JP2021513569A - 抗菌及び殺精子潤滑剤 - Google Patents

抗菌及び殺精子潤滑剤 Download PDF

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Publication number
JP2021513569A
JP2021513569A JP2020565535A JP2020565535A JP2021513569A JP 2021513569 A JP2021513569 A JP 2021513569A JP 2020565535 A JP2020565535 A JP 2020565535A JP 2020565535 A JP2020565535 A JP 2020565535A JP 2021513569 A JP2021513569 A JP 2021513569A
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weight
guanidine
composition
composition according
biocide
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Pending
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JP2020565535A
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English (en)
Japanese (ja)
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JP2021513569A5 (enExample
Inventor
マイヤーホーファー ルーカス
マイヤーホーファー ルーカス
Original Assignee
ベーツェーエスカー バイオシッド ゲゼルシャフト ミット ベシュレンクテル ハフツング
ベーツェーエスカー バイオシッド ゲゼルシャフト ミット ベシュレンクテル ハフツング
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Publication of JP2021513569A publication Critical patent/JP2021513569A/ja
Publication of JP2021513569A5 publication Critical patent/JP2021513569A5/ja
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    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N47/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
    • A01N47/40—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having a double or triple bond to nitrogen, e.g. cyanates, cyanamides
    • A01N47/42—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having a double or triple bond to nitrogen, e.g. cyanates, cyanamides containing —N=CX2 groups, e.g. isothiourea
    • A01N47/44—Guanidine; Derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/74—Synthetic polymeric materials
    • A61K31/785—Polymers containing nitrogen
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N31/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic oxygen or sulfur compounds
    • A01N31/02—Acyclic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/075—Ethers or acetals
    • A61K31/085—Ethers or acetals having an ether linkage to aromatic ring nuclear carbon
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/13—Amines
    • A61K31/155—Amidines (), e.g. guanidine (H2N—C(=NH)—NH2), isourea (N=C(OH)—NH2), isothiourea (—N=C(SH)—NH2)
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/74—Synthetic polymeric materials
    • A61K31/765—Polymers containing oxygen
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/10—Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/36—Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
    • A61K47/38—Cellulose; Derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0034—Urogenital system, e.g. vagina, uterus, cervix, penis, scrotum, urethra, bladder; Personal lubricants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/02—Suppositories; Bougies; Bases therefor; Ovules
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/06—Ointments; Bases therefor; Other semi-solid forms, e.g. creams, sticks, gels
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/16—Masculine contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/18—Feminine contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2300/00—Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Reproductive Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Endocrinology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Gynecology & Obstetrics (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Plant Pathology (AREA)
  • Zoology (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Urology & Nephrology (AREA)
  • Dentistry (AREA)
  • Wood Science & Technology (AREA)
  • Environmental Sciences (AREA)
  • Inorganic Chemistry (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
JP2020565535A 2018-02-08 2019-02-08 抗菌及び殺精子潤滑剤 Pending JP2021513569A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP18155747.1 2018-02-08
EP18155747.1A EP3524055A1 (de) 2018-02-08 2018-02-08 Antibakterielles und spermizides gleitmittel
PCT/EP2019/053127 WO2019154983A1 (de) 2018-02-08 2019-02-08 Antibakterielles und spermizides gleitmittel

Publications (2)

Publication Number Publication Date
JP2021513569A true JP2021513569A (ja) 2021-05-27
JP2021513569A5 JP2021513569A5 (enExample) 2022-02-17

Family

ID=61188675

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JP2020565535A Pending JP2021513569A (ja) 2018-02-08 2019-02-08 抗菌及び殺精子潤滑剤

Country Status (9)

Country Link
US (1) US20210038637A1 (enExample)
EP (2) EP3524055A1 (enExample)
JP (1) JP2021513569A (enExample)
KR (1) KR20200119829A (enExample)
CN (1) CN111787802A (enExample)
BR (1) BR112020015955A2 (enExample)
MX (1) MX2020008140A (enExample)
RU (1) RU2020129407A (enExample)
WO (1) WO2019154983A1 (enExample)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE102022121007A1 (de) 2022-08-19 2024-02-22 pjur group Luxembourg S.A. Wasserbasierte Gleitmittelzusammensetzung
DE102022121008A1 (de) 2022-08-19 2024-02-22 pjur group Luxembourg S.A. Wasserfreie silikonbasierte Gleitmittelzusammensetzung

Citations (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH07145063A (ja) * 1993-07-28 1995-06-06 Johnson & Johnson Consumer Prod Inc 殺精子・抗ウイルス性潤滑剤組成物およびその使用方法
JP2006520329A (ja) * 2003-03-20 2006-09-07 ゲオファルマ プロドゥクツィオンスゲーエムベーハー 抗菌作用を有し、ジアミンをベースとするグアニジン誘導体
US20080051740A1 (en) * 2006-06-16 2008-02-28 Family Health International Vaginal drug delivery system and method
WO2008031105A1 (en) * 2006-09-08 2008-03-13 Delaval Holdings Ab Polymeric guanidine salt-based germicides
JP2010507721A (ja) * 2006-10-23 2010-03-11 アーチ・ケミカルズ・インコーポレーテッド 末端アミンの少ないビグアニド組成物
US20110269936A1 (en) * 2009-10-08 2011-11-03 Viktor Veniaminovich Tets Method for Producing Biocidal Polyguanidine, and Biocidal Polyguanidine
WO2015074730A1 (de) * 2013-11-21 2015-05-28 Farco-Pharma Gmbh Zusammensetzung, insbesondere in form eines gleitgels enthaltend ein lokalanästhetikum und polyhexanid
JP2017088603A (ja) * 2015-11-12 2017-05-25 グロック・ヘルス・サイエンス・アンド・リサーチ・ゲゼルシャフト・ミト・ベシュレンクテル・ハフツング 膣炎の治療

