JP2021522206A5 - - Google Patents

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Publication number
JP2021522206A5
JP2021522206A5 JP2020558018A JP2020558018A JP2021522206A5 JP 2021522206 A5 JP2021522206 A5 JP 2021522206A5 JP 2020558018 A JP2020558018 A JP 2020558018A JP 2020558018 A JP2020558018 A JP 2020558018A JP 2021522206 A5 JP2021522206 A5 JP 2021522206A5
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Japan
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disease
group
pharmaceutically acceptable
ring
acceptable salt
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JP2020558018A
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English (en)
Japanese (ja)
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JP2021522206A (ja
JP7398391B2 (ja
JPWO2019204537A5 (https=
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JP2020558018A 2018-04-20 2019-04-18 Ｎ－［４－オキソ－２，３－ジヒドロ－１，５－ベンズオキサゼピン－３－イル］－５，６－ジヒドロ－４Ｈ－ピロロ［１，２－ｂ］ピラゾール－２－カルボキサミド誘導体及び例えば過敏性腸症候群（ＩＢＳ）を処置するためのＲＩＰ１キナーゼ阻害剤としての関連化合物 Active JP7398391B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201862660397P 2018-04-20 2018-04-20
US62/660,397 2018-04-20
PCT/US2019/028011 WO2019204537A1 (en) 2018-04-20 2019-04-18 N-[4-oxo-2,3-dihydro-1,5-benzoxazepin-3-yl]-5,6-dihydro-4h-pyrrolo[1,2-b]pyrazol e-2-carboxamide derivatives and related compounds as rip1 kinase inhibitors for treating e.g. irritable bowel syndrome (ibs)

Publications (4)

Publication Number Publication Date
JP2021522206A JP2021522206A (ja) 2021-08-30
JPWO2019204537A5 JPWO2019204537A5 (https=) 2022-04-22
JP2021522206A5 true JP2021522206A5 (https=) 2022-04-22
JP7398391B2 JP7398391B2 (ja) 2023-12-14

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JP2020558018A Active JP7398391B2 (ja) 2018-04-20 2019-04-18 Ｎ－［４－オキソ－２，３－ジヒドロ－１，５－ベンズオキサゼピン－３－イル］－５，６－ジヒドロ－４Ｈ－ピロロ［１，２－ｂ］ピラゾール－２－カルボキサミド誘導体及び例えば過敏性腸症候群（ＩＢＳ）を処置するためのＲＩＰ１キナーゼ阻害剤としての関連化合物

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US (1) US11634436B2 (https=)
EP (1) EP3781571B1 (https=)
JP (1) JP7398391B2 (https=)
CN (1) CN112074519B (https=)
WO (1) WO2019204537A1 (https=)

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