JP2021523240A5 - - Google Patents
Info
- Publication number
- JP2021523240A5 JP2021523240A5 JP2021514291A JP2021514291A JP2021523240A5 JP 2021523240 A5 JP2021523240 A5 JP 2021523240A5 JP 2021514291 A JP2021514291 A JP 2021514291A JP 2021514291 A JP2021514291 A JP 2021514291A JP 2021523240 A5 JP2021523240 A5 JP 2021523240A5
- Authority
- JP
- Japan
- Prior art keywords
- formula
- hydrogen
- ring
- pharmaceutically acceptable
- group
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2023142664A JP7656669B2 (ja) | 2018-05-15 | 2023-09-04 | マトリックスメタロプロテイナーゼ(mmp)阻害剤及びその使用方法 |
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201862671753P | 2018-05-15 | 2018-05-15 | |
| US62/671,753 | 2018-05-15 | ||
| PCT/US2019/032127 WO2019222154A1 (en) | 2018-05-15 | 2019-05-14 | Matrix metalloproteinase (mmp) inhibitors and methods of use thereof |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2023142664A Division JP7656669B2 (ja) | 2018-05-15 | 2023-09-04 | マトリックスメタロプロテイナーゼ(mmp)阻害剤及びその使用方法 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2021523240A JP2021523240A (ja) | 2021-09-02 |
| JP2021523240A5 true JP2021523240A5 (enExample) | 2022-05-11 |
| JP7344959B2 JP7344959B2 (ja) | 2023-09-14 |
Family
ID=66690981
Family Applications (4)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2021514291A Active JP7344959B2 (ja) | 2018-05-15 | 2019-05-14 | マトリックスメタロプロテイナーゼ(mmp)阻害剤及びその使用方法 |
| JP2021514292A Active JP7343571B2 (ja) | 2018-05-15 | 2019-05-14 | マトリックスメタロプロテイナーゼ(mmp)阻害剤及びその使用方法 |
| JP2023140718A Pending JP2023164905A (ja) | 2018-05-15 | 2023-08-31 | マトリックスメタロプロテイナーゼ(mmp)阻害剤及びその使用方法 |
| JP2023142664A Active JP7656669B2 (ja) | 2018-05-15 | 2023-09-04 | マトリックスメタロプロテイナーゼ(mmp)阻害剤及びその使用方法 |
Family Applications After (3)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2021514292A Active JP7343571B2 (ja) | 2018-05-15 | 2019-05-14 | マトリックスメタロプロテイナーゼ(mmp)阻害剤及びその使用方法 |
| JP2023140718A Pending JP2023164905A (ja) | 2018-05-15 | 2023-08-31 | マトリックスメタロプロテイナーゼ(mmp)阻害剤及びその使用方法 |
| JP2023142664A Active JP7656669B2 (ja) | 2018-05-15 | 2023-09-04 | マトリックスメタロプロテイナーゼ(mmp)阻害剤及びその使用方法 |
Country Status (20)
| Country | Link |
|---|---|
| US (6) | US12258335B1 (enExample) |
| EP (4) | EP4349332A3 (enExample) |
| JP (4) | JP7344959B2 (enExample) |
| KR (3) | KR102861502B1 (enExample) |
| CN (3) | CN119462623A (enExample) |
| AU (3) | AU2019269409B2 (enExample) |
| BR (1) | BR112020023269A2 (enExample) |
| CA (2) | CA3100319A1 (enExample) |
| DK (2) | DK3793992T3 (enExample) |
| ES (2) | ES2978192T3 (enExample) |
| FI (2) | FI3793995T3 (enExample) |
| HU (2) | HUE066627T2 (enExample) |
| LT (1) | LT3793995T (enExample) |
| MY (1) | MY199200A (enExample) |
| PL (1) | PL3793995T3 (enExample) |
| PT (2) | PT3793992T (enExample) |
| SG (2) | SG11202011316RA (enExample) |
| SI (1) | SI3793995T1 (enExample) |
| TW (3) | TWI798435B (enExample) |
| WO (2) | WO2019222154A1 (enExample) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US10532102B2 (en) | 2016-08-19 | 2020-01-14 | Foresee Pharmaceuticals Co., Ltd. | Pharmaceutical composition and methods of uses |
| KR102861502B1 (ko) * | 2018-05-15 | 2025-09-18 | 포시 파마슈티컬스 유에스에이 인코포레이티드 | 기질 금속단백분해효소 (mmp) 억제제 및 이의 사용 방법 |
| CN115667227B (zh) | 2019-11-14 | 2024-11-01 | 逸达生物科技股份有限公司 | 基质金属蛋白酶(mmp)抑制剂及其使用方法 |
| JP2024520818A (ja) * | 2021-06-08 | 2024-05-24 | フォアシー ファーマシューティカルズ カンパニー リミテッド | 急性呼吸促迫症候群を処置するためのmmp阻害薬の使用 |
| EP4351566A4 (en) * | 2021-06-08 | 2025-04-23 | Foresee Pharmaceuticals USA, Inc. | SAFE ADMINISTRATION OF MMP-12 INHIBITOR |
