JP2021523240A5 - - Google Patents

Info

Publication number
JP2021523240A5
JP2021523240A5 JP2021514291A JP2021514291A JP2021523240A5 JP 2021523240 A5 JP2021523240 A5 JP 2021523240A5 JP 2021514291 A JP2021514291 A JP 2021514291A JP 2021514291 A JP2021514291 A JP 2021514291A JP 2021523240 A5 JP2021523240 A5 JP 2021523240A5
Authority
JP
Japan
Prior art keywords
formula
hydrogen
ring
pharmaceutically acceptable
group
Prior art date
Application number
JP2021514291A
Other languages
English (en)
Japanese (ja)
Other versions
JP7344959B2 (ja
JPWO2019222154A5 (https=
JP2021523240A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2019/032127 external-priority patent/WO2019222154A1/en
Publication of JP2021523240A publication Critical patent/JP2021523240A/ja
Publication of JPWO2019222154A5 publication Critical patent/JPWO2019222154A5/ja
Publication of JP2021523240A5 publication Critical patent/JP2021523240A5/ja
Priority to JP2023142664A priority Critical patent/JP7656669B2/ja
Application granted granted Critical
Publication of JP7344959B2 publication Critical patent/JP7344959B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2021514291A 2018-05-15 2019-05-14 マトリックスメタロプロテイナーゼ(mmp)阻害剤及びその使用方法 Active JP7344959B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2023142664A JP7656669B2 (ja) 2018-05-15 2023-09-04 マトリックスメタロプロテイナーゼ(mmp)阻害剤及びその使用方法

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201862671753P 2018-05-15 2018-05-15
US62/671,753 2018-05-15
PCT/US2019/032127 WO2019222154A1 (en) 2018-05-15 2019-05-14 Matrix metalloproteinase (mmp) inhibitors and methods of use thereof

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2023142664A Division JP7656669B2 (ja) 2018-05-15 2023-09-04 マトリックスメタロプロテイナーゼ(mmp)阻害剤及びその使用方法

Publications (4)

Publication Number Publication Date
JP2021523240A JP2021523240A (ja) 2021-09-02
JPWO2019222154A5 JPWO2019222154A5 (https=) 2022-05-11
JP2021523240A5 true JP2021523240A5 (https=) 2022-05-11
JP7344959B2 JP7344959B2 (ja) 2023-09-14

Family

ID=66690981

Family Applications (4)

Application Number Title Priority Date Filing Date
JP2021514292A Active JP7343571B2 (ja) 2018-05-15 2019-05-14 マトリックスメタロプロテイナーゼ(mmp)阻害剤及びその使用方法
JP2021514291A Active JP7344959B2 (ja) 2018-05-15 2019-05-14 マトリックスメタロプロテイナーゼ(mmp)阻害剤及びその使用方法
JP2023140718A Pending JP2023164905A (ja) 2018-05-15 2023-08-31 マトリックスメタロプロテイナーゼ(mmp)阻害剤及びその使用方法
JP2023142664A Active JP7656669B2 (ja) 2018-05-15 2023-09-04 マトリックスメタロプロテイナーゼ(mmp)阻害剤及びその使用方法

Family Applications Before (1)

Application Number Title Priority Date Filing Date
JP2021514292A Active JP7343571B2 (ja) 2018-05-15 2019-05-14 マトリックスメタロプロテイナーゼ(mmp)阻害剤及びその使用方法

Family Applications After (2)

Application Number Title Priority Date Filing Date
JP2023140718A Pending JP2023164905A (ja) 2018-05-15 2023-08-31 マトリックスメタロプロテイナーゼ(mmp)阻害剤及びその使用方法
JP2023142664A Active JP7656669B2 (ja) 2018-05-15 2023-09-04 マトリックスメタロプロテイナーゼ(mmp)阻害剤及びその使用方法

Country Status (20)

Country Link
US (6) US20190352288A1 (https=)
EP (4) EP4335499A3 (https=)
JP (4) JP7343571B2 (https=)
KR (3) KR102861502B1 (https=)
CN (3) CN112424186A (https=)
AU (3) AU2019269409B2 (https=)
BR (1) BR112020023269A2 (https=)
CA (2) CA3100320A1 (https=)
DK (2) DK3793995T3 (https=)
ES (2) ES2978192T3 (https=)
FI (2) FI3793992T3 (https=)
HU (2) HUE066619T2 (https=)
LT (1) LT3793995T (https=)
MY (1) MY199200A (https=)
PL (1) PL3793995T3 (https=)
PT (2) PT3793992T (https=)
SG (2) SG11202011316RA (https=)
SI (1) SI3793995T1 (https=)
TW (3) TWI827601B (https=)
WO (2) WO2019222157A1 (https=)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US10532102B2 (en) * 2016-08-19 2020-01-14 Foresee Pharmaceuticals Co., Ltd. Pharmaceutical composition and methods of uses
SI3793995T1 (sl) 2018-05-15 2024-05-31 Foresee Pharmaceuticals Usa, Inc. Zaviralci matrične metaloproteinaze (mmp)in načini njihove uporabe
CA3158234A1 (en) * 2019-11-14 2021-05-20 Foresee Pharmaceuticals Co., Ltd. Matrix metalloproteinase (mmp) inhibitors and methods of use thereof
EP4351566A4 (en) * 2021-06-08 2025-04-23 Foresee Pharmaceuticals USA, Inc. SAFE ADMINISTRATION OF MMP-12 INHIBITOR
TW202313011A (zh) * 2021-06-08 2023-04-01 逸達生物科技股份有限公司 Mmp抑制劑於治療急性呼吸窘迫綜合症之用途
EP4198033A1 (en) 2021-12-14 2023-06-21 Basf Se Heterocyclic compounds for the control of invertebrate pests
WO2023110473A1 (en) 2021-12-14 2023-06-22 Basf Se Heterocyclic compounds for the control of invertebrate pests

