JP2022504181A5 - - Google Patents

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Publication number
JP2022504181A5
JP2022504181A5 JP2021518472A JP2021518472A JP2022504181A5 JP 2022504181 A5 JP2022504181 A5 JP 2022504181A5 JP 2021518472 A JP2021518472 A JP 2021518472A JP 2021518472 A JP2021518472 A JP 2021518472A JP 2022504181 A5 JP2022504181 A5 JP 2022504181A5
Authority
JP
Japan
Prior art keywords
scleroderma
systemic sclerosis
compound
composition
solvate
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2021518472A
Other languages
English (en)
Japanese (ja)
Other versions
JP2022504181A (ja
JP7265620B2 (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2019/054576 external-priority patent/WO2020072824A1/en
Publication of JP2022504181A publication Critical patent/JP2022504181A/ja
Publication of JP2022504181A5 publication Critical patent/JP2022504181A5/ja
Priority to JP2023055658A priority Critical patent/JP2023082117A/ja
Application granted granted Critical
Publication of JP7265620B2 publication Critical patent/JP7265620B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2021518472A 2018-10-03 2019-10-03 強皮症の治療のための方法 Active JP7265620B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2023055658A JP2023082117A (ja) 2018-10-03 2023-03-30 強皮症の治療のための方法

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201862740855P 2018-10-03 2018-10-03
US62/740,855 2018-10-03
PCT/US2019/054576 WO2020072824A1 (en) 2018-10-03 2019-10-03 Methods for the treatment of scleroderma

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2023055658A Division JP2023082117A (ja) 2018-10-03 2023-03-30 強皮症の治療のための方法

Publications (3)

Publication Number Publication Date
JP2022504181A JP2022504181A (ja) 2022-01-13
JP2022504181A5 true JP2022504181A5 (https=) 2022-09-29
JP7265620B2 JP7265620B2 (ja) 2023-04-26

Family

ID=68290393

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2021518472A Active JP7265620B2 (ja) 2018-10-03 2019-10-03 強皮症の治療のための方法
JP2023055658A Pending JP2023082117A (ja) 2018-10-03 2023-03-30 強皮症の治療のための方法

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2023055658A Pending JP2023082117A (ja) 2018-10-03 2023-03-30 強皮症の治療のための方法

Country Status (5)

Country Link
US (1) US20210386706A1 (https=)
EP (1) EP3860590B1 (https=)
JP (2) JP7265620B2 (https=)
ES (1) ES2951870T3 (https=)
WO (1) WO2020072824A1 (https=)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP5856980B2 (ja) 2010-01-27 2016-02-10 アリーナ ファーマシューティカルズ, インコーポレイテッド (R)−2−(7−(4−シクロペンチル−3−(トリフルオロメチル)ベンジルオキシ)−1,2,3,4−テトラヒドロシクロペンタ[b]インドール−3−イル)酢酸およびその塩の調製のためのプロセス
PL3242666T3 (pl) 2015-01-06 2025-02-17 Arena Pharmaceuticals, Inc. Związek do zastosowania w leczeniu dolegliwości związanych z receptorem s1p1
BR112017027656B1 (pt) 2015-06-22 2023-12-05 Arena Pharmaceuticals, Inc. Hábito cristalino de placa livre de sal de l-arginina de ácido (r)-2-(7-(4- ciclopentil-3-(trifluorometil)benzilóxi)- 1,2,3,4-tetra-hidrociclo-penta[b]indol-3- il)acético, composição farmacêutica que o compreende, seus usos e método de preparação do mesmo
MX2019009841A (es) 2017-02-16 2020-01-30 Arena Pharm Inc Compuestos y metodos para el tratamiento de la colangitis biliar primaria.
MX2019009843A (es) 2017-02-16 2020-01-30 Arena Pharm Inc Compuestos y metodos para el tratamiento de la enfermedad inflamatoria intestinal con manifestaciones extraintestinales.
CA3102136A1 (en) 2018-06-06 2019-12-12 Arena Pharmaceuticals, Inc. Methods of treating conditions related to the s1p1 receptor

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2001003739A1 (fr) * 1999-07-12 2001-01-18 Ono Pharmaceutical Co., Ltd. Inhibiteurs de fibrose contenant comme ingredient actif l'agoniste du recepteur de sphingosine-1-phosphate ou la sphingosine-1-phosphate
US8580841B2 (en) * 2008-07-23 2013-11-12 Arena Pharmaceuticals, Inc. Substituted 1,2,3,4-tetrahydrocyclopenta[b]indol-3-yl)acetic acid derivatives useful in the treatment of autoimmune and inflammatory disorders
JP5856980B2 (ja) 2010-01-27 2016-02-10 アリーナ ファーマシューティカルズ, インコーポレイテッド (R)−2−(7−(4−シクロペンチル−3−(トリフルオロメチル)ベンジルオキシ)−1,2,3,4−テトラヒドロシクロペンタ[b]インドール−3−イル)酢酸およびその塩の調製のためのプロセス
PL3242666T3 (pl) 2015-01-06 2025-02-17 Arena Pharmaceuticals, Inc. Związek do zastosowania w leczeniu dolegliwości związanych z receptorem s1p1
BR112017027656B1 (pt) * 2015-06-22 2023-12-05 Arena Pharmaceuticals, Inc. Hábito cristalino de placa livre de sal de l-arginina de ácido (r)-2-(7-(4- ciclopentil-3-(trifluorometil)benzilóxi)- 1,2,3,4-tetra-hidrociclo-penta[b]indol-3- il)acético, composição farmacêutica que o compreende, seus usos e método de preparação do mesmo
MX2019009841A (es) * 2017-02-16 2020-01-30 Arena Pharm Inc Compuestos y metodos para el tratamiento de la colangitis biliar primaria.
MX2019009843A (es) * 2017-02-16 2020-01-30 Arena Pharm Inc Compuestos y metodos para el tratamiento de la enfermedad inflamatoria intestinal con manifestaciones extraintestinales.
CA3102136A1 (en) * 2018-06-06 2019-12-12 Arena Pharmaceuticals, Inc. Methods of treating conditions related to the s1p1 receptor
CN113874009A (zh) * 2019-01-08 2021-12-31 艾尼纳制药公司 治疗与s1p1受体有关的病况的方法

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