| WO2023110473A1 (en) | 2021-12-14 | 2023-06-22 | Basf Se | Heterocyclic compounds for the control of invertebrate pests |
| EP4198033A1 (en) | 2021-12-14 | 2023-06-21 | Basf Se | Heterocyclic compounds for the control of invertebrate pests |
Family Cites Families (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2482618A1 (fr) | 1980-05-16 | 1981-11-20 | Inst Corps Gras Iterg | Procede de conjugaison catalytique de corps gras polyinsatures, produits obtenus et application |
| US6352976B1 (en) | 1998-12-31 | 2002-03-05 | Aventis Pharmaceuticals Inc. | Selective inhibitors of MMP-12 |
| AU1817700A (en) | 1998-12-31 | 2000-07-24 | Aventis Pharmaceuticals Inc. | 1-carboxymethyl-2-oxo-azepan derivatives useful as selective inhibitors of mmp-12 |
| AU4882101A (en) | 2000-04-28 | 2001-11-12 | Shionogi & Co., Ltd. | Mmp-12 inhibitors |
| SE0100903D0 (sv) | 2001-03-15 | 2001-03-15 | Astrazeneca Ab | Compounds |
| KR20030082990A (ko) * | 2001-03-15 | 2003-10-23 | 아스트라제네카 아베 | 메탈로프로테이나제 억제제 |
| CA2447475A1 (en) | 2001-05-25 | 2002-12-05 | Chu-Biao Xue | Hydantion derivatives as inhibitors of matrix metalloproteinases |
| EP1394159A1 (fr) | 2002-08-13 | 2004-03-03 | Warner-Lambert Company LLC | Nouveaux dérivés de thiophène, leur procédé de préparation et les compositions pharmaceutiques qui les contiennent |
| SE0202539D0 (sv) | 2002-08-27 | 2002-08-27 | Astrazeneca Ab | Compounds |
| US7041693B2 (en) | 2002-10-04 | 2006-05-09 | Bristol-Myers Squibb Company | Hydantoin derivatives as inhibitors of matrix metalloproteinases and/or TNF-α converting enzyme (TACE) |
| US7132432B2 (en) | 2003-06-05 | 2006-11-07 | Bristol-Myers Squibb Company | Hydantoin derivatives as inhibitors of tumor necrosis factor-alpha converting enzyme (TACE) |
| DK1789036T3 (da) * | 2004-08-19 | 2011-06-27 | Quest Pharmaceutical Services | 5-[3-(4-benzyloxyphenylthio)-fur-2-yl]-imidazolidin-2,4-dion og analoger som inhibitorer af makrofagelastase |
| JP5357365B1 (ja) | 2011-12-21 | 2013-12-04 | パナソニック株式会社 | データ処理装置、データ送信装置、データ処理システム、データ処理方法、及び、データ送信方法 |
| KR102861502B1 (ko) | 2018-05-15 | 2025-09-18 | 포시 파마슈티컬스 유에스에이 인코포레이티드 | 기질 금속단백분해효소 (mmp) 억제제 및 이의 사용 방법 |
-
2019
- 2019-05-14 KR KR1020207035504A patent/KR102861502B1/ko active Active
- 2019-05-14 CN CN202411619226.XA patent/CN119462623A/zh active Pending
- 2019-05-14 ES ES19728197T patent/ES2978192T3/es active Active
- 2019-05-14 JP JP2021514291A patent/JP7344959B2/ja active Active
- 2019-05-14 CA CA3100319A patent/CA3100319A1/en active Pending
- 2019-05-14 WO PCT/US2019/032127 patent/WO2019222154A1/en not_active Ceased
- 2019-05-14 CN CN201980047375.4A patent/CN112424192B/zh active Active
- 2019-05-14 PT PT197313745T patent/PT3793992T/pt unknown
- 2019-05-14 KR KR1020207035503A patent/KR102761591B1/ko active Active
- 2019-05-14 AU AU2019269409A patent/AU2019269409B2/en active Active
- 2019-05-14 JP JP2021514292A patent/JP7343571B2/ja active Active
- 2019-05-14 ES ES19731374T patent/ES2984594T3/es active Active
- 2019-05-14 TW TW108116632A patent/TWI798435B/zh active
- 2019-05-14 FI FIEP19728197.5T patent/FI3793995T3/fi active
- 2019-05-14 US US17/055,483 patent/US12258335B1/en active Active
- 2019-05-14 MY MYPI2020005983A patent/MY199200A/en unknown
- 2019-05-14 DK DK19731374.5T patent/DK3793992T3/da active
- 2019-05-14 SI SI201930733T patent/SI3793995T1/sl unknown
- 2019-05-14 SG SG11202011316RA patent/SG11202011316RA/en unknown
- 2019-05-14 CN CN201980047333.0A patent/CN112424186A/zh active Pending