Family Cites Families (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2482618A1 (fr) 1980-05-16 1981-11-20 Inst Corps Gras Iterg Procede de conjugaison catalytique de corps gras polyinsatures, produits obtenus et application
US6352976B1 (en) 1998-12-31 2002-03-05 Aventis Pharmaceuticals Inc. Selective inhibitors of MMP-12
EP1150975A1 (en) 1998-12-31 2001-11-07 Aventis Pharmaceuticals Inc. 1-carboxymethyl-2-oxo-azepan derivatives useful as selective inhibitors of mmp-12
EP1288199A4 (en) 2000-04-28 2005-10-12 Shionogi & Co INHIBITORS OF MMP-12
JP2004527511A (ja) 2001-03-15 2004-09-09 アストラゼネカ・アクチエボラーグ メタロプロテイナーゼ阻害剤
SE0100903D0 (sv) 2001-03-15 2001-03-15 Astrazeneca Ab Compounds
US6890915B2 (en) 2001-05-25 2005-05-10 Bristol-Myers Squibb Pharma Company Hydantoins and related heterocycles as inhibitors of matrix metalloproteinases and/or TNF-α converting enzyme (TACE)
EP1394159A1 (fr) 2002-08-13 2004-03-03 Warner-Lambert Company LLC Nouveaux dérivés de thiophène, leur procédé de préparation et les compositions pharmaceutiques qui les contiennent
SE0202539D0 (sv) 2002-08-27 2002-08-27 Astrazeneca Ab Compounds
AU2003282920A1 (en) 2002-10-04 2004-05-04 Bristol-Myers Squibb Company Hydantoin derivatives as inhibitors of matrix metalloproteinases and/or tnf-alpha converting enzyme (tace)
US7132432B2 (en) * 2003-06-05 2006-11-07 Bristol-Myers Squibb Company Hydantoin derivatives as inhibitors of tumor necrosis factor-alpha converting enzyme (TACE)
JP5042833B2 (ja) 2004-08-19 2012-10-03 クエスト ファーマシューティカル サーヴィシーズ マクロファージエラスターゼの阻害剤としての5−[3−(4−ベンジルオキシフェニルチオ)−フラ−2−イル]−イミダゾリジン−2,4−ジオン及び類似体
EP2797002A4 (en) 2011-12-21 2015-05-20 Panasonic Corp DATA PROCESSING DEVICE, DATA TRANSMISSION DEVICE, DATA PROCESSING SYSTEM, DATA PROCESSING METHOD AND DATA TRANSMISSION METHOD
SI3793995T1 (sl) * 2018-05-15 2024-05-31 Foresee Pharmaceuticals Usa, Inc. Zaviralci matrične metaloproteinaze (mmp)in načini njihove uporabe

Similar Documents

Publication Publication Date Title
JP2021523240A5 (https=)
CA2913634C (en) Small molecule inhibitors of fibrosis
CA2509981C (en) Hetero substitued sodium channel blockers
AU2003211135B2 (en) Sodium channel blockers
CN109863140A (zh) 3-氧代-2,6-二苯基-2,3-二氢哒嗪-4-甲酰胺
JP2019519598A5 (https=)
RU2020121150A (ru) Твердые формы ингибитора калликреина плазмы и его солей
RU2006134020A (ru) Конденсированные производные пиразола
JP2021523241A5 (https=)
JP6039549B2 (ja) 化学療法または放射線療法によって誘発される嘔吐を予防および/または治療するためのシグマリガンド
JP2014503574A5 (https=)
UA104997C2 (uk) Аміди азотвмісних насичених гетероциклів та 3,5-діаміно-6-хлор-2-піразинкарбонової кислоти як лікарський засіб
TW200911232A (en) Novel therapeutic compounds
US10336735B2 (en) Small molecule inhibitors of fibrosis
RU2713179C2 (ru) Антимитотические амиды для лечения рака и пролиферативных заболеваний
CA3159791A1 (en) Hexahydro-2h-pyrazino[1,2-a]pyrazine-6,9-dione derivatives and pharmaceutical compositions for prevention or treatment of cancer comprising same
JPWO2019222154A5 (https=)
JPWO2019031470A1 (ja) 新規アミド系化合物、並びにそれを用いたPin1阻害剤、炎症性疾患の治療剤及び癌の治療剤
JP6982716B2 (ja) 複素環式化合物及びその使用
CA2903464A1 (en) Treatment of cancer and other conditions using a transcription factor modulator
KR101392086B1 (ko) 신규 5각 헤테로 고리 유도체 및 그 제조방법
JPWO2019222157A5 (https=)
RU2010118458A (ru) Производное изоксазола для лечения рака
KR102315866B1 (ko) 섬유화 질환 복합 치료제 개발
JP2017506617A (ja) 未制御細胞成長の阻害のための化合物