Family Cites Families (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2325586A (en) 1940-03-21 1943-08-03 Du Pont Polymeric guanidines and process for preparing the same
BR6568736D0 (pt) 1964-04-09 1973-08-14 Drug Inc Sterling Processo para preparar uma bisguanida
US5182104A (en) * 1991-07-16 1993-01-26 Stanley Marcus Topical virucidal composition for treatment of mucocutaneous tissue
US6028115A (en) 1995-10-13 2000-02-22 Rush-Presbyterian-St. Luke's Medical Center Method for preventing sexually transmitted diseases
AT406163B (de) 1998-04-22 2000-03-27 P O C Oil Industry Technology Verfahren zur gewinnung eines desinfektionsmittels
CN1121855C (zh) * 1999-04-28 2003-09-24 孙廷柱 可溶性杀菌消毒避孕套
CA2408191C (en) 2000-05-11 2006-11-14 P.O.C. Oil Industry Technology Beratungsges.M.B.H. Biocidal polymers based on guanidine salts
AT408302B (de) 2000-05-11 2001-10-25 P O C Oil Industry Technology Biozide polymere der reihe der polyoxyalkylen-guanidin-hydrochloride und verfahren zu deren herstellung
AT411060B (de) 2000-10-23 2003-09-25 P O C Oil Industry Technology Biozide polymere guanidinderivate auf der basis von diaminen und verfahren zur gewinnung von solchen salzen
WO2002030877A1 (fr) 2000-09-29 2002-04-18 Regionalnaya Obschestvennaya Organizatsya-Institut Ekologo-Tekhnologicheskikh Problem Procede de production d'un desinfectant
UA64406A (en) * 2003-05-27 2004-02-16 Neonila Havrylivna Barannik Ointment for complex treatment of ulcerated necrotic gingivostomatitis
AT505102B1 (de) 2004-11-05 2010-05-15 Schmidt Oskar Biozid, insbesondere fungizid wirkendes mittel
CA2676461A1 (en) 2006-12-29 2008-07-10 Aka Technology Gmbh Use of polymeric guanidines for controlling microorganisms
EP2071954A1 (de) * 2007-12-19 2009-06-24 Bayer CropScience AG Verwendung von polymeren Guanidin-Derivaten zum Bekämpfen von unerwünschten Mikro-organismen im Pflanzenschutz
AT505514B1 (de) 2007-07-16 2011-10-15 Aka Technology Gmbh Silikatischer füllstoff
EP2084967A1 (de) 2008-01-24 2009-08-05 Aka Central Research Laboratories GmbH Verfahren zur Bekämpfung unerwünschter Mikroorganismen an Bananenpflanzen
EP2230259A1 (de) 2009-03-18 2010-09-22 Mindinvest Holdings Ltd. Mikrobiozid wirkendes Polymergemisch
US20140228528A1 (en) 2011-11-02 2014-08-14 Mindinvest Holdings Ltd. Polyguanidine silicate and use thereof
US9386772B2 (en) * 2012-02-14 2016-07-12 Allegiance Corporation Antimicrobial elastomeric articles
AT513858B1 (de) 2013-01-25 2014-08-15 Sealife Pharma Gmbh Neue bioaktive Polymere
AT516070B1 (de) 2014-07-31 2016-08-15 Sealife Pharma Gmbh Verfahren zur Herstellung von Polyguanidinen

Patent Citations (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH07145063A (ja) * 1993-07-28 1995-06-06 Johnson & Johnson Consumer Prod Inc 殺精子・抗ウイルス性潤滑剤組成物およびその使用方法
JP2006520329A (ja) * 2003-03-20 2006-09-07 ゲオファルマ プロドゥクツィオンスゲーエムベーハー 抗菌作用を有し、ジアミンをベースとするグアニジン誘導体
US20080051740A1 (en) * 2006-06-16 2008-02-28 Family Health International Vaginal drug delivery system and method
WO2008031105A1 (en) * 2006-09-08 2008-03-13 Delaval Holdings Ab Polymeric guanidine salt-based germicides
JP2010507721A (ja) * 2006-10-23 2010-03-11 アーチ・ケミカルズ・インコーポレーテッド 末端アミンの少ないビグアニド組成物
US20110269936A1 (en) * 2009-10-08 2011-11-03 Viktor Veniaminovich Tets Method for Producing Biocidal Polyguanidine, and Biocidal Polyguanidine
WO2015074730A1 (de) * 2013-11-21 2015-05-28 Farco-Pharma Gmbh Zusammensetzung, insbesondere in form eines gleitgels enthaltend ein lokalanästhetikum und polyhexanid
JP2017088603A (ja) * 2015-11-12 2017-05-25 グロック・ヘルス・サイエンス・アンド・リサーチ・ゲゼルシャフト・ミト・ベシュレンクテル・ハフツング 膣炎の治療

Also Published As

Publication number Publication date
WO2019154983A1 (de) 2019-08-15
EP3749095A1 (de) 2020-12-16
EP3524055A1 (de) 2019-08-14
CN111787802A (zh) 2020-10-16
BR112020015955A2 (pt) 2020-12-15
RU2020129407A (ru) 2022-03-09
MX2020008140A (es) 2020-10-12
US20210038637A1 (en) 2021-02-11
KR20200119829A (ko) 2020-10-20

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