JP2021533087A5 - - Google Patents
Info
- Publication number
- JP2021533087A5 JP2021533087A5 JP2020571842A JP2020571842A JP2021533087A5 JP 2021533087 A5 JP2021533087 A5 JP 2021533087A5 JP 2020571842 A JP2020571842 A JP 2020571842A JP 2020571842 A JP2020571842 A JP 2020571842A JP 2021533087 A5 JP2021533087 A5 JP 2021533087A5
- Authority
- JP
- Japan
- Prior art keywords
- group
- substituted
- unsubstituted
- alkyl
- cyano
- Prior art date
Links
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2024096077A JP2024133496A (ja) | 2018-06-26 | 2024-06-13 | 神経炎症におけるマクロファージコロニー刺激因子１受容体（ｃｓｆ１ｒ）をイメージングするための陽電子放射断層撮影（ｐｅｔ）放射性トレーサー |
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201862689958P | 2018-06-26 | 2018-06-26 | |
| US62/689,958 | 2018-06-26 | ||
| PCT/US2019/039234 WO2020006075A1 (en) | 2018-06-26 | 2019-06-26 | Positron emission tomography (pet) radiotracers for imaging macrophage colony-stimulating factor 1 receptor (csf1r) in neuroinflammation |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2024096077A Division JP2024133496A (ja) | 2018-06-26 | 2024-06-13 | 神経炎症におけるマクロファージコロニー刺激因子１受容体（ｃｓｆ１ｒ）をイメージングするための陽電子放射断層撮影（ｐｅｔ）放射性トレーサー |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2021533087A JP2021533087A (ja) | 2021-12-02 |
| JP2021533087A5 true JP2021533087A5 (https=) | 2022-07-25 |
| JPWO2020006075A5 JPWO2020006075A5 (https=) | 2022-07-25 |
Family
ID=68985080
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2020571842A Pending JP2021533087A (ja) | 2018-06-26 | 2019-06-26 | 神経炎症におけるマクロファージコロニー刺激因子１受容体（ｃｓｆ１ｒ）をイメージングするための陽電子放射断層撮影（ｐｅｔ）放射性トレーサー |
| JP2024096077A Pending JP2024133496A (ja) | 2018-06-26 | 2024-06-13 | 神経炎症におけるマクロファージコロニー刺激因子１受容体（ｃｓｆ１ｒ）をイメージングするための陽電子放射断層撮影（ｐｅｔ）放射性トレーサー |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2024096077A Pending JP2024133496A (ja) | 2018-06-26 | 2024-06-13 | 神経炎症におけるマクロファージコロニー刺激因子１受容体（ｃｓｆ１ｒ）をイメージングするための陽電子放射断層撮影（ｐｅｔ）放射性トレーサー |
Country Status (12)
| Country | Link |
|---|---|
| US (1) | US20210290784A1 (https=) |
| EP (1) | EP3813890A4 (https=) |
| JP (2) | JP2021533087A (https=) |
| KR (1) | KR20210013769A (https=) |
| CN (2) | CN118743770A (https=) |
| AU (1) | AU2019294699B2 (https=) |
| BR (1) | BR112020026602A2 (https=) |
| CA (1) | CA3104520A1 (https=) |
| EA (1) | EA202092843A1 (https=) |
| IL (1) | IL279768B2 (https=) |
| MX (1) | MX2021000141A (https=) |
| WO (1) | WO2020006075A1 (https=) |
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2020132651A1 (en) | 2018-12-20 | 2020-06-25 | Amgen Inc. | Kif18a inhibitors |
| EP3898616B1 (en) | 2018-12-20 | 2024-10-02 | Amgen Inc. | Heteroaryl amides useful as kif18a inhibitors |
| JP7676308B2 (ja) * | 2018-12-20 | 2025-05-14 | アムジエン・インコーポレーテツド | Ｋｉｆ１８ａ阻害剤として有用なヘテロアリールアミド |
| US12540129B2 (en) | 2019-08-02 | 2026-02-03 | Amgen Inc. | KIF18A inhibitors |
| WO2021026099A1 (en) | 2019-08-02 | 2021-02-11 | Amgen Inc. | Kif18a inhibitors |
| EP4269404A4 (en) * | 2020-12-25 | 2024-12-04 | Xizang Haisco Pharmaceutical Co., Ltd. | KETOHEXOKINASE INHIBITORS AND USE THEREOF |
| CA3221884A1 (en) * | 2021-06-11 | 2022-12-15 | Norman Lafrance | Expert scoring system for measurement of severity, treatment response and prognosis of peripheral arterial disease |
| AU2024214768A1 (en) * | 2023-01-30 | 2025-08-07 | The Johns Hopkins University | 18 f-labeled pet radiotracers for imaging macrophage colony stimulating factor 1 receptor |
| CN118027009B (zh) * | 2024-04-15 | 2024-07-12 | 北京师范大学 | 一类靶向于csf1r激酶的苯基酰胺类化合物及其应用 |
| CN119498255B (zh) * | 2024-10-24 | 2025-11-25 | 香港理工大学深圳研究院 | 一种抑郁症小鼠模型及其构建方法与应用 |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2006047504A1 (en) * | 2004-10-22 | 2006-05-04 | Janssen Pharmaceutica, N.V. | Aromatic amides as inhibitors of c-fms kinase |
| CN109069666B (zh) * | 2016-04-29 | 2023-04-04 | 纪念斯隆凯特琳癌症中心 | 使靶向颗粒穿透、分布和响应于恶性脑肿瘤中的组合物和方法 |
-
2019
- 2019-06-26 CN CN202410732670.6A patent/CN118743770A/zh active Pending
- 2019-06-26 WO PCT/US2019/039234 patent/WO2020006075A1/en not_active Ceased
- 2019-06-26 AU AU2019294699A patent/AU2019294699B2/en active Active
- 2019-06-26 EA EA202092843A patent/EA202092843A1/ru unknown
- 2019-06-26 MX MX2021000141A patent/MX2021000141A/es unknown
- 2019-06-26 CA CA3104520A patent/CA3104520A1/en active Pending
- 2019-06-26 US US17/253,336 patent/US20210290784A1/en active Pending
- 2019-06-26 EP EP19825817.0A patent/EP3813890A4/en active Pending
- 2019-06-26 CN CN201980056945.6A patent/CN112638431A/zh active Pending
- 2019-06-26 BR BR112020026602-7A patent/BR112020026602A2/pt unknown
- 2019-06-26 JP JP2020571842A patent/JP2021533087A/ja active Pending
- 2019-06-26 KR KR1020217002632A patent/KR20210013769A/ko not_active Ceased
- 2019-06-26 IL IL279768A patent/IL279768B2/en unknown
-
2024
- 2024-06-13 JP JP2024096077A patent/JP2024133496A/ja active Pending
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