun n-terminal. |
| JP2014511391A (ja) * | 2011-03-07 | 2014-05-15 | フォンダッツィオーネ・テレソン | Ｔｆｅｂリン酸化阻害剤およびその使用 |
| ES2928714T3 (es) * | 2015-01-16 | 2022-11-22 | Massachusetts Gen Hospital | Compuestos para mejorar el empalme del ARNm |
| JP7114076B2 (ja) | 2015-12-22 | 2022-08-08 | シャイ・セラピューティクス・エルエルシー | がん及び炎症性疾患の処置のための化合物 |
| SG11201809693SA (en) * | 2016-05-05 | 2018-11-29 | Lysosomal Therapeutics Inc | SUBSTITUTED IMIDAZO[1,2-b]PYRIDAZINES, SUBSTITUTED IMIDAZO[1,5-b]PYRIDAZINES, RELATED COMPOUNDS, AND THEIR USE IN THE TREATMENT OF MEDICAL DISORDERS |
| WO2017214505A1 (en) * | 2016-06-10 | 2017-12-14 | Biomarin Pharmaceutical Inc. | Ceramide galactosyltransferase inhibitors for the treatment of disease |
| MY193511A (en) * | 2016-11-02 | 2022-10-17 | Janssen Pharmaceutica Nv | [1,2,4]triazolo[1,5-a]pyrimidine derivatives as pde2 inhibitors |
| WO2018118838A1 (en) * | 2016-12-20 | 2018-06-28 | Biomarin Pharmaceutical Inc. | Ceramide galactosyltransferase inhibitors for the treatment of disease |
| EP3619209A1 (en) * | 2017-05-04 | 2020-03-11 | Glenmark Pharmaceuticals S.A. | Substituted bicyclic heterocyclic compounds as nadph oxidase inhibitors |
| JP7514005B2 (ja) | 2017-06-21 | 2024-07-10 | シャイ・セラピューティクス・エルエルシー | がん、炎症性疾患、ラソパシー、及び線維性疾患の治療のためのｒａｓスーパーファミリーと相互作用する化合物 |
-
2019
- 2019-10-01 SG SG11202102987VA patent/SG11202102987VA/en unknown
- 2019-10-01 EP EP19791011.0A patent/EP3861000A1/en active Pending
- 2019-10-01 CA CA3114722A patent/CA3114722A1/en active Pending
- 2019-10-01 CN CN201980076707.1A patent/CN113423711B/zh active Active
- 2019-10-01 AU AU2019355870A patent/AU2019355870B2/en active Active
- 2019-10-01 IL IL281811A patent/IL281811B2/en unknown
- 2019-10-01 KR KR1020217013167A patent/KR102903997B1/ko active Active
- 2019-10-01 WO PCT/US2019/054085 patent/WO2020072504A1/en not_active Ceased
- 2019-10-01 US US16/590,027 patent/US11098056B2/en active Active
- 2019-10-01 BR BR112021005914-8A patent/BR112021005914A2/pt unknown
- 2019-10-01 MA MA53043A patent/MA53043B2/fr unknown
- 2019-10-01 JP JP2021542086A patent/JP7545979B2/ja active Active
- 2019-10-01 MX MX2021003794A patent/MX2021003794A/es unknown
- 2019-10-01 TW TW108135781A patent/TWI821426B/zh active
-
2021
- 2021-04-29 CO CONC2021/0005738A patent/CO2021005738A2/es unknown
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| US11739098B2 (en) | Substituted indole compounds | |
| KR101812357B1 (ko) | Ｃｄｋ4/6의 억제제로서의 피롤로피리미딘 화합물 | |
| HRP20210177T1 (hr) | Supstituirani spojevi pirazolo[1,5-a]piridina kao inhibitori ret kinaze | |
| JPWO2020005877A5 (https=) | ||
| HRP20210935T1 (hr) | Spojevi 5-kloro-2-difluorometoksifenil pirazolopirimidina koji predstavljaju inhibitore jak | |
| JP2014506929A5 (https=) | ||
| JP2021519291A5 (https=) | ||
| JP2018530557A5 (https=) | ||
| JP2018530557A (ja) | 置換ピラゾロ［３，４−ｂ］ピリジン−６−カルボン酸およびこの使用 | |
| JPWO2019191229A5 (https=) | ||
| RU2016135637A (ru) | 6-гетероарилокси- и 6-арилоксихинолин-2-карбоксамиды и их применение | |
| JP2015522002A5 (https=) | ||
| JP2015523387A5 (https=) | ||
| HRP20250272T1 (hr) | Derivati benzimidazola i njihova uporaba | |
| JP2017505327A5 (https=) | ||
| JP2015537010A5 (https=) | ||
| JP2018529743A (ja) | Ｎ−スルホニル化ピラゾロ［３，４−ｂ］ピリジン−６−カルボキサミドおよび使用法 | |
| JPWO2020005873A5 (https=) | ||
| JP2015504057A5 (https=) | ||
| RU2020129785A (ru) | Фармацевтические производные 6,5-гетеробициклического кольца | |
| US11840528B2 (en) | Isoxazolyl ether derivatives as GABAA α5 PAM | |
| JPWO2022147246A5 (https=) | ||
| JPWO2020231977A5 (https=) | ||
| JP2022508523A5 (https=) | ||
| RU2020127848A (ru) | Производные 4-гидроксипиперидина и их применение в качестве ингибиторов убиквитин-специфической протеазы 19 (usp19) |