JP2022502400A5 - - Google Patents
Info
- Publication number
- JP2022502400A5 JP2022502400A5 JP2021516883A JP2021516883A JP2022502400A5 JP 2022502400 A5 JP2022502400 A5 JP 2022502400A5 JP 2021516883 A JP2021516883 A JP 2021516883A JP 2021516883 A JP2021516883 A JP 2021516883A JP 2022502400 A5 JP2022502400 A5 JP 2022502400A5
- Authority
- JP
- Japan
- Prior art keywords
- compound
- optionally
- dimethyl sulfoxide
- reaction mass
- water
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB1815695.0 | 2018-09-26 | ||
| GBGB1815695.0A GB201815695D0 (en) | 2018-09-26 | 2018-09-26 | Synthetic method |
| PCT/GB2019/052718 WO2020065323A1 (en) | 2018-09-26 | 2019-09-26 | Synthetic method for the preparation of a 3-[5-amino-4-(3-cyanobenzoyl)-pyrazol compound |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2022502400A JP2022502400A (ja) | 2022-01-11 |
| JP2022502400A5 true JP2022502400A5 (https=) | 2022-12-14 |
| JP7291782B2 JP7291782B2 (ja) | 2023-06-15 |
Family
ID=64024269
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2021516883A Active JP7291782B2 (ja) | 2018-09-26 | 2019-09-26 | ３－［５－アミノ－４－（３－シアノベンゾイル）－ピラゾール化合物の調製のための合成方法 |
Country Status (12)
| Country | Link |
|---|---|
| US (1) | US11649213B2 (https=) |
| EP (1) | EP3856721B1 (https=) |
| JP (1) | JP7291782B2 (https=) |
| KR (1) | KR102711257B1 (https=) |
| CN (1) | CN112839928B (https=) |
| AU (1) | AU2019350525B2 (https=) |
| CA (1) | CA3112993A1 (https=) |
| DK (1) | DK3856721T3 (https=) |
| ES (1) | ES2943289T3 (https=) |
| GB (1) | GB201815695D0 (https=) |
| IL (1) | IL281636B2 (https=) |
| WO (1) | WO2020065323A1 (https=) |
Family Cites Families (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE1809386A1 (de) | 1968-11-16 | 1970-06-11 | Bayer Ag | Verfahren zur Herstellung von 1,5-disubstituierten 4-Cyanopyrazolen |
| US4686221A (en) * | 1985-10-01 | 1987-08-11 | Kanebo, Ltd. | Quinolinecarboxylic acid compounds and antimicrobial agent containing the same |
| US6005109A (en) * | 1997-10-30 | 1999-12-21 | Pflizer Inc. | Pyrazoles and pyrazolopyrimidines having CRF antagonistic activity |
| US6103900A (en) * | 1992-12-17 | 2000-08-15 | Pfizer Inc | Pyrazoles and pyrazolopyrimidines having CRF antagonistic activity |
| FR2732967B1 (fr) | 1995-04-11 | 1997-07-04 | Sanofi Sa | 1-phenylpyrazole-3-carboxamides substitues, actifs sur la neurotensine, leur preparation, les compositions pharmaceutiques en contenant |
| GB9608435D0 (en) * | 1996-04-24 | 1996-06-26 | Celltech Therapeutics Ltd | Chemical compounds |
| HRP20000724A2 (en) * | 1998-05-05 | 2001-06-30 | Hoffmann La Roche | Pyrazole derivatives as p-38 map kinase inhibitors |
| PL2298743T3 (pl) | 2003-06-26 | 2013-02-28 | Novartis Ag | Inhibitory kinaz P38 na bazie 5-członowych heterocykli |
| WO2005007632A1 (en) | 2003-07-18 | 2005-01-27 | Pharmacia Corporation | Substituted pyridazinones as inhibitors of p38 |
| US7485657B2 (en) | 2004-05-12 | 2009-02-03 | Boehringer Ingelheim Pharmaceuticals, Inc. | Anti-cytokine heterocyclic compounds |
| ATE510836T1 (de) | 2006-01-19 | 2011-06-15 | Matrix Lab Ltd | Umwandlung eines aromatischen diazoniumsalzes in ein arylhydrazin |
| AU2008281594A1 (en) | 2007-08-02 | 2009-02-05 | Generics [Uk] Limited | Novel process |
| WO2009088025A1 (ja) | 2008-01-10 | 2009-07-16 | Hokko Chemical Industry Co., Ltd. | フェニルトリアゾリノン類の製造法 |
| JP5602387B2 (ja) | 2008-05-02 | 2014-10-08 | キヤノン株式会社 | インクジェット用インク、インクジェット記録方法、インクカートリッジ、記録ユニット、及びインクジェット記録装置 |
| CN102964270B (zh) | 2012-11-21 | 2015-01-07 | 合肥星宇化学有限责任公司 | 一种亚硫酸钠还原重氮盐合成肼的方法 |
| WO2018059533A1 (zh) | 2016-09-29 | 2018-04-05 | 南京明德新药研发股份有限公司 | p38αMAPK激酶抑制剂及其制备方法和应用 |
-
2018
- 2018-09-26 GB GBGB1815695.0A patent/GB201815695D0/en not_active Ceased
-
2019
- 2019-09-26 CN CN201980063294.3A patent/CN112839928B/zh active Active
- 2019-09-26 WO PCT/GB2019/052718 patent/WO2020065323A1/en not_active Ceased
- 2019-09-26 KR KR1020217008904A patent/KR102711257B1/ko active Active
- 2019-09-26 EP EP19780305.9A patent/EP3856721B1/en active Active
- 2019-09-26 IL IL281636A patent/IL281636B2/en unknown
- 2019-09-26 ES ES19780305T patent/ES2943289T3/es active Active
- 2019-09-26 US US17/279,553 patent/US11649213B2/en active Active
- 2019-09-26 CA CA3112993A patent/CA3112993A1/en active Pending
- 2019-09-26 JP JP2021516883A patent/JP7291782B2/ja active Active
- 2019-09-26 DK DK19780305.9T patent/DK3856721T3/da active
- 2019-09-26 AU AU2019350525A patent/AU2019350525B2/en active Active
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