JP2021512140A5 - - Google Patents

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Publication number
JP2021512140A5
JP2021512140A5 JP2020558858A JP2020558858A JP2021512140A5 JP 2021512140 A5 JP2021512140 A5 JP 2021512140A5 JP 2020558858 A JP2020558858 A JP 2020558858A JP 2020558858 A JP2020558858 A JP 2020558858A JP 2021512140 A5 JP2021512140 A5 JP 2021512140A5
Authority
JP
Japan
Prior art keywords
pharmaceutically acceptable
acceptable salt
methoxyquinoline
ethylpiperazine
methylureido
Prior art date
Application number
JP2020558858A
Other languages
English (en)
Japanese (ja)
Other versions
JPWO2019139977A5 (https=
JP7352569B2 (ja
JP2021512140A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2019/012886 external-priority patent/WO2019139977A1/en
Publication of JP2021512140A publication Critical patent/JP2021512140A/ja
Publication of JPWO2019139977A5 publication Critical patent/JPWO2019139977A5/ja
Publication of JP2021512140A5 publication Critical patent/JP2021512140A5/ja
Priority to JP2023149903A priority Critical patent/JP7665700B2/ja
Application granted granted Critical
Publication of JP7352569B2 publication Critical patent/JP7352569B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2020558858A 2018-01-10 2019-01-09 肝細胞癌の治療のための併用療法 Active JP7352569B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2023149903A JP7665700B2 (ja) 2018-01-10 2023-09-15 肝細胞癌の治療のための併用療法

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201862615848P 2018-01-10 2018-01-10
US62/615,848 2018-01-10
PCT/US2019/012886 WO2019139977A1 (en) 2018-01-10 2019-01-09 Combination therapies for the treatment of hepatocellular carcinoma

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2023149903A Division JP7665700B2 (ja) 2018-01-10 2023-09-15 肝細胞癌の治療のための併用療法

Publications (4)

Publication Number Publication Date
JP2021512140A JP2021512140A (ja) 2021-05-13
JPWO2019139977A5 JPWO2019139977A5 (https=) 2022-01-18
JP2021512140A5 true JP2021512140A5 (https=) 2022-01-18
JP7352569B2 JP7352569B2 (ja) 2023-09-28

Family

ID=65411938

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2020558858A Active JP7352569B2 (ja) 2018-01-10 2019-01-09 肝細胞癌の治療のための併用療法
JP2023149903A Active JP7665700B2 (ja) 2018-01-10 2023-09-15 肝細胞癌の治療のための併用療法

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2023149903A Active JP7665700B2 (ja) 2018-01-10 2023-09-15 肝細胞癌の治療のための併用療法

Country Status (13)

Country Link
US (1) US11833119B2 (https=)
EP (2) EP3737377B1 (https=)
JP (2) JP7352569B2 (https=)
KR (2) KR102811519B1 (https=)
CN (1) CN111787922A (https=)
AU (1) AU2019206480A1 (https=)
BR (1) BR112020014112A2 (https=)
CA (1) CA3088292A1 (https=)
IL (1) IL275981A (https=)
MA (1) MA51570A (https=)
MX (1) MX2020007375A (https=)
SG (1) SG11202006617RA (https=)
WO (1) WO2019139977A1 (https=)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2023533903A (ja) * 2020-05-15 2023-08-07 エーザイ・アール・アンド・ディー・マネジメント株式会社 Fgfr4阻害剤の経口製剤によるがんの治療方法
CN117479958A (zh) * 2022-05-30 2024-01-30 石药集团中奇制药技术(石家庄)有限公司 用于治疗癌症的药物组合和药物组合物

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE60137273D1 (de) 2000-10-20 2009-02-12 Eisai R&D Man Co Ltd Verfahren zur Herstellung von 4-Phenoxy chinolin Derivaten
PL1698623T3 (pl) 2003-12-25 2015-08-31 Eisai R&D Man Co Ltd Postać krystaliczna soli 4-(3-chloro-4-(cyklopropyloaminokarbonylo)aminofenoksy)-7-metoksy-6-chinolinokarboksamidu lub jej solwatu i sposoby ich wytwarzania
RU2448708C3 (ru) 2006-05-18 2017-09-28 Эйсай Ар Энд Ди Менеджмент Ко., Лтд. Противоопухолевое средство против рака щитовидной железы
KR101513326B1 (ko) 2007-11-09 2015-04-17 에자이 알앤드디 매니지먼트 가부시키가이샤 혈관 신생 저해 물질과 항종양성 백금 착물의 병용
JP2015505562A (ja) * 2012-01-31 2015-02-23 ノバルティス アーゲー Rtk阻害剤と抗エストロゲン剤との組合せ、およびがん治療のためのその使用
KR102265952B1 (ko) 2013-06-26 2021-06-16 에자이 알앤드디 매니지먼트 가부시키가이샤 암 치료 병용요법으로서 에리불린 및 렌바티닙의 용도
MX378288B (es) 2013-10-18 2025-03-10 Eisai R&D Man Co Ltd Inhibidores de pirimidina del fgfr4.
MX373150B (es) * 2014-03-26 2020-04-21 Astex Therapeutics Ltd Combinaciones de un inhibidor del factor de crecimiento de fibroblasto (fgfr) y un inhibidor del receptor del factor de crecimiento 1 similar a insulina (igf1r).
US20160089365A1 (en) * 2014-09-25 2016-03-31 Eisai R&D Management Co., Ltd. Immunostimulatory compound
SG10201810057UA (en) 2015-04-14 2018-12-28 Eisai R&D Man Co Ltd Crystalline fgfr4 inhibitor compound and uses thereof
CN107304188A (zh) * 2016-04-20 2017-10-31 成都融科博海科技有限公司 一种氘代激酶选择性抑制剂及其应用
EP3454898B1 (en) * 2016-05-10 2021-11-10 Eisai R&D Management Co., Ltd. Drug combinations for reducing cell viability and/or cell proliferation

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