- 2019-05-14 HU HUE19731374A patent/HUE066627T2/hu unknown
- 2019-05-14 US US17/055,459 patent/US11739080B2/en active Active
- 2019-05-14 TW TW108116631A patent/TWI827601B/zh active
- 2019-05-14 HU HUE19728197A patent/HUE066619T2/hu unknown
- 2019-05-14 KR KR1020257002624A patent/KR20250021604A/ko active Pending
- 2019-05-14 LT LTEPPCT/US2019/032131T patent/LT3793995T/lt unknown
- 2019-05-14 FI FIEP19731374.5T patent/FI3793992T3/fi active
- 2019-05-14 PT PT197281975T patent/PT3793995T/pt unknown
- 2019-05-14 SG SG11202011318QA patent/SG11202011318QA/en unknown
- 2019-05-14 WO PCT/US2019/032131 patent/WO2019222157A1/en not_active Ceased
- 2019-05-14 EP EP24150920.7A patent/EP4349332A3/en active Pending
- 2019-05-14 PL PL19728197.5T patent/PL3793995T3/pl unknown
- 2019-05-14 BR BR112020023269-6A patent/BR112020023269A2/pt unknown
- 2019-05-14 AU AU2019270975A patent/AU2019270975B2/en active Active
- 2019-05-14 EP EP24150915.7A patent/EP4335499A3/en active Pending
- 2019-05-14 US US16/411,402 patent/US10851089B2/en active Active
- 2019-05-14 EP EP19731374.5A patent/EP3793992B1/en active Active
- 2019-05-14 DK DK19728197.5T patent/DK3793995T3/da active
- 2019-05-14 TW TW112115526A patent/TWI895726B/zh active
- 2019-05-14 CA CA3100320A patent/CA3100320A1/en active Pending
- 2019-05-14 EP EP19728197.5A patent/EP3793995B1/en active Active
- 2019-05-14 US US16/411,336 patent/US20190352288A1/en not_active Abandoned
-
2023
- 2023-07-06 US US18/347,674 patent/US12215096B2/en active Active
- 2023-08-31 JP JP2023140718A patent/JP2023164905A/ja active Pending
- 2023-09-04 JP JP2023142664A patent/JP7656669B2/ja active Active
-
2024
- 2024-01-18 AU AU2024200323A patent/AU2024200323B2/en active Active
- 2024-12-17 US US18/983,692 patent/US20250115590A1/en active Pending
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| JP2021523240A5 (enExample) | ||
| CA2913634C (en) | Small molecule inhibitors of fibrosis | |
| CA2509981C (en) | Hetero substitued sodium channel blockers | |
| AU2003211135B2 (en) | Sodium channel blockers | |
| JP2019519598A5 (enExample) | ||
| RU2020121150A (ru) | Твердые формы ингибитора калликреина плазмы и его солей | |
| RU2006134020A (ru) | Конденсированные производные пиразола | |
| JP2021523241A5 (enExample) | ||
| JP2014503574A5 (enExample) | ||
| MY152955A (en) | Pyrazine-2-carboxamide derivatives to treat diseases mediated by blockade of the epithelial sodium channel | |
| TW200911232A (en) | Novel therapeutic compounds | |
| JP6019126B2 (ja) | 有機ニトロチオエーテル化合物およびその医療用途 | |
| US10336735B2 (en) | Small molecule inhibitors of fibrosis | |
| JP2016199563A (ja) | 化学療法または放射線療法によって誘発される嘔吐を予防および/または治療するためのシグマリガンド | |
| JP2022514254A5 (enExample) | ||
| JPWO2019031472A1 (ja) | 新規アントラニル酸系化合物、並びにそれを用いたPin1阻害剤、炎症性疾患の治療剤及び癌の治療剤 | |
| CA3159791A1 (en) | Hexahydro-2h-pyrazino[1,2-a]pyrazine-6,9-dione derivatives and pharmaceutical compositions for prevention or treatment of cancer comprising same | |
| JPWO2019031470A1 (ja) | 新規アミド系化合物、並びにそれを用いたPin1阻害剤、炎症性疾患の治療剤及び癌の治療剤 | |
| JP6982716B2 (ja) | 複素環式化合物及びその使用 | |
| CA2903464A1 (en) | Treatment of cancer and other conditions using a transcription factor modulator | |
| RU2010118458A (ru) | Производное изоксазола для лечения рака | |
| KR102315866B1 (ko) | 섬유화 질환 복합 치료제 개발 | |
| KR20110095200A (ko) | 신규 5각 헤테로 고리 유도체 및 그 제조방법 | |
| JP2017506617A (ja) | 未制御細胞成長の阻害のための化合物 | |
| RU2801811C1 (ru) | Новое соединение и содержащая это соединение фармацевтическая композиция для предотвращения или лечения рака |