JP2022502415A - ヒドラジン化合物の調製のための合成方法 - Google Patents

ヒドラジン化合物の調製のための合成方法 Download PDF

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Publication number
JP2022502415A
JP2022502415A JP2021516992A JP2021516992A JP2022502415A JP 2022502415 A JP2022502415 A JP 2022502415A JP 2021516992 A JP2021516992 A JP 2021516992A JP 2021516992 A JP2021516992 A JP 2021516992A JP 2022502415 A JP2022502415 A JP 2022502415A
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Japan
Prior art keywords
compound
nitrite
sulfite
reaction mass
reaction
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Pending
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JP2021516992A
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Japanese (ja)
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JP2022502415A5 (https=
Inventor
リ，ユンジョン
ジアン，シャオビン
ヨハネス ロンド，ニエック
ルイズ，カルメン
ドーヴェルヌ，ジェローム
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メレオ バイオファーマ １ リミテッド
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Publication of JP2022502415A publication Critical patent/JP2022502415A/ja
Publication of JP2022502415A5 publication Critical patent/JP2022502415A5/ja
Pending legal-status Critical Current

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C241/00—Preparation of compounds containing chains of nitrogen atoms singly-bound to each other, e.g. hydrazines, triazanes
    • C07C241/02—Preparation of hydrazines
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C243/00—Compounds containing chains of nitrogen atoms singly-bound to each other, e.g. hydrazines, triazanes
    • C07C243/10—Hydrazines
    • C07C243/22—Hydrazines having nitrogen atoms of hydrazine groups bound to carbon atoms of six-membered aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C255/00—Carboxylic acid nitriles
    • C07C255/49—Carboxylic acid nitriles having cyano groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton
    • C07C255/56—Carboxylic acid nitriles having cyano groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton containing cyano groups and doubly-bound oxygen atoms bound to the carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/38—Nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00—Systems containing only non-condensed rings
    • C07C2601/12—Systems containing only non-condensed rings with a six-membered ring
    • C07C2601/16—Systems containing only non-condensed rings with a six-membered ring the ring being unsaturated

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
JP2021516992A 2018-09-26 2019-09-26 ヒドラジン化合物の調製のための合成方法 Pending JP2022502415A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GBGB1815696.8A GB201815696D0 (en) 2018-09-26 2018-09-26 Synthetic method
GB1815696.8 2018-09-26
PCT/GB2019/052719 WO2020065324A1 (en) 2018-09-26 2019-09-26 Synthetic method for the preparation of an hydrazine compound

Publications (2)

Publication Number Publication Date
JP2022502415A true JP2022502415A (ja) 2022-01-11
JP2022502415A5 JP2022502415A5 (https=) 2022-09-02

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ID=64024292

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JP2021516992A Pending JP2022502415A (ja) 2018-09-26 2019-09-26 ヒドラジン化合物の調製のための合成方法

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US (1) US20210340108A1 (https=)
EP (1) EP3856711B1 (https=)
JP (1) JP2022502415A (https=)
KR (1) KR20210065111A (https=)
CN (1) CN112839923A (https=)
AU (1) AU2019349863A1 (https=)
CA (1) CA3112998A1 (https=)
DK (1) DK3856711T3 (https=)
ES (1) ES2933568T3 (https=)
GB (1) GB201815696D0 (https=)
IL (1) IL281637A (https=)
WO (1) WO2020065324A1 (https=)

Citations (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2007521278A (ja) * 2003-06-26 2007-08-02 ノバルティス アクチエンゲゼルシャフト ５員ヘテロ環を基礎とするｐ３８キナーゼ阻害剤
WO2009088025A1 (ja) * 2008-01-10 2009-07-16 Hokko Chemical Industry Co., Ltd. フェニルトリアゾリノン類の製造法
JP2009293016A (ja) * 2008-05-02 2009-12-17 Canon Inc インクジェット用インク、インクジェット記録方法、インクカートリッジ、記録ユニット、及びインクジェット記録装置
JP2010535187A (ja) * 2007-08-02 2010-11-18 ジェネリクス・（ユーケー）・リミテッド 新規な方法
JP2016204436A (ja) * 2015-04-17 2016-12-08 日本化薬株式会社 水溶性アゾ化合物又はその塩、インク組成物及び着色体

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2732967B1 (fr) * 1995-04-11 1997-07-04 Sanofi Sa 1-phenylpyrazole-3-carboxamides substitues, actifs sur la neurotensine, leur preparation, les compositions pharmaceutiques en contenant
CN1326029C (zh) * 2003-07-10 2007-07-11 富士施乐株式会社 印刷装置、印刷指示装置、印刷处理系统及印刷处理方法
US7485657B2 (en) * 2004-05-12 2009-02-03 Boehringer Ingelheim Pharmaceuticals, Inc. Anti-cytokine heterocyclic compounds
CN102964270B (zh) * 2012-11-21 2015-01-07 合肥星宇化学有限责任公司 一种亚硫酸钠还原重氮盐合成肼的方法
WO2018059533A1 (zh) * 2016-09-29 2018-04-05 南京明德新药研发股份有限公司 p38αMAPK激酶抑制剂及其制备方法和应用

Patent Citations (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2007521278A (ja) * 2003-06-26 2007-08-02 ノバルティス アクチエンゲゼルシャフト ５員ヘテロ環を基礎とするｐ３８キナーゼ阻害剤
JP2010535187A (ja) * 2007-08-02 2010-11-18 ジェネリクス・（ユーケー）・リミテッド 新規な方法
WO2009088025A1 (ja) * 2008-01-10 2009-07-16 Hokko Chemical Industry Co., Ltd. フェニルトリアゾリノン類の製造法
JP2009293016A (ja) * 2008-05-02 2009-12-17 Canon Inc インクジェット用インク、インクジェット記録方法、インクカートリッジ、記録ユニット、及びインクジェット記録装置
JP2016204436A (ja) * 2015-04-17 2016-12-08 日本化薬株式会社 水溶性アゾ化合物又はその塩、インク組成物及び着色体

Also Published As

Publication number Publication date
DK3856711T3 (da) 2022-12-12
IL281637A (en) 2021-05-31
GB201815696D0 (en) 2018-11-07
AU2019349863A1 (en) 2021-04-15
CA3112998A1 (en) 2020-04-02
EP3856711B1 (en) 2022-11-16
ES2933568T3 (es) 2023-02-10
US20210340108A1 (en) 2021-11-04
WO2020065324A1 (en) 2020-04-02
KR20210065111A (ko) 2021-06-03
EP3856711A1 (en) 2021-08-04
CN112839923A (zh) 2021-05-